메뉴 건너뛰기




Volumn 39, Issue 1, 1996, Pages 54-107

α1 Adrenoceptor subtypes: A synopsis of their pharmacology and molecular biology

Author keywords

Adrenergic agonists; Adrenergic antagonists; Receptors, adrenergic, 1; Receptors, catecholamine; Sympathomimetics

Indexed keywords

1 (4 AMINO 6,7 DIMETHOXY 2 QUINAZOLINYL) 4 (BICYCLO[2.2.2]OCTA 2,5 DIEN 2 YLCARBONYL)PIPERAZINE; 5 METHYLURAPIDIL; ABANOQUIL; ADRENERGIC RECEPTOR BLOCKING AGENT; ADRENERGIC RECEPTOR STIMULATING AGENT; ALFUZOSIN; ALPHA 1 ADRENERGIC RECEPTOR; BENEXTRAMINE; CHLOROETHYLCLONIDINE; CYCLAZOCINE; DOXAZOSIN; NIFEDIPINE; PHENOXYBENZAMINE; PHENYLEPHRINE; PRAZOSIN; RECEPTOR SUBTYPE; TERAZOSIN;

EID: 0030497401     PISSN: 02724391     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1098-2299(19960901)39:1<54::AID-DDR7>3.0.CO;2-J     Document Type: Review
Times cited : (70)

References (376)
  • 2
    • 0027509730 scopus 로고
    • 1-adrenoceptor mediating contractions of rat aorta, vas deferens and spleen
    • 1-adrenoceptor mediating contractions of rat aorta, vas deferens and spleen. Br J Pharmacol 109:80-87.
    • (1993) Br J Pharmacol , vol.109 , pp. 80-87
    • Aboud, R.1    Shafii, M.2    Docherty, J.R.3
  • 3
    • 0029098058 scopus 로고
    • 1c-adrenoceptor antagonist: A randomized, controlled trial in patients with benign prostatic "obstruction" (symptomatic BPH)
    • 1c-adrenoceptor antagonist: A randomized, controlled trial in patients with benign prostatic "obstruction" (symptomatic BPH). Br J Urol 76:325-336.
    • (1995) Br J Urol , vol.76 , pp. 325-336
    • Abrams, P.1    Schulman, C.C.2    Vaage, S.3
  • 4
    • 84951653316 scopus 로고
    • A study of the adrenotropic receptors
    • Ahlquist RP (1948): A study of the adrenotropic receptors. Am J Physiol 153:586-600.
    • (1948) Am J Physiol , vol.153 , pp. 586-600
    • Ahlquist, R.P.1
  • 5
    • 0029965503 scopus 로고    scopus 로고
    • Binding and competitive inhibition of amine uptake at postsynaptic neurones (transport-P) by tricyclic antidepressants
    • Al-Damluji S, Kopin IJ (1996): Binding and competitive inhibition of amine uptake at postsynaptic neurones (transport-P) by tricyclic antidepressants. Br J Pharmacol 117:811-816.
    • (1996) Br J Pharmacol , vol.117 , pp. 811-816
    • Al-Damluji, S.1    Kopin, I.J.2
  • 6
    • 0027501903 scopus 로고
    • Pharmacology of lower urinary tract smooth muscles and penile erectile tissues
    • Andersson K-E (1993): Pharmacology of lower urinary tract smooth muscles and penile erectile tissues. Pharmacol Rev 45:253-308.
    • (1993) Pharmacol Rev , vol.45 , pp. 253-308
    • Andersson, K.-E.1
  • 7
    • 0028985753 scopus 로고
    • Alphal adrenergic receptor blockade in the male lower urinary tract and other body systems
    • Andersson K-E (1994): Alphal adrenergic receptor blockade in the male lower urinary tract and other body systems. Scand J Urol Nephrol 29:13-20.
    • (1994) Scand J Urol Nephrol , vol.29 , pp. 13-20
    • Andersson, K.-E.1
  • 8
    • 12644272798 scopus 로고    scopus 로고
    • Pharma Projects
    • Anonymous (1996a): NS-49, Urological. Pharma Projects, m 1577.
    • (1996) NS-49, Urological , pp. 1577
  • 9
    • 12644291204 scopus 로고    scopus 로고
    • Recordati's urologicals disappoint
    • Anonymous (1996b): Recordati's urologicals disappoint. Scrip 2129:25.
    • (1996) Scrip , vol.2129 , pp. 25
  • 10
    • 0023731352 scopus 로고
    • Investigations into the mechanism of the anti-hypertensive effect of SGB-1534, a novel ocpadrenoceptor antagonist, in rats
    • Aono J, Sakai K (1988): Investigations into the mechanism of the anti-hypertensive effect of SGB-1534, a novel ocpadrenoceptor antagonist, in rats. Jap J Pharmacol 48:229-239.
    • (1988) Jap J Pharmacol , vol.48 , pp. 229-239
    • Aono, J.1    Sakai, K.2
  • 13
    • 0015147450 scopus 로고
    • Synthesis and hypotensive activity of benzamidopiperidylethylindoles
    • Archibald JL, Alps BJ, Cavalla JF, Jackson JL (1971): Synthesis and hypotensive activity of benzamidopiperidylethylindoles. J Med Chem 14:1054-1059.
    • (1971) J Med Chem , vol.14 , pp. 1054-1059
    • Archibald, J.L.1    Alps, B.J.2    Cavalla, J.F.3    Jackson, J.L.4
  • 14
    • 0016158725 scopus 로고
    • Benzainidopiperidines. 2. Heterocyclic compounds related to indoramin
    • Archibald JL, Benke, GA (1974a): Benzainidopiperidines. 2. Heterocyclic compounds related to indoramin. J Med Chem 17:736-739.
    • (1974) J Med Chem , vol.17 , pp. 736-739
    • Archibald, J.L.1    Benke, G.A.2
  • 15
    • 0016197145 scopus 로고
    • Benzamidopiperidines. 3. Carbocyclic derivatives related to indoramin
    • Archibald JL, Fairbrother P, Jackson JL (1974b): Benzamidopiperidines. 3. Carbocyclic derivatives related to indoramin. J Med Chem 17:739-744.
    • (1974) J Med Chem , vol.17 , pp. 739-744
    • Archibald, J.L.1    Fairbrother, P.2    Jackson, J.L.3
  • 16
    • 12644297014 scopus 로고
    • UK-52,046, a novel alphal-adrenoceptor antagonist with antidysrhythmic activity
    • Aubry ML, Davey MJ, Fetch B (1988): UK-52,046, a novel alphal-adrenoceptor antagonist with antidysrhythmic activity. Br J Pharmacol 95 (Suppl):752P.
    • (1988) Br J Pharmacol , vol.95 , Issue.SUPPL.
    • Aubry, M.L.1    Davey, M.J.2    Fetch, B.3
  • 17
  • 18
    • 0028828774 scopus 로고
    • Preliminary observations on the use of midodrine in treating orthostatic hypotension in familial dysautonomia
    • Axelrod FB, Krey L, Glickstein JS, Allison JW, Friedman D (1995): Preliminary observations on the use of midodrine in treating orthostatic hypotension in familial dysautonomia. J Autonom Nerv Sys 55:29-35.
    • (1995) J Autonom Nerv Sys , vol.55 , pp. 29-35
    • Axelrod, F.B.1    Krey, L.2    Glickstein, J.S.3    Allison, J.W.4    Friedman, D.5
  • 19
    • 0025670092 scopus 로고
    • 1-adrenergic receptor subtypes modulate catecholamine-induced increases and decreases in ventricular automaticity
    • 1-adrenergic receptor subtypes modulate catecholamine-induced increases and decreases in ventricular automaticity. Circ Res 67:1535-1551.
