Binding, partial agonism, and potentiation of α1-adrenergic receptor function by benzodiazepines: A potential site of allosteric modulation

Journal of Pharmacology and Experimental Therapeutics

Volumn 291, Issue 3, 1999, Pages 1164-1171

  Waugh, David J J ^a   Gaivin, Robert J ^a   Damron, Derek S ^a   Murray, Paul A ^a   Perez, Dianne M ^a  

^a LERNER RESEARCH INSTITUTE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

4 AMINOBUTYRIC ACID A RECEPTOR; ADRENALIN; ALPHA 1 ADRENERGIC RECEPTOR BLOCKING AGENT; BENZODIAZEPINE; CLONIDINE; DIAZEPAM; FLUNITRAZEPAM; LORAZEPAM; METHOXAMINE; MIDAZOLAM; MUSCIMOL; N SEC BUTYL 1 (2 CHLOROPHENYL) N METHYL 3 ISOQUINOLINECARBOXAMIDE; PHENYLEPHRINE; PRAZOSIN; RECEPTOR SUBTYPE;

ADRENERGIC SYSTEM; ANIMAL CELL; ARTICLE; BINDING SITE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; FIBROBLAST CULTURE; LIGAND BINDING; NONHUMAN; PRIORITY JOURNAL; RAT; SIGNAL TRANSDUCTION; VASCULAR RESISTANCE; VASCULAR SMOOTH MUSCLE;

ADRENERGIC ALPHA-AGONISTS; ADRENERGIC ALPHA-ANTAGONISTS; ANIMALS; BENZODIAZEPINES; CELL MEMBRANE; CELLS, CULTURED; COS CELLS; DRUG SYNERGISM; EPINEPHRINE; FIBROBLASTS; INOSITOL PHOSPHATES; LIGANDS; MOLECULAR CONFORMATION; PHENYLEPHRINE; RADIOLIGAND ASSAY; RATS; RECEPTORS, ADRENERGIC, ALPHA-1; SIGNAL TRANSDUCTION; TRANSFECTION;

EID: 0032705772     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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