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Volumn , Issue 11, 2008, Pages 1839-1850

Synthetic strategies for oseltamivir phosphate

Author keywords

Analogue synthesis; Asymmetric catalysis; Influenza; Oseltamivir phosphate; Process chemistry; Tamiflu

Indexed keywords


EID: 46849088854     PISSN: 1434193X     EISSN: 10990690     Source Type: Journal    
DOI: 10.1002/ejoc.200800033     Document Type: Short Survey
Times cited : (126)

References (56)
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    • For a recent review on the synthesis of 6, see: V. Farina, J. D. Brown, Angew. Chem. Int. Ed. 2006, 45, 7330-7334.
    • b) For a recent review on the synthesis of 6, see: V. Farina, J. D. Brown, Angew. Chem. Int. Ed. 2006, 45, 7330-7334.
  • 13
    • 0035937274 scopus 로고    scopus 로고
    • For an azide-free route using allylamine, see
    • b) For an azide-free route using allylamine, see: M. Karpf, R. Trussardi, J. Org. Chem. 2001, 66, 2044-2051.
    • (2001) J. Org. Chem , vol.66 , pp. 2044-2051
    • Karpf, M.1    Trussardi, R.2
  • 17
    • 34548827964 scopus 로고    scopus 로고
    • The conversion from 53 to 56 is an improved method in relation to the original report in ref. [9], see: Y.-Y. Yeung, E. J. Corey, Tetrahedron Lett. 2007, 48, 7567-7570.
    • The conversion from 53 to 56 is an improved method in relation to the original report in ref. [9], see: Y.-Y. Yeung, E. J. Corey, Tetrahedron Lett. 2007, 48, 7567-7570.
  • 20
    • 0033581774 scopus 로고    scopus 로고
    • For other examples of catalytic asymmetric aziridine-opening reactions with nitrogen nucleophiles, see: a
    • For other examples of catalytic asymmetric aziridine-opening reactions with nitrogen nucleophiles, see: a) Z. Li, M. Fernández, E. N. Jacobsen, Org. Lett. 1999, 1, 1611-1613;
    • (1999) Org. Lett , vol.1 , pp. 1611-1613
    • Li, Z.1    Fernández, M.2    Jacobsen, E.N.3
  • 22
    • 21544444468 scopus 로고    scopus 로고
    • For reviews of the utility of asymmetric catalysts derived from ligand 67, see: a M. Kanai, N. Kato, E. Ichikawa, M. Shibasaki, Synlett 2005, 1491-1508;
    • For reviews of the utility of asymmetric catalysts derived from ligand 67, see: a) M. Kanai, N. Kato, E. Ichikawa, M. Shibasaki, Synlett 2005, 1491-1508;
  • 30
    • 38149121471 scopus 로고    scopus 로고
    • The conversion from 74 to 6 is an improved method in relation to the original report in ref.[13] See: M. Morita, T. Sone, K. Yamatsugu, Y. Sohtome, S. Matsunaga, M. Kanai, Y. Watanabe, M. Shibasaki, Bioorg. Med. Chem. Lett. 2008, 18, 600-602.
    • The conversion from 74 to 6 is an improved method in relation to the original report in ref.[13] See: M. Morita, T. Sone, K. Yamatsugu, Y. Sohtome, S. Matsunaga, M. Kanai, Y. Watanabe, M. Shibasaki, Bioorg. Med. Chem. Lett. 2008, 18, 600-602.
  • 39
    • 34548847746 scopus 로고    scopus 로고
    • For references relating to the effects of oseltamivir on the nervous system, see: a
    • For references relating to the effects of oseltamivir on the nervous system, see: a) Y. Izumi, K. Tokuda, K. A. O'Dell, C. F. Zorumski, T. Narahashi, Neurosci. Lett. 2007, 426, 54-58;
    • (2007) Neurosci. Lett , vol.426 , pp. 54-58
    • Izumi, Y.1    Tokuda, K.2    O'Dell, K.A.3    Zorumski, C.F.4    Narahashi, T.5
  • 48
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    • Our studies indicated that the introduction of a 3-pentyl group at the C-3 oxygen in compounds related to 100 (containing C-4-acetamide and C-1-ester functions) was impossible Y. Kimura, K. Yamatsugu, M. Kanai, M. Shibasaki, unpublished results
    • Our studies indicated that the introduction of a 3-pentyl group at the C-3 oxygen in compounds related to 100 (containing C-4-acetamide and C-1-ester functions) was impossible (Y. Kimura, K. Yamatsugu, M. Kanai, M. Shibasaki, unpublished results).


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.