    • (1990) Circ Res , vol.67 , pp. 1535-1551
    • Del Balzo, U.1    Rosen, M.R.2    Malfatto, G.3    Kaplan, L.M.4    Steinberg, S.F.5
  • 20
    • 0018381173 scopus 로고
    • Cardiac muscarinic blocking and atropinic blocking effects of a tetramine disulfide with α-adrenoceptor blocking activity
    • Benfey BG, Yong MS, Belleau B, Melchiorre C (1979): Cardiac muscarinic blocking and atropinic blocking effects of a tetramine disulfide with α-adrenoceptor blocking activity. Can J Physiol Pharmacol 57:41-47.
    • (1979) Can J Physiol Pharmacol , vol.57 , pp. 41-47
    • Benfey, B.G.1    Yong, M.S.2    Belleau, B.3    Melchiorre, C.4
  • 21
    • 0029899133 scopus 로고    scopus 로고
    • Use of modafinil in the treatment of narcolepsy: A long-term follow-up-study
    • Besset A, Chetrit M, Carlander B, Billiard M (1996): Use of modafinil in the treatment of narcolepsy: a long-term follow-up-study. Clin Neurophysiol 26:60-66.
    • (1996) Clin Neurophysiol , vol.26 , pp. 60-66
    • Besset, A.1    Chetrit, M.2    Carlander, B.3    Billiard, M.4
  • 25
    • 0023880485 scopus 로고
    • Influence of a receptor reserve on the inhibition by calcium channel blockers of alpha adrenoceptor-mediated responses in rat isolated vascular tissues
    • Bognar IT, Enero MA (1988): Influence of a receptor reserve on the inhibition by calcium channel blockers of alpha adrenoceptor-mediated responses in rat isolated vascular tissues. J Pharmacol Exp Ther 245:673-681.
    • (1988) J Pharmacol Exp Ther , vol.245 , pp. 673-681
    • Bognar, I.T.1    Enero, M.A.2
  • 27
    • 0023874865 scopus 로고
    • Resolution and pharmacological properties of the enantiomers of the potent α-adrenoceptor antagonist l-[2-ethoxy-2-(3′-pyridyl)ethyl]-4-(2′-methoxy-phenyl)piperazine
    • Bonacchi G, Agostini O, Fedi M, Bacciarelli C, Boni P, Castellucci A, Perretti F, Manzini S (1988): Resolution and pharmacological properties of the enantiomers of the potent α-adrenoceptor antagonist l-[2-ethoxy-2-(3′-pyridyl)ethyl]-4-(2′-methoxy-phenyl)piperazine. Arzneim-Forsch/Drug Res 38:650-654.
    • (1988) Arzneim-Forsch/Drug Res , vol.38 , pp. 650-654
    • Bonacchi, G.1    Agostini, O.2    Fedi, M.3    Bacciarelli, C.4    Boni, P.5    Castellucci, A.6    Perretti, F.7    Manzini, S.8
  • 28
    • 0008619087 scopus 로고
    • The use of phenoxybenzamine to discriminate 5-HT receptors mediating endothelium-dependent and -independent vasorelaxation
    • Browning C, Giles H, Martin GR (1995): The use of phenoxybenzamine to discriminate 5-HT receptors mediating endothelium-dependent and -independent vasorelaxation. Br J Pharmacol 116:262P.
    • (1995) Br J Pharmacol , vol.116
    • Browning, C.1    Giles, H.2    Martin, G.R.3
  • 29
    • 0028961804 scopus 로고
    • Pharmacological antagonism of α-adrenergic agonist induced increases in canine intra-urethral pressure in vivo
    • Brune ME, Buckner SA, Polakowski J, Kerwin JF, Hancock AA (1995): Pharmacological antagonism of α-adrenergic agonist induced increases in canine intra-urethral pressure in vivo. Drug Dev Res 34:267-275.
    • (1995) Drug Dev Res , vol.34 , pp. 267-275
    • Brune, M.E.1    Buckner, S.A.2    Polakowski, J.3    Kerwin, J.F.4    Hancock, A.A.5
  • 34
  • 39
    • 0019226219 scopus 로고
    • Effects of tiodazosin, prazosin, trimazosin and phentolamine on blood pressure, heart rate and on pre- And postsynaptic α-adrenergic receptors in the rat
    • Buyniski JP, Pircio AW, Schurig JE, Campbell JA (1980): Effects of tiodazosin, prazosin, trimazosin and phentolamine on blood pressure, heart rate and on pre- and postsynaptic α-adrenergic receptors in the rat. Clin Exp Hypertens 2:1039-1066.
    • (1980) Clin Exp Hypertens , vol.2 , pp. 1039-1066
    • Buyniski, J.P.1    Pircio, A.W.2    Schurig, J.E.3    Campbell, J.A.4
  • 40
    • 0021992772 scopus 로고
    • Heterogeneity of alpha-2 adrenergic receptors
    • Bylund DB (1985): Heterogeneity of alpha-2 adrenergic receptors. Pharmacol Biochem Behav 22:835-843.
    • (1985) Pharmacol Biochem Behav , vol.22 , pp. 835-843
    • Bylund, D.B.1
  • 41
    • 12644286596 scopus 로고
    • ARC-239 is a selective antagonist at alpha-2B adrenergic receptors
    • Bylund DB, Ray-Prenger C (1987): ARC-239 is a selective antagonist at alpha-2B adrenergic receptors. Fed Proc 46:1445.
    • (1987) Fed Proc , vol.46 , pp. 1445
    • Bylund, D.B.1    Ray-Prenger, C.2
  • 47
    • 0028790561 scopus 로고
    • A Belgian post-marketing study of terazosin for the treatment of benign prostate hypertrophy
    • Gauchie P Croons AM, Hubloux A (1995): A Belgian post-marketing study of terazosin for the treatment of benign prostate hypertrophy. Acta Therapeut 21:257-269.
    • (1995) Acta Therapeut , vol.21 , pp. 257-269
    • Gauchie, P.1    Croons, A.M.2    Hubloux, A.3
  • 49
    • 0028998873 scopus 로고
    • 1-adrenoceptor selectivity?
    • 1-adrenoceptor selectivity? Br J Urology 76 (Suppl 1):47-55.
    • (1995) Br J Urology , vol.76 , Issue.1 SUPPL. , pp. 47-55
    • Chapple, C.R.1
  • 51
    • 0030065315 scopus 로고    scopus 로고
    • 1A-adrenoceptor antagonist: A metaanalysis of two randomized, placebo-controlled, multicentre studies in patients with benign prostatic obstruction (symptomatic BPH)
    • 1A-adrenoceptor antagonist: A metaanalysis of two randomized, placebo-controlled, multicentre studies in patients with benign prostatic obstruction (symptomatic BPH). Eur Urol 29:155-167.
    • (1996) Eur Urol , vol.29 , pp. 155-167
    • Chapple, C.R.1    Wyndaele, J.J.2    Nordling, J.3    Boeminghaus, F.4    Ypma, A.F.G.V.M.5    Abrams, P.6
  • 52
    • 0028971744 scopus 로고
    • 1-adrenoceptor subtypes involved in the antinatriuretic response to intrarenal infusion of phenylephrine
    • 1-adrenoceptor subtypes involved in the antinatriuretic response to intrarenal infusion of phenylephrine. Eur J Pharmacol 287:1-6.
    • (1995) Eur J Pharmacol , vol.287 , pp. 1-6
    • Chen, C.1    Lokhandwala, M.F.2
  • 53
    • 0028839704 scopus 로고
    • Bioactive constituents from the flower buds and peduncles of Lindera megaphylla
    • Chen CC, Lin CE Huang YL, Ko FN, Teng, CM (1995): Bioactive constituents from the flower buds and peduncles of Lindera megaphylla. J Natural Prod 58:1423-1425.
