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Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 7, 2005, Pages 1847-1850

Structure-activity relationship of the novel bivalent and C-terminal modified analogues of endomorphin-2

(6) Gao, Yanfeng a Liu, Xin a Wei, Jie a Zhu, Beibei a Chen, Qiang a Wang, Rui a,b

a LANZHOU UNIVERSITY (China)

b LANZHOU INSTITUTE OF CHEMICAL PHYSICS (China)

Author keywords

Dimerization; Endomorphin 2; Modification; Opioid peptide; Structure activity relationship

Indexed keywords

ENDOMORPHIN 2; MU OPIATE RECEPTOR;

ANALGESIC ACTIVITY; ARTICLE; CARBOXY TERMINAL SEQUENCE; CHEMICAL MODIFICATION; DIMERIZATION; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; IC 50; PHARMACOPHORE; RECEPTOR AFFINITY; STRUCTURE ACTIVITY RELATION;

EID: 15044364083 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2005.02.021 Document Type: Article

Times cited : (25)

References (27)

1
- 0035840823
- R. Przewlocki, and B. Przewlocka Eur. J. Pharmacol. 429 2001 79 91
- (2001) Eur. J. Pharmacol. , vol.429 , pp. 79-91
- Przewlocki, R.¹ Przewlocka, B.²

2
- 0035064736
- M. Narita, M. Funada, and T. Suzuki Pharmacol. Ther. 89 2001 1 15
- (2001) Pharmacol. Ther. , vol.89 , pp. 1-15
- Narita, M.¹ Funada, M.² Suzuki, T.³

3
- 2942705905
- J. Fichna, Jean-Claude do-Rego, J. Costentin, N.N. Chung, P.W. Schiller, P. Kosson, and A. Janecka Biochem. Biophys. Res. Commun. 320 2004 531 536
- (2004) Biochem. Biophys. Res. Commun. , vol.320 , pp. 531-536
- Fichna, J.¹ Do-Rego, J.-C.² Costentin, J.³ Chung, N.N.⁴ Schiller, P.W.⁵ Kosson, P.⁶ Janecka, A.⁷

4
- 0033588946
- A.W. Lipkowski, A. Misicka, P. Davis, D. Stropova, J. Janders, M. Lachwa, F. Porreca, H.I. Yamamura, and V.J. Hruby Bioorg. Med. Chem. Lett. 9 1999 2763 2766
- (1999) Bioorg. Med. Chem. Lett. , vol.9 , pp. 2763-2766
- Lipkowski, A.W.¹ Misicka, A.² Davis, P.³ Stropova, D.⁴ Janders, J.⁵ Lachwa, M.⁶ Porreca, F.⁷ Yamamura, H.I.⁸ Hruby, V.J.⁹

5
- 0020414774
- A.W. Lipkowski, A.M. Konecka, and I. Sroczynska Peptides 3 1982 697 700
- (1982) Peptides , vol.3 , pp. 697-700
- Lipkowski, A.W.¹ Konecka, A.M.² Sroczynska, I.³

6
- 0035919718
- M. Yamazaki, T. Suzuki, M. Narita, and A.W. Lipkowski Life Sci. 69 2001 1023 1028
- (2001) Life Sci. , vol.69 , pp. 1023-1028
- Yamazaki, M.¹ Suzuki, T.² Narita, M.³ Lipkowski, A.W.⁴

7
- 0031763418
- R.D. Egleton, T.J. Abbruscato, S.A. Thomas, and T.P. Davis J. Pharm. Sci. 87 1998 1433 1439
- (1998) J. Pharm. Sci. , vol.87 , pp. 1433-1439
- Egleton, R.D.¹ Abbruscato, T.J.² Thomas, S.A.³ Davis, T.P.⁴

8
- 0030933655
- J.E. Zadina, L. Hackler, L.J. Ge, and A.J. Kastin Nature 386 1997 499 502
- (1997) Nature , vol.386 , pp. 499-502
- Zadina, J.E.¹ Hackler, L.² Ge, L.J.³ Kastin, A.J.⁴

9
- 0031426851
- L. Hackler, J.E. Zadina, L.J. Ge, and A.J. Kastin Peptides 18 1997 1635 1639
- (1997) Peptides , vol.18 , pp. 1635-1639
- Hackler, L.¹ Zadina, J.E.² Ge, L.J.³ Kastin, A.J.⁴

10
- 0032893243
- S. Sakurada, J.E. Zadina, A.J. Kastin, S. Katsuyama, T. Fujimura, K. Murayama, M. Yuki, H. Ueda, and T. Sakurada Eur. J. Pharmacol. 372 1999 25 30
- (1999) Eur. J. Pharmacol. , vol.372 , pp. 25-30
- Sakurada, S.¹ Zadina, J.E.² Kastin, A.J.³ Katsuyama, S.⁴ Fujimura, T.⁵ Murayama, K.⁶ Yuki, M.⁷ Ueda, H.⁸ Sakurada, T.⁹

