Subtype-selective noncompetitive or competitive inhibition of human α1-adrenergic receptors by ρ-TIA

Journal of Biological Chemistry

Volumn 279, Issue 34, 2004, Pages 35326-35333

  Chen, Zhongjian ^a   Rogge, George ^a   Hague, Chris ^a   Alewood, Dianne ^b   Colless, Barbara ^b   Lewis, Richard J ^b   Minneman, Kenneth P ^a  

^a EMORY UNIVERSITY SCHOOL OF MEDICINE   (United States)

^b Xenome Ltd   (Australia)

Author keywords

[No Author keywords available]

Indexed keywords

ALCOHOLS; BIOCHEMISTRY; CELLS; LIVING SYSTEMS STUDIES; MUTAGENESIS; PHOSPHATES; PROTEINS;

ALANINE-SCANNING MUTAGENESIS; PEPTIDE LIGANDS;

AMINO ACIDS;

ALANINE; ALPHA 1 ADRENERGIC RECEPTOR; ALPHA 1A ADRENERGIC RECEPTOR; ALPHA 1B ADRENERGIC RECEPTOR; ALPHA 1D ADRENERGIC RECEPTOR; INOSITOL PHOSPHATE; ISOLEUCINE; MUTANT PROTEIN; NORADRENALIN; PEPTIDE; RADIOLIGAND; RECEPTOR SUBTYPE; RECOMBINANT PROTEIN; RHO FACTOR; RHO TIA PEPTIDE; UNCLASSIFIED DRUG;

AMINO TERMINAL SEQUENCE; ARTICLE; BINDING SITE; CELL LINE; CELL STRAIN HEK293; COMPETITIVE INHIBITION; HAMSTER; HUMAN; HUMAN CELL; INCUBATION TIME; LIGAND BINDING; MOLECULAR INTERACTION; MUTAGENESIS; NONCOMPETITIVE INHIBITION; NONHUMAN; PRIORITY JOURNAL; RECEPTOR AFFINITY; RECEPTOR DOWN REGULATION;

ANIMALS; BINDING SITES; BINDING, COMPETITIVE; CARRIER PROTEINS; CONOTOXINS; CRICETINAE; HUMANS; ISOLEUCINE; RADIOLIGAND ASSAY; RECEPTORS, ADRENERGIC, ALPHA-1;

CRICETINAE;

EID: 4143122196     PISSN: 00219258     EISSN: None     Source Type: Journal    
DOI: 10.1074/jbc.M403703200     Document Type: Article

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