    • (1995) J Natural Prod , vol.58 , pp. 1423-1425
    • Chen, C.C.1    Lin, C.E.2    Huang, Y.L.3    Ko, F.N.4    Teng, C.M.5
  • 54
    • 12544260786 scopus 로고
    • Receptor and tissue dependent effects of abanoquil (UK52046)
    • Chess-Williams R, Jackson AH (1993): Receptor and tissue dependent effects of abanoquil (UK52046). Br J Pharmacol 108 (Suppl):115P.
    • (1993) Br J Pharmacol , vol.108 , Issue.SUPPL.
    • Chess-Williams, R.1    Jackson, A.H.2
  • 59
    • 0030000076 scopus 로고    scopus 로고
    • Inhibition by tamsulosin of tension responses of human hyperplastic prostate to electrical field stimulation
    • Chueh S-C, Guh J-H, Chen J, Lai M-K, Ko F-N, Teng C-M (1996): Inhibition by tamsulosin of tension responses of human hyperplastic prostate to electrical field stimulation. Eur J Pharmacol 305:177-180.
    • (1996) Eur J Pharmacol , vol.305 , pp. 177-180
    • Chueh, S.-C.1    Guh, J.-H.2    Chen, J.3    Lai, M.-K.4    Ko, F.-N.5    Teng, C.-M.6
  • 61
    • 0020056976 scopus 로고
    • The existence of a new subtype of α-adrenoceptor on the rat anococcygeus is revealed by SGD 101/75 and phenoxybenzamine
    • Coates J, Jahn U, Weetman DF (1982): The existence of a new subtype of α-adrenoceptor on the rat anococcygeus is revealed by SGD 101/75 and phenoxybenzamine. Br J Pharmacol 75:549-552.
    • (1982) Br J Pharmacol , vol.75 , pp. 549-552
    • Coates, J.1    Jahn, U.2    Weetman, D.F.3
  • 62
    • 0019133163 scopus 로고
    • In vitro comparison of the pre- And postsynaptic alpha adrenergic receptor blocking properties of prazosin and tiodazosin (BL5111)
    • Cohen ML, Wiley KW, Landry SAS (1980): In vitro comparison of the pre- and postsynaptic alpha adrenergic receptor blocking properties of prazosin and tiodazosin (BL5111). Clin Exp Hypertens 2:1067-1082.
    • (1980) Clin Exp Hypertens , vol.2 , pp. 1067-1082
    • Cohen, M.L.1    Wiley, K.W.2    Landry, S.A.S.3
  • 63
    • 0028815327 scopus 로고
    • Novel and highly selective postsynaptic α-adrenoreceptor antagonists: Synthesis and structure-activity relationships of alkane-bridged[4-(phenoxyethyl)-l-piperazinyl]-3(2H)-pyridazinones
    • Corsano S, Scapicchi R, Strappaghetti G, Marucci G, Paparelli F (1995): Novel and highly selective postsynaptic α-adrenoreceptor antagonists: Synthesis and structure-activity relationships of alkane-bridged[4-(phenoxyethyl)-l-piperazinyl]-3(2H)-pyridazinones. Eur J Med Chem 30:71-75.
    • (1995) Eur J Med Chem , vol.30 , pp. 71-75
    • Corsano, S.1    Scapicchi, R.2    Strappaghetti, G.3    Marucci, G.4    Paparelli, F.5
  • 65
    • 0023718592 scopus 로고
    • 1-adrenergic receptor antagonists for the treatment of hypertension: Role of vascular alpha receptors in the control of peripheral resistance
    • 1-adrenergic receptor antagonists for the treatment of hypertension: Role of vascular alpha receptors in the control of peripheral resistance. Am Heart J 116:133-162.
    • (1988) Am Heart J , vol.116 , pp. 133-162
    • Cubeddu, L.X.1
  • 70
    • 0020622573 scopus 로고
    • An investigation of presynaptic α-adrenoceptor subtypes in the pithed rat
    • Docherty JR (1983): An investigation of presynaptic α-adrenoceptor subtypes in the pithed rat. Br J Pharmacol 78:655-658.
    • (1983) Br J Pharmacol , vol.78 , pp. 655-658
    • Docherty, J.R.1
  • 72
    • 0028050150 scopus 로고
    • 1-adrenoceptor mediated prostatic smooth muscle contraction
    • 1-adrenoceptor mediated prostatic smooth muscle contraction. Urol Res 22:143-146.
    • (1994) Urol Res , vol.22 , pp. 143-146
    • Drescher, P.1    Eckert, R.E.2    Madsen, P.O.3
  • 73
    • 0021961876 scopus 로고
    • What do antagonists tell us about α-adrenoceptors?
    • Drew CM (1985): What do antagonists tell us about α-adrenoceptors? Clin Sci 68 (Suppl. 10):15S-19S.
    • (1985) Clin Sci , vol.68 , Issue.10 SUPPL.
    • Drew, C.M.1
  • 74
    • 0018861853 scopus 로고
    • Lack of correlation between inhibition of noradrenaline release and end organ response during nerve stimulation
    • Dubocovich ML, Langer SZ, Massingham R (1980): Lack of correlation between inhibition of noradrenaline release and end organ response during nerve stimulation. Br J Pharmacol 69:81-89.
    • (1980) Br J Pharmacol , vol.69 , pp. 81-89
    • Dubocovich, M.L.1    Langer, S.Z.2    Massingham, R.3
  • 75
  • 77
    • 0028181642 scopus 로고
    • 1bAdrenoceptors mediate renal tubular sodium and water reabsorption in the rat
    • 1bAdrenoceptors mediate renal tubular sodium and water reabsorption in the rat. Br J Pharmacol 111:819-824.
    • (1994) Br J Pharmacol , vol.111 , pp. 819-824
    • Elhawary, A.M.1    Pang, C.C.Y.2
  • 78
    • 0026585158 scopus 로고
    • Subtype-selective alphal-adrenoceptor alleviation in the rat kidney and its effect on the vascular presser response
    • Elhawary AM, Pettinger WA, Wolff DW (1992): Subtype-selective alphal-adrenoceptor alleviation in the rat kidney and its effect on the vascular presser response. J Pharmacol Exp Ther 260:709-713.
    • (1992) J Pharmacol Exp Ther , vol.260 , pp. 709-713
    • Elhawary, A.M.1    Pettinger, W.A.2    Wolff, D.W.3
  • 79
    • 0028170294 scopus 로고
    • 1-adrenoceptor subtype mediating contraction of guinea-pig spleen
    • 1-adrenoceptor subtype mediating contraction of guinea-pig spleen. Eur J Pharmacol 260:211-220.
    • (1994) Eur J Pharmacol , vol.260 , pp. 211-220
    • Eltze, M.1
  • 80
  • 81
    • 0026564466 scopus 로고
    • 1B-adrenoceptor subtypes in vas deferens, kidney and aorta of the rat
    • 1B-adrenoceptor subtypes in vas deferens, kidney and aorta of the rat. Eur J Pharmacol 224:125-136.
    • (1992) Eur J Pharmacol , vol.224 , pp. 125-136
    • Eltze, M.1    Boer, R.2
  • 83
    • 0029946203 scopus 로고    scopus 로고
    • 1-adrenoceptors that regulate contractile function: Subtypes and subcellular signal transduction mechanisms
    • 1-adrenoceptors that regulate contractile function: Subtypes and subcellular signal transduction mechanisms. Neurochem Res 21:217-229.
    • (1996) Neurochem Res , vol.21 , pp. 217-229
    • Endoh, M.1
  • 85
    • 0027295516 scopus 로고
    • 1-adrenergic receptor subtypes and signal transduction in SK-N-MC and NB41A3 neuronal cell lines
    • 1-adrenergic receptor subtypes and signal transduction in SK-N-MC and NB41A3 neuronal cell lines. Mol Pharmacol 44:76-86.