11
- 18444361816
- I. Lengyel, G. Orosz, D. Biyashev, L. Kocsis, M. Al-Khrasani, A.Z. Ronai, C. Tomboly, Z. Furst, G. Toth, and A. Borsodi Biochem. Biophys. Res. Commun. 290 2002 153 161
- (2002) Biochem. Biophys. Res. Commun. , vol.290 , pp. 153-161
- Lengyel, I.¹ Orosz, G.² Biyashev, D.³ Kocsis, L.⁴ Al-Khrasani, M.⁵ Ronai, A.Z.⁶ Tomboly, C.⁷ Furst, Z.⁸ Toth, G.⁹ Borsodi, A.¹⁰

12
- 3042599035
- Y. Fujita, Y. Tsuda, T.Y. Li, T. Motoyama, M. Takahashi, Y. Shimizu, T. Yokoi, Y. Sasaki, A. Ambo, A. Kita, Y. Jinsmaa, S.D. Bryant, L.H. Lazarus, and Y. Okada J. Med. Chem. 47 2004 3591 3599
- (2004) J. Med. Chem. , vol.47 , pp. 3591-3599
- Fujita, Y.¹ Tsuda, Y.² Li, T.Y.³ Motoyama, T.⁴ Takahashi, M.⁵ Shimizu, Y.⁶ Yokoi, T.⁷ Sasaki, Y.⁸ Ambo, A.⁹ Kita, A.¹⁰ Jinsmaa, Y.¹¹ Bryant, S.D.¹² Lazarus, L.H.¹³ Okada, Y.¹⁴

13
- 0037356635
- Y. Sasaki, A. Sasaki, H. Niizuma, H. Goto, and A. Ambo Bioorg. Med. Chem. 11 2003 675 678
- (2003) Bioorg. Med. Chem. , vol.11 , pp. 675-678
- Sasaki, Y.¹ Sasaki, A.² Niizuma, H.³ Goto, H.⁴ Ambo, A.⁵

14
- 0037401355
- Y. Okada, Y. Fujita, T. Motoyama, Y. Tsuda, T. Yokoi, T.Y. Li, Y. Sasaki, A. Ambo, Y. Jinsmaa, S.D. Bryant, and L.H. Lazarus Bioorg. Med. Chem. 11 2003 1983 1994
- (2003) Bioorg. Med. Chem. , vol.11 , pp. 1983-1994
- Okada, Y.¹ Fujita, Y.² Motoyama, T.³ Tsuda, Y.⁴ Yokoi, T.⁵ Li, T.Y.⁶ Sasaki, Y.⁷ Ambo, A.⁸ Jinsmaa, Y.⁹ Bryant, S.D.¹⁰ Lazarus, L.H.¹¹

15
- 4744353375
- G. Cardillo, L. Gentilucci, A. Tolomelli, R. Spinosa, M. Calienni, A.R. Qasem, and S. Spampinato J. Med. Chem. 47 2004 5198 6203
- (2004) J. Med. Chem. , vol.47 , pp. 5198-6203
- Cardillo, G.¹ Gentilucci, L.² Tolomelli, A.³ Spinosa, R.⁴ Calienni, M.⁵ Qasem, A.R.⁶ Spampinato, S.⁷

16
- 9144253110
- C. Tomboly, K.E. Kover, A. Peter, D. Tourwe, D. Biyashev, S. Benyhe, A. Borsodi, M. Al-Khrasani, A.Z. Ronai, and G. Toth J. Med. Chem. 47 2004 735 743
- (2004) J. Med. Chem. , vol.47 , pp. 735-743
- Tomboly, C.¹ Kover, K.E.² Peter, A.³ Tourwe, D.⁴ Biyashev, D.⁵ Benyhe, S.⁶ Borsodi, A.⁷ Al-Khrasani, M.⁸ Ronai, A.Z.⁹ Toth, G.¹⁰

17
- 0035829437
- M. Keller, C. Boissard, L. Patiny, N.N. Chung, C. Lemieux, M. Mutter, and P.W. Schiller J. Med. Chem. 44 2001 3896 3903
- (2001) J. Med. Chem. , vol.44 , pp. 3896-3903
- Keller, M.¹ Boissard, C.² Patiny, L.³ Chung, N.N.⁴ Lemieux, C.⁵ Mutter, M.⁶ Schiller, P.W.⁷

18
- 0037468538
- B.A. Harrison, G.W. Pasternak, and G.L. Verdine J. Med. Chem. 46 2003 677 680
- (2003) J. Med. Chem. , vol.46 , pp. 677-680
- Harrison, B.A.¹ Pasternak, G.W.² Verdine, G.L.³

