Structure-activity relationships of the dimeric analogues of endomorphin-2 with different lengths of spacers

Protein and Peptide Letters

Volumn 15, Issue 3, 2008, Pages 275-279

  Gao, Yan Feng ^a   Zhai, Ming Xia ^a   Liu, Wei Xia ^b   Liu, Xin ^b   Yuan, Ye ^b   Qi, Yuan Ming ^a   Wang, Rui ^b  

^a ZHENGZHOU UNIVERSITY   (China)

^b LANZHOU UNIVERSITY   (China)

Author keywords

Analogue; Balanced agonist; Dimerization; Endomorphin 2; Opioid receptor; Structure activity relationships

Indexed keywords

DELTA OPIATE RECEPTOR; ENDOMORPHIN 2; NARCOTIC ANALGESIC AGENT; OLIGOPEPTIDE;

ANIMAL; ARTICLE; BINDING SITE; CHEMISTRY; GUINEA PIG; MALE; METABOLISM; MOUSE; RAT; STRUCTURE ACTIVITY RELATION; WISTAR RAT;

ANALGESICS, OPIOID; ANIMALS; BINDING SITES; GUINEA PIGS; MALE; MICE; OLIGOPEPTIDES; RATS; RATS, WISTAR; RECEPTORS, OPIOID, DELTA; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 41449106914     PISSN: 09298665     EISSN: None     Source Type: Journal    
DOI: 10.2174/092986608783744199     Document Type: Article

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