    • (1993) Mol Pharmacol , vol.44 , pp. 76-86
    • Esbenshade, T.A.1    Han, C.2    Murphy, R.J.3    Minneman, K.P.4
  • 87
    • 0022947140 scopus 로고
    • α-Adrenoceptor subclassification in vascular smooth muscle
    • Flavahan NA, Vanhoutte PM (1986): α-Adrenoceptor subclassification in vascular smooth muscle. Trends Pharmacol Sci 7:347-349.
    • (1986) Trends Pharmacol Sci , vol.7 , pp. 347-349
    • Flavahan, N.A.1    Vanhoutte, P.M.2
  • 88
    • 0028981636 scopus 로고
    • 1-adrenoceptors to characterize subtype selectivity of drugs for the treatment of prostatic hypertrophy
    • 1-adrenoceptors to characterize subtype selectivity of drugs for the treatment of prostatic hypertrophy. Eur J Pharmacol 288:201-207.
    • (1995) Eur J Pharmacol , vol.288 , pp. 201-207
    • Foglar, R.1    Shibata, K.2    Horie, K.3    Hirasawa, A.4    Tsujimoto, G.5
  • 95
    • 0029561818 scopus 로고
    • Alpha sympathomimetic treatment of autonomic insufficiency with orthostatic hypotension
    • Fouad-Tarazi FM, Okabe M, Goren H (1995): Alpha sympathomimetic treatment of autonomic insufficiency with orthostatic hypotension. Am J Med 99:604-610.
    • (1995) Am J Med , vol.99 , pp. 604-610
    • Fouad-Tarazi, F.M.1    Okabe, M.2    Goren, H.3
  • 96
    • 0021909138 scopus 로고
    • Recovery of α-adrenoreceptor mediated responses and binding site number after intravenous benextramine in the rabbit
    • Furnace G, Hamilton CA, Reid JL, Sumner DJ (1985): Recovery of α-adrenoreceptor mediated responses and binding site number after intravenous benextramine in the rabbit. J Auton Pharmacol 5:13-17.
    • (1985) J Auton Pharmacol , vol.5 , pp. 13-17
    • Furnace, G.1    Hamilton, C.A.2    Reid, J.L.3    Sumner, D.J.4
  • 103
    • 0029614872 scopus 로고
    • Chloroethylclonidine increases the incidence of lethal arrhythmias during coronary occlusion in anesthetized dogs
    • Geller JC, Cua M, Prieto L, Guo S-D, Danilo P Jr, Rosen MR (1995): Chloroethylclonidine increases the incidence of lethal arrhythmias during coronary occlusion in anesthetized dogs. Eur J Pharmacol 294:423-428.
    • (1995) Eur J Pharmacol , vol.294 , pp. 423-428
    • Geller, J.C.1    Cua, M.2    Prieto, L.3    Guo, S.-D.4    Danilo Jr., P.5    Rosen, M.R.6
  • 107
    • 0026356256 scopus 로고
    • Ability of SK&F 104078 and SK&F 104856 to identify alpha-2 adrenoceptor subtypes in NCB20 cells and guinea pig lung
    • Cleason MM, Hieble JP (1991): Ability of SK&F 104078 and SK&F 104856 to identify alpha-2 adrenoceptor subtypes in NCB20 cells and guinea pig lung. J Pharmacol Exp Ther 259:1124-1132.
    • (1991) J Pharmacol Exp Ther , vol.259 , pp. 1124-1132
    • Cleason, M.M.1    Hieble, J.P.2
  • 110
    • 0020686545 scopus 로고
    • Actions of nifedipine on calcium fluxes and contraction in isolated rat arteries
    • Godfraind T (1983): Actions of nifedipine on calcium fluxes and contraction in isolated rat arteries. J Pharmacol Exp Ther 224:443-450.
    • (1983) J Pharmacol Exp Ther , vol.224 , pp. 443-450
    • Godfraind, T.1
  • 111
    • 0028125160 scopus 로고
    • Characterization of alpha-1 adrenoceptor subtypes in human and canine prostate membranes
    • Goetz AS, Lutz MW, Rimele TJ, Saussy DL Jr (1994): Characterization of alpha-1 adrenoceptor subtypes in human and canine prostate membranes. J Pharmacol Exp Ther 271:1228-1233.
    • (1994) J Pharmacol Exp Ther , vol.271 , pp. 1228-1233
    • Goetz, A.S.1    Lutz, M.W.2    Rimele, T.J.3    Saussy Jr., D.L.4
  • 114
    • 0029920873 scopus 로고    scopus 로고
    • 1-adrenoceptor antagonists in the treatment of benign prostatic hyperplasia: The concept of uroselectivity
    • 1-adrenoceptor antagonists in the treatment of benign prostatic hyperplasia: The concept of uroselectivity. Eur Urol 29:378-384.
    • (1996) Eur Urol , vol.29 , pp. 378-384
    • Graham, D.1    Arbilla, S.2    Pimoule, C.3    Langer, S.Z.4
  • 115
    • 0020365397 scopus 로고
    • 1-adrenergic receptor and identification of the hormone binding subunit
    • 1-adrenergic receptor and identification of the hormone binding subunit. J Biol Chem 257:15174-15181.
    • (1982) J Biol Chem , vol.257 , pp. 15174-15181
    • Graham, R.M.1    Hess, H.J.2    Homey, C.J.3
  • 117
    • 0018332473 scopus 로고
    • Binding characteristics of 3H-prazosin to rat brain alpha-adrenergic receptors
    • Greengrass R Bremner R (1979): Binding characteristics of 3H-prazosin to rat brain alpha-adrenergic receptors. Eur J Pharmacol 55:323-326.
    • (1979) Eur J Pharmacol , vol.55 , pp. 323-326
    • Greengrass, R.1    Bremner, R.2
  • 122
    • 0028989378 scopus 로고
    • 1-adrenoceptor subtypes in tension response of human prostate to electrical field stimulation
    • 1-adrenoceptor subtypes in tension response of human prostate to electrical field stimulation. Br J Pharmacol 115:142-146.
    • (1995) Br J Pharmacol , vol.115 , pp. 142-146
    • Guh, J.-H.1    Chueh, S.A.-C.2    Ko, F.-N.3    Teng, C.-M.4
  • 123
    • 0029017730 scopus 로고
    • Pharmacological evaluation of N-methyl-actinodaphnine, a new vascular Ot-adrenoceptor antagonist, isolated from Illigera luzonensis
    • Guh J-H, Ko F-N, Yu S-M, Wu Y-C, Teng C-M (1995b): Pharmacological evaluation of N-methyl-actinodaphnine, a new vascular Ot-adrenoceptor antagonist, isolated from Illigera luzonensis. Eur J Pharmacol 279:33-41.
    • (1995) Eur J Pharmacol , vol.279 , pp. 33-41
    • Guh, J.-H.1    Ko, F.-N.2    Yu, S.-M.3    Wu, Y.-C.4    Teng, C.-M.5
  • 124
    • 0019390398 scopus 로고
    • 3H]-dihydroergocryptine to rat cardiac a-adrenoceptors
    • 3H]-dihydroergocryptine to rat cardiac a-adrenoceptors. Br J Pharmacol 73:33-39.
    • (1981) Br J Pharmacol , vol.73 , pp. 33-39
    • Guicheney, P.1    Meyer, P.2
  • 127
    • 0023513551 scopus 로고
    • 1-adrenergic receptors revealed by chlorethylclonidine
    • 1-adrenergic receptors revealed by chlorethylclonidine. Mol Pharmacol 32:505-510.