19
- 0038204635
- Z.J. Shi, B.A. Harrison, and G.L. Verdine Org. Lett. 5 2003 633 636
- (2003) Org. Lett. , vol.5 , pp. 633-636
- Shi, Z.J.¹ Harrison, B.A.² Verdine, G.L.³

20
- 0037073163
- B.A. Harrison, T.M. Gierasch, C. Neilan, G.W. Pasternak, and G.L. Verdine J. Am. Chem. Soc. 124 2002 13352 13353
- (2002) J. Am. Chem. Soc. , vol.124 , pp. 13352-13353
- Harrison, B.A.¹ Gierasch, T.M.² Neilan, C.³ Pasternak, G.W.⁴ Verdine, G.L.⁵

21
- 0025901024
- L.H. Lazarus, S. Salvadori, R. Tomatis, and W.E. Wilson Biochem. Biophys. Res. Commun. 178 1991 110 115
- (1991) Biochem. Biophys. Res. Commun. , vol.178 , pp. 110-115
- Lazarus, L.H.¹ Salvadori, S.² Tomatis, R.³ Wilson, W.E.⁴

22
- 0036201028
- J.L. Flippen-Anderson, J.R. Deschamps, C. George, V.J. Hruby, A. Misicka, and A.W. Lipkowski J. Pept. Res. 59 2002 123 133
- (2002) J. Pept. Res. , vol.59 , pp. 123-133
- Flippen-Anderson, J.L.¹ Deschamps, J.R.² George, C.³ Hruby, V.J.⁴ Misicka, A.⁵ Lipkowski, A.W.⁶

23
- 0032477944
- G.G. Li, W. Haq, L. Xiang, Bih-Show. Lou, R. Hughes, I.A. De Leon, P. Davis, T.J. Gillespie, M. Romanowski, X.Y. Zhu, A. Misicka, A.W. Lipkowski, F. Porreca, T.P. Davis, H.I. Yamamura, D.F. O'Brien, and V.J. Hruby Bioorg. Med. Chem. Lett. 8 1998 555 560
- (1998) Bioorg. Med. Chem. Lett. , vol.8 , pp. 555-560
- Li, G.G.¹ Haq, W.² Xiang, L.³ Lou, Bih-Show.⁴ Hughes, R.⁵ De Leon, I.A.⁶ Davis, P.⁷ Gillespie, T.J.⁸ Romanowski, M.⁹ Zhu, X.Y.¹⁰ Misicka, A.¹¹ Lipkowski, A.W.¹² Porreca, F.¹³ Davis, T.P.¹⁴ Yamamura, H.I.¹⁵ O'Brien, D.F.¹⁶ Hruby, V.J.¹⁷

24
- 0038155285
- Y. Okada, Y. Tsuda, Y. Fujita, T. Yokoi, Y. Sasaki, A. Ambo, R. Konishi, M. Nagata, S. Salvadori, Y. Jinsmaa, S.D. Bryant, and L.H. Lazarus J. Med. Chem. 46 2003 3201 3209
- (2003) J. Med. Chem. , vol.46 , pp. 3201-3209
- Okada, Y.¹ Tsuda, Y.² Fujita, Y.³ Yokoi, T.⁴ Sasaki, Y.⁵ Ambo, A.⁶ Konishi, R.⁷ Nagata, M.⁸ Salvadori, S.⁹ Jinsmaa, Y.¹⁰ Bryant, S.D.¹¹ Lazarus, L.H.¹²

25
- 0015861774
- Y.C. Cheng, and W.H. Prusoff Biochem. Pharmacol. 22 1973 3099 3108
- (1973) Biochem. Pharmacol. , vol.22 , pp. 3099-3108
- Cheng, Y.C.¹ Prusoff, W.H.²

26
- 0000440578
- H.I. Mosberg, R. Hurst, V.J. Hruby, K. Gee, H.I. Yamamura, J.J. Galligan, and T.F. Burks Proc. Natl. Acad. Sci. U.S.A. 80 1983 5871 5874
- (1983) Proc. Natl. Acad. Sci. U.S.A. , vol.80 , pp. 5871-5874
- Mosberg, H.I.¹ Hurst, R.² Hruby, V.J.³ Gee, K.⁴ Yamamura, H.I.⁵ Galligan, J.J.⁶ Burks, T.F.⁷

27
- 0021970967
- T. Costa, M. Wuster, A. Herz, Y. Shimohigashi, H.C. Chen, and D. Rodbard Biochem. Pharmacol. 34 1985 25 30
- (1985) Biochem. Pharmacol. , vol.34 , pp. 25-30
- Costa, T.¹ Wuster, M.² Herz, A.³ Shimohigashi, Y.⁴ Chen, H.C.⁵ Rodbard, D.⁶

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