    • (1987) Mol Pharmacol , vol.32 , pp. 505-510
    • Han, C.1    Abel, P.W.2    Minneman, K.P.3
  • 128
    • 0026077322 scopus 로고
    • 1-adrenergic receptor binding sites in rat tissues
    • 1-adrenergic receptor binding sites in rat tissues. Mol Pharmacol 40:531-538.
    • (1991) Mol Pharmacol , vol.40 , pp. 531-538
    • Han, G.1    Minneman, K.P.2
  • 130
    • 84966016554 scopus 로고
    • Structure-activity relationships of imidazolines and related compounds at subtypes of Alpha-2 adrenergic receptors
    • Hancock AA, Hutchins CW, Basha FZ, DeBernardis JF (1991): Structure-activity relationships of imidazolines and related compounds at subtypes of Alpha-2 adrenergic receptors. FASEB J 5:A856.
    • (1991) FASEB J , vol.5
    • Hancock, A.A.1    Hutchins, C.W.2    Basha, F.Z.3    DeBernardis, J.F.4
  • 131
    • 0028914116 scopus 로고
    • Preclinical pharmacological actions of (±)-(1'R*,3R*)-3-phenyl-l-[(1′,2′,3′, 4′-tetrahydro-5′,6′-methylene-dioxy-1′-naphthalenyl) methyl] pyrrolidine methanesulfonate (ABT-200), a potential antidepressant agent that antagonizes alpha-2 adrenergic receptors and inhibits the neuronal uptake of norepinephrine
    • Hancock AA, Buckner SA, Giardina WJ, Brune ME, Lee JY, Morse PA, Oheim KW, Stanisic DS, Warner RB, Kerkman DJ, DeBernardis JF (1995a): Preclinical pharmacological actions of (±)-(1'R*,3R*)-3-phenyl-l-[(1′,2′,3′, 4′-tetrahydro-5′,6′-methylene-dioxy-1′-naphthalenyl) methyl] pyrrolidine methanesulfonate (ABT-200), a potential antidepressant agent that antagonizes alpha-2 adrenergic receptors and inhibits the neuronal uptake of norepinephrine. J Pharmacol Exp Ther 272:1160-1169.
    • (1995) J Pharmacol Exp Ther , vol.272 , pp. 1160-1169
    • Hancock, A.A.1    Buckner, S.A.2    Giardina, W.J.3    Brune, M.E.4    Lee, J.Y.5    Morse, P.A.6    Oheim, K.W.7    Stanisic, D.S.8    Warner, R.B.9    Kerkman, D.J.10    DeBernardis, J.F.11
  • 133
    • 0013509712 scopus 로고
    • 1-adrenoceptor binding sites in the rat heart: Subtype-selective agonists and antagonists
    • 1-adrenoceptor binding sites in the rat heart: Subtype-selective agonists and antagonists. Br J Pharmacol 98:652P.
    • (1989) Br J Pharmacol , vol.98
    • Hanft, G.1    Gross, G.2
  • 134
    • 0024360634 scopus 로고
    • 1-adrenoceptor recognition sites by urapidil derivatives and other selective antagonists
    • 1-adrenoceptor recognition sites by urapidil derivatives and other selective antagonists. Br J Pharmacol 97:691-700.
    • (1989) Br J Pharmacol , vol.97 , pp. 691-700
    • Hanft, G.1    Gross, G.2
  • 139
    • 0020520859 scopus 로고
    • 1-adrenergic receptor: Synthesis and effects on membrane and affinity-purified receptors
    • 1-adrenergic receptor: Synthesis and effects on membrane and affinity-purified receptors. Proc Natl Acad Sci USA 80:2102-2106.
    • (1983) Proc Natl Acad Sci USA , vol.80 , pp. 2102-2106
    • Hess, H.J.1    Graham, R.M.2    Homey, C.J.3
  • 140
    • 0025881062 scopus 로고
    • Three-dimensional models of neurotransmitter G-binding protein-coupled receptors
    • Hibert ME Trumpp-Kallmeyer S, Bruinvels A, Hoflack J (1991): Three-dimensional models of neurotransmitter G-binding protein-coupled receptors. Mol Pharmacol 40:8-15.
    • (1991) Mol Pharmacol , vol.40 , pp. 8-15
    • Hibert, M.E.1    Trumpp-Kallmeyer, S.2    Bruinvels, A.3    Hoflack, J.4
  • 142
    • 10344266591 scopus 로고
    • 2-adrenoceptor subtype selectivity in tissue homogenates and cell lines
    • 2-adrenoceptor subtype selectivity in tissue homogenates and cell lines. Pharmacologist 35:166.
    • (1993) Pharmacologist , vol.35 , pp. 166
    • Hieble, J.P.1    Naselsky, D.P.2
  • 143
    • 0023025411 scopus 로고
    • Comparison of the α-adrenoceptor characteristics in human and canine prostate
    • Hieble JP, Boyce AJ, Gaine M (1986): Comparison of the α-adrenoceptor characteristics in human and canine prostate. Fed Proc 45:2609-2614.
    • (1986) Fed Proc , vol.45 , pp. 2609-2614
    • Hieble, J.P.1    Boyce, A.J.2    Gaine, M.3
  • 144
    • 0029134812 scopus 로고
    • α- And β-Adrenoceptors: From the gene to the clinic. 1. Molecular biology and adrenoceptor subclassification
    • Hieble JP Bondinell WE, Ruffolo RR Jr (1995a): α- and β-Adrenoceptors: From the gene to the clinic. 1. Molecular biology and adrenoceptor subclassification. J Med Chem 38:3415-3444.
    • (1995) J Med Chem , vol.38 , pp. 3415-3444
    • Hieble, J.P.1    Bondinell, W.E.2    Ruffolo Jr., R.R.3
  • 151
    • 0018909648 scopus 로고
    • [3H]-WB4101 - Caution about its role as an alpha-adrenergic subtype selective radioligand
    • Huffman BB, Lefkowitz RJ (1980): [3H]-WB4101 - Caution about its role as an alpha-adrenergic subtype selective radioligand. Biochem Pharmacol 29:1537-1541.
    • (1980) Biochem Pharmacol , vol.29 , pp. 1537-1541
    • Huffman, B.B.1    Lefkowitz, R.J.2
  • 152
    • 0018609223 scopus 로고
    • Alpha-adrenergic receptor subtypes: Quantitative assessment by ligand binding
    • Huffman BB, DeLean A, Wood CL, Schocken DD, Lefkowitz RJ (1979): Alpha-adrenergic receptor subtypes: Quantitative assessment by ligand binding. Life Sci 24:1739-1746.
    • (1979) Life Sci , vol.24 , pp. 1739-1746
    • Huffman, B.B.1    DeLean, A.2    Wood, C.L.3    Schocken, D.D.4    Lefkowitz, R.J.5
  • 153
    • 0022974478 scopus 로고
    • Alpha-1 adrenoceptor antagonist effects of the optical isomers of YM-12617 in rabbit lower urinary tract and prostate
    • Honda K, Nakagawa C (1986): Alpha-1 adrenoceptor antagonist effects of the optical isomers of YM-12617 in rabbit lower urinary tract and prostate. J Pharmacol Exp Ther 239:512-516.
    • (1986) J Pharmacol Exp Ther , vol.239 , pp. 512-516
    • Honda, K.1    Nakagawa, C.2
  • 159
    • 0028039636 scopus 로고
    • Three-dimensional models of the D1 and D2 dopamine receptors
    • Hutchins C (1994): Three-dimensional models of the D1 and D2 dopamine receptors. Endocr J 2:7-23.
    • (1994) Endocr J , vol.2 , pp. 7-23
    • Hutchins, C.1
  • 160
    • 12644255702 scopus 로고    scopus 로고
    • Models of ligand binding and receptor function of the G protein-coupled receptors
    • Schwartz TW, Hjorth SA, Kastrup JS (eds): Kopenhagen: Munksgaard
    • Hutchins C (1996): Models of ligand binding and receptor function of the G protein-coupled receptors. In Schwartz TW, Hjorth SA, Kastrup JS (eds): Structure and Function of 7TM Receptors. Kopenhagen: Munksgaard, pp 213-226.
    • (1996) Structure and Function of 7TM Receptors , pp. 213-226
    • Hutchins, C.1
  • 161
    • 0029117219 scopus 로고
    • 1-adrenergic receptor subtype selective agonist binding
    • 1-adrenergic receptor subtype selective agonist binding. J Biol Chem 270:23189-23195.
    • (1995) J Biol Chem , vol.270 , pp. 23189-23195
    • Hwa, J.1    Graham, R.M.2    Ferez, D.M.3
  • 166
    • 0023637604 scopus 로고
    • Analysis of putative Alpha-1s adrenoceptor agonism by Sgd 101/75 in the rat anococcygeus muscle
    • James MK, Leighton HJ (1987): Analysis of putative Alpha-1s adrenoceptor agonism by Sgd 101/75 in the rat anococcygeus muscle. J Pharmacol Exp Ther 242:772-776.
    • (1987) J Pharmacol Exp Ther , vol.242 , pp. 772-776
    • James, M.K.1    Leighton, H.J.2
  • 167
    • 0027371594 scopus 로고
    • Long-term treatment of benign prostatic hyperplasia with alfuzosin: A 12-18 month assessment
    • Jardin A, Bensadoun H, Delauche-Cavallier MC, Attali P, BPHALF group (1993): Long-term treatment of benign prostatic hyperplasia with alfuzosin: A 12-18 month assessment. Br J Urol 72:615-620.
    • (1993) Br J Urol , vol.72 , pp. 615-620
    • Jardin, A.1    Bensadoun, H.2    Delauche-Cavallier, M.C.3    Attali, P.4
  • 168
    • 0022479786 scopus 로고
    • 1-adrenoceptor mediated pressor responses by calcium channel antagonists in the pithed rat
    • 1-adrenoceptor mediated pressor responses by calcium channel antagonists in the pithed rat. J Pharmacol Exp Ther 238:89-94.
    • (1986) J Pharmacol Exp Ther , vol.238 , pp. 89-94
    • Jim, K.F.1    Maria, R.A.2    Matthews, W.D.3
  • 170
    • 0028970777 scopus 로고
    • 1-adrenoceptor agonist, SDZ NVI-085, in guinea pigs
    • 1-adrenoceptor agonist, SDZ NVI-085, in guinea pigs. Eur J Pharmacol 285:313-315.
    • (1995) Eur J Pharmacol , vol.285 , pp. 313-315
    • Kalkman, H.1    Neumann, V.2
  • 172
    • 0029914810 scopus 로고    scopus 로고
    • Efficacy of nonsurgical therapy for urinary incontinence
    • Karram MM, Partoll L, Rahe J (1996): Efficacy of nonsurgical therapy for urinary incontinence. J Reprod Med 41:215-219.
    • (1996) J Reprod Med , vol.41 , pp. 215-219
    • Karram, M.M.1    Partoll, L.2    Rahe, J.3
  • 173
    • 0023924985 scopus 로고
    • Treatment of orthostatic hypotension due to autonomic failure with a peripheral alpha-adrenergic agonist (midodrine)
    • Kaufmann H, Brannan T, Krakoff L, Yahr MD, Mandeli J (1988): Treatment of orthostatic hypotension due to autonomic failure with a peripheral alpha-adrenergic agonist (midodrine). Neurology 38:951-956.
    • (1988) Neurology , vol.38 , pp. 951-956
    • Kaufmann, H.1    Brannan, T.2    Krakoff, L.3    Yahr, M.D.4    Mandeli, J.5
  • 174
    • 84977404328 scopus 로고
    • Analysis of alpha-1 adrenoceptors in human prostate
    • Kawabe K (1993): Analysis of alpha-1 adrenoceptors in human prostate. Aktuel Urol 24:82-85.
    • (1993) Aktuel Urol , vol.24 , pp. 82-85
    • Kawabe, K.1
  • 175
    • 0029034556 scopus 로고
    • Efficacy and safety of tamsulosin in the treatment of benign prostatic hyperplasia
    • Kawabe K (1995): Efficacy and safety of tamsulosin in the treatment of benign prostatic hyperplasia. Br J Urol 76 (Suppl 1):63-67.
    • (1995) Br J Urol , vol.76 , Issue.1 SUPPL. , pp. 63-67
    • Kawabe, K.1
  • 176
    • 21344471853 scopus 로고    scopus 로고
    • 1-blocker, in the treatment of BPH (benign prostatic hyperplasia)
    • 1-blocker, in the treatment of BPH (benign prostatic hyperplasia). Aktuel Urol 27:25-26.
    • (1996) Aktuel Urol , vol.27 , pp. 25-26
    • Kawabe, K.1
  • 182
    • 0025891495 scopus 로고
    • 1-adrenergic receptor subtypes: MDCK-D1 cells, but not rat cortical membranes possess a single population of receptors
    • 1-adrenergic receptor subtypes: MDCK-D1 cells, but not rat cortical membranes possess a single population of receptors. Mol Pharmacol 39:407-413.
    • (1990) Mol Pharmacol , vol.39 , pp. 407-413
    • Klijn, K.1    Slivka, S.R.2    Bell, K.3    Insel, P.A.4
  • 184
    • 0027198082 scopus 로고
    • Pharmacological activity of (-)-discretamine, a novel vascular α-adrenoceptor and 5-hydroxytryptamine receptor antagonist, isolated from Fissistigma glaucenscens
    • Ko FN, Yu SM, Su MJ, Wu YC, Teng CM (1993): Pharmacological activity of (-)-discretamine, a novel vascular (α-adrenoceptor and 5-hydroxytryptamine receptor antagonist, isolated from Fissistigma glaucenscens. Br J Pharmacol 110:882-88.
    • (1993) Br J Pharmacol , vol.110 , pp. 882-888
    • Ko, F.N.1    Yu, S.M.2    Su, M.J.3    Wu, Y.C.4    Teng, C.M.5
  • 187
    • 0027332577 scopus 로고
    • 1A-adrenoceptor subtypes in rabbit: Differentiation by a selective antagonist, HV723
    • 1A-adrenoceptor subtypes in rabbit: differentiation by a selective antagonist, HV723. Eur J Pharmacol 250:95-101.
    • (1993) Eur J Pharmacol , vol.250 , pp. 95-101
    • Kohi, M.1    Yang, H.-T.2    Endoh, M.3
  • 189
    • 0028875731 scopus 로고
    • Effects of α-adrenergic blockade on regional myocardial function in canine ischemic myocardium during β-adrenergic blockade
    • Kono M, Morita S, Rubsamen R (1995): Effects of α-adrenergic blockade on regional myocardial function in canine ischemic myocardium during β-adrenergic blockade. J Cardiothoracic Vase Anesthes 9:525-533.
    • (1995) J Cardiothoracic Vase Anesthes , vol.9 , pp. 525-533
    • Kono, M.1    Morita, S.2    Rubsamen, R.3
  • 190
    • 0026762882 scopus 로고
    • Effects of adrenergic agonists on an experimental urinary incontinence model in anesthetized rabbits
    • Kontani H, Nakagawa M, Sakai T (1992): Effects of adrenergic agonists on an experimental urinary incontinence model in anesthetized rabbits. Jap J Pharmacol 58:339-346.
    • (1992) Jap J Pharmacol , vol.58 , pp. 339-346
    • Kontani, H.1    Nakagawa, M.2    Sakai, T.3
  • 198
    • 0001423969 scopus 로고
    • Presynaptic regulation of catecholamine release
    • Langer SZ (1974): Presynaptic regulation of catecholamine release. Br J Pharmacol 60:481-497.
    • (1974) Br J Pharmacol , vol.60 , pp. 481-497
    • Langer, S.Z.1
  • 201
    • 0002556259 scopus 로고
    • In vivo uroselectivity of alfuzosin compared to prazosin and terazosin
    • Lefèvre-Borg F Lechaire J, O'Connor S (1992): In vivo uroselectivity of alfuzosin compared to prazosin and terazosin. Br J Pharmacol 106 (Suppl):84P.
    • (1992) Br J Pharmacol , vol.106 , Issue.SUPPL.
    • Lefèvre-Borg, F.1    Lechaire, J.2    O'Connor, S.3
  • 203
    • 0029002424 scopus 로고
    • Alpha blockade for the treatment of benign prostatic hyperplasia
    • Lepor H, (1995): Alpha blockade for the treatment of benign prostatic hyperplasia. Urol Clin North Am 22:375-386.
    • (1995) Urol Clin North Am , vol.22 , pp. 375-386
    • Lepor, H.1
  • 204
    • 0027530990 scopus 로고
    • Alphal adrenoceptor subtypes in the human prostate
    • Lepor H, Tang R, Meretyk S, Shapiro E (1993a): Alphal adrenoceptor subtypes in the human prostate. J Urol 149:640-642.
    • (1993) J Urol , vol.149 , pp. 640-642
    • Lepor, H.1    Tang, R.2    Meretyk, S.3    Shapiro, E.4
  • 205
    • 0027222669 scopus 로고
    • The alpha-adrenoceptor subtype mediating the tension of human prostatic smooth muscle
    • Lepor H, Tang R, Shapiro E (1993b): The alpha-adrenoceptor subtype mediating the tension of human prostatic smooth muscle. Prostate 22:301-307.
    • (1993) Prostate , vol.22 , pp. 301-307
    • Lepor, H.1    Tang, R.2    Shapiro, E.3
  • 206
    • 0028092817 scopus 로고
    • A comparison of the binding and functional properties of alpha-1 adrenoceptors and area density of smooth muscle in the human, canine and rat prostates
    • Lepor H, Zhang W, Kobayashi S, Tang R, Wang B, Shapiro E (1994): A comparison of the binding and functional properties of alpha-1 adrenoceptors and area density of smooth muscle in the human, canine and rat prostates. J Pharmacol Exp Ther 270:722-727.
    • (1994) J Pharmacol Exp Ther , vol.270 , pp. 722-727
    • Lepor, H.1    Zhang, W.2    Kobayashi, S.3    Tang, R.4    Wang, B.5    Shapiro, E.6
  • 208
    • 0023878170 scopus 로고
    • Identification of receptor subtypes in the rabbit and human urinary bladder by selective radio-ligand binding
    • Levin RM, Ruggieri MR, Wein AJ (1988): Identification of receptor subtypes in the rabbit and human urinary bladder by selective radio-ligand binding. J Urol 139:844-848.
    • (1988) J Urol , vol.139 , pp. 844-848
    • Levin, R.M.1    Ruggieri, M.R.2    Wein, A.J.3
  • 209
    • 0026675087 scopus 로고
    • Role of catecholamines in the modaflnil and amphetamine induced wakefulness, a comparative pharmacological study in the cat
    • Lin JS, Roussel B, Akaoka H, Fort P Debilly G, Jouvet M (1992): Role of catecholamines in the modaflnil and amphetamine induced wakefulness, a comparative pharmacological study in the cat. Brain Res 591:319-326.
    • (1992) Brain Res , vol.591 , pp. 319-326
    • Lin, J.S.1    Roussel, B.2    Akaoka, H.3    Fort, P.4    Debilly, G.5    Jouvet, M.6
  • 214
    • 0028004411 scopus 로고
    • Interactions of chloroethylclonidine with rauwolscine- And prazosin-sensitive adrenoceptors in dogsaphenous vein
    • Low AM, Bowdish DM, Prashad TR, Caspar V (1994): Interactions of chloroethylclonidine with rauwolscine- and prazosin-sensitive adrenoceptors in dogsaphenous vein. Br J Pharmacol 113:1263-1268.
    • (1994) Br J Pharmacol , vol.113 , pp. 1263-1268
    • Low, A.M.1    Bowdish, D.M.2    Prashad, T.R.3    Caspar, V.4
  • 215
    • 0030058397 scopus 로고    scopus 로고
    • Safety profile of 3 months therapy with alfuzosin in 13,389 patients suffering from benign prostatic hypertrophy
    • Lukacs B, Blondin P, MacCarthy C, Du Boys B, Grippon P, Lassale C (1996): Safety profile of 3 months therapy with alfuzosin in 13,389 patients suffering from benign prostatic hypertrophy. Eur Urol 29:29-35.
    • (1996) Eur Urol , vol.29 , pp. 29-35
    • Lukacs, B.1    Blondin, P.2    MacCarthy, C.3    Du Boys, B.4    Grippon, P.5    Lassale, C.6
  • 216
    • 0018875038 scopus 로고
    • Multiple central WB-4101 binding sites and the selectivity of prazosin
    • Lyon TF Randall WC (1980): Multiple central WB-4101 binding sites and the selectivity of prazosin. Life Sci 26:1121-1129.
    • (1980) Life Sci , vol.26 , pp. 1121-1129
    • Lyon, T.F.1    Randall, W.C.2
  • 217
    • 0026504481 scopus 로고
    • 1B-adrenoceptor mediated components in the tension response of the rat vas deferens to electrical field stimulation
    • 1B-adrenoceptor mediated components in the tension response of the rat vas deferens to electrical field stimulation. Br J Pharmacol 105:727-731.
    • (1992) Br J Pharmacol , vol.105 , pp. 727-731
    • Mallard, N.J.1    Marshall, R.W.2    Sithers, A.J.3    Spriggs, T.L.B.4
  • 222
    • 4243567036 scopus 로고
    • Effects of alfuzosin on urethral and blood pressures in conscious male rats
    • Martin D, Jammes D, Angel I (1995): Effects of alfuzosin on urethral and blood pressures in conscious male rats. Life Sci 57:387-391.
    • (1995) Life Sci , vol.57 , pp. 387-391
    • Martin, D.1    Jammes, D.2    Angel, I.3
  • 223
    • 0022972136 scopus 로고
    • Hypotensive effect in dogs and rats of intravenous injections of the α1-adrenoreceptor antagonist benoxathian
    • Massi M, Venturi F, Brasili L, Melchiorre C (1986): Hypotensive effect in dogs and rats of intravenous injections of the α1-adrenoreceptor antagonist benoxathian. Pharmacol Res Commun 18:813-829.
    • (1986) Pharmacol Res Commun , vol.18 , pp. 813-829
    • Massi, M.1    Venturi, F.2    Brasili, L.3    Melchiorre, C.4
  • 225
    • 0024385133 scopus 로고
    • Midodrine: A review of its pharmacological properties and therapeutic use in orthostatic hypotension and secondary hypotensive disorders
    • McTavish D, Goa KL (1989): Midodrine: A review of its pharmacological properties and therapeutic use in orthostatic hypotension and secondary hypotensive disorders. Drugs 38:757-777.
    • (1989) Drugs , vol.38 , pp. 757-777
    • McTavish, D.1    Goa, K.L.2
  • 226
    • 0018119235 scopus 로고
    • Molecular properties of the adrenergic receptor. 2. Optimum covalent inhibition by two different prototypes of polyamine disulphides
    • Melchiorre C, Young MS, Benfey BG, Belleau B (1978): Molecular properties of the adrenergic receptor. 2. Optimum covalent inhibition by two different prototypes of polyamine disulphides. J Med Chem 21:1126-1132.
    • (1978) J Med Chem , vol.21 , pp. 1126-1132
    • Melchiorre, C.1    Young, M.S.2    Benfey, B.G.3    Belleau, B.4
  • 236
    • 0028015747 scopus 로고
    • Modafinil binds to the dopamine uptake carrier site with low affinity
    • Mignot E, Nishino S, Guilleminault C, Dement WC (1994): Modafinil binds to the dopamine uptake carrier site with low affinity. Sleep 17:436-437.
    • (1994) Sleep , vol.17 , pp. 436-437
    • Mignot, E.1    Nishino, S.2    Guilleminault, C.3    Dement, W.C.4
  • 242
    • 0023912857 scopus 로고
    • 1-adrenergic receptor subtypes distinguished by chlorethylclonidine and WB 4101
    • 1-adrenergic receptor subtypes distinguished by chlorethylclonidine and WB 4101. Mol Pharmacol 33:509-514.
    • (1988) Mol Pharmacol , vol.33 , pp. 509-514
    • Minneman, K.P.1    Han, C.2    Abel, P.3
  • 244
    • 0029588298 scopus 로고
    • Novel French antidepressants not available in the United States
    • Mitchell PB (1995): Novel French antidepressants not available in the United States. Psychopharmacol Bull 31:509-519.
    • (1995) Psychopharmacol Bull , vol.31 , pp. 509-519
    • Mitchell, P.B.1
  • 245
    • 0028053819 scopus 로고
    • 1-adrenoceptor-blocking activity in experimental animals
    • 1-adrenoceptor-blocking activity in experimental animals. Am J Hypertens 7:1315-1405.
    • (1994) Am J Hypertens , vol.7 , pp. 1315-1405
    • Miyazaki, M.1
  • 249
    • 0021929317 scopus 로고
    • 2-adrenoceptor antagonist in guinea-pit ileum
    • 2-adrenoceptor antagonist in guinea-pit ileum. Gen Pharmacol 16:367-370.
    • (1985) Gen Pharmacol , vol.16 , pp. 367-370
    • Mottram, D.R.1    Saggar, P.2
  • 250
    • 0020517823 scopus 로고
    • Tissue specific susceptibility of alpha-adrenoceptor mediated vasoconstriction to nifedipine
    • Müller-Schweinitzer E (1983): Tissue specific susceptibility of alpha-adrenoceptor mediated vasoconstriction to nifedipine. Naunyn-Schmiedeberg Arch Pharmacol 324:64-69.
    • (1983) Naunyn-Schmiedeberg Arch Pharmacol , vol.324 , pp. 64-69
    • Müller-Schweinitzer, E.1
  • 251
    • 0025048314 scopus 로고
    • 1-adrenoceptors in noradrenaline contraction of the rabbit thoracic aorta
    • 1-adrenoceptors in noradrenaline contraction of the rabbit thoracic aorta. Br J Pharmacol 101:662-666.
    • (1990) Br J Pharmacol , vol.101 , pp. 662-666
    • Muramatsu, I.1    Kigoshi, S.2    Oshita, M.3
  • 253
    • 0026343250 scopus 로고
    • 1-adrenoceptors involved in noradrenaline-induced contractions of rat thoracic aorta and dog carotid artery
    • 1-adrenoceptors involved in noradrenaline-induced contractions of rat thoracic aorta and dog carotid artery. Br J Pharmacol 57:535-544.
    • (1991) Br J Pharmacol , vol.57 , pp. 535-544
    • Muramatsu, I.1    Kigoshi, S.2    Ohmura, T.3
  • 258
    • 0023850458 scopus 로고
    • Characterization of alpha-2 adrenergic receptors in the OK cell, an opossum kidney cell line
    • Murphy TJ, Bylund DB (1988): Characterization of alpha-2 adrenergic receptors in the OK cell, an opossum kidney cell line. J Pharmacol Exp Ther 244:571-578.
    • (1988) J Pharmacol Exp Ther , vol.244 , pp. 571-578
    • Murphy, T.J.1    Bylund, D.B.2
  • 259
    • 0027156224 scopus 로고
    • Nonamphetamine awakening agent modafinil induces feeding changes in the rat
    • Nicolaidis S, de Saint Hilaire Z (1993): Nonamphetamine awakening agent modafinil induces feeding changes in the rat. Brain Res Bull 32:87-90.
    • (1993) Brain Res Bull , vol.32 , pp. 87-90
    • Nicolaidis, S.1    De Saint Hilaire, Z.2
  • 260
    • 0027519506 scopus 로고
    • Further characterization of the alpha-1 receptor subtype involved in the control of cataplexy in canine narcolepsy
    • Nishino S, Fruhstorfer B, Arrigoni J, Guilleminault C, Dement WC, Mignot E (1993): Further characterization of the alpha-1 receptor subtype involved in the control of cataplexy in canine narcolepsy. J Pharmacol Exp Ther 264:1079-1084.
    • (1993) J Pharmacol Exp Ther , vol.264 , pp. 1079-1084
    • Nishino, S.1    Fruhstorfer, B.2    Arrigoni, J.3    Guilleminault, C.4    Dement, W.C.5    Mignot, E.6
  • 261
    • 0028198502 scopus 로고
    • Clinical effect of midodrine hydrochloride on the patients with urinary incontinence
    • Nito H (1994): Clinical effect of midodrine hydrochloride on the patients with urinary incontinence. Hinyokika Kiyo 40:91-94.
    • (1994) Hinyokika Kiyo , vol.40 , pp. 91-94
    • Nito, H.1
  • 264
    • 0028988260 scopus 로고
    • Pharmacological characterization of α1-adrenoceptor subtypes in rat heart: A binding study
    • Noguchi H, Muraoka R, Kigoshi S, Muramatsu I (1995): Pharmacological characterization of α1-adrenoceptor subtypes in rat heart: A binding study. Br J Pharmacol 114:1026-1030.
    • (1995) Br J Pharmacol , vol.114 , pp. 1026-1030
    • Noguchi, H.1    Muraoka, R.2    Kigoshi, S.3    Muramatsu, I.4
  • 269
  • 273
    • 0029161759 scopus 로고
    • Investigation of the actions of chloroethylclonidine in rat aorta
    • O'Rourke M, Kearns S, Docherty JR (1995): Investigation of the actions of chloroethylclonidine in rat aorta. Br J Pharmacol 115:1399-1406.
    • (1995) Br J Pharmacol , vol.115 , pp. 1399-1406
    • O'Rourke, M.1    Kearns, S.2    Docherty, J.R.3
  • 274
    • 0343549703 scopus 로고
    • 1-adrenoceptor subtypes and causes relaxation of arterial smooth muscle by raising cGMP levels
    • 1-adrenoceptor subtypes and causes relaxation of arterial smooth muscle by raising cGMP levels. Br J Pharmacol 115:215P.
    • (1994) Br J Pharmacol , vol.115
    • Orsetti, M.1    DiStilo, A.2
  • 276
    • 0027049650 scopus 로고
    • 1-adrenoceptor antagonist, anti-arrhythmic
    • 1-adrenoceptor antagonist, anti-arrhythmic. Drugs Future 17:983-986.
    • (1992) Drugs Future , vol.17 , pp. 983-986
    • Pento, J.1
  • 278
    • 0030049488 scopus 로고    scopus 로고
    • Constitutive activation of a single effector pathway: Evidence for multiple activation states of a G protein-coupled receptor
    • Perez DM, Hwa J, Gaivin R, Mathur M, Brown E Graham RM (1996): Constitutive activation of a single effector pathway: Evidence for multiple activation states of a G protein-coupled receptor. Mol Pharmacol 49:112-122.
    • (1996) Mol Pharmacol , vol.49 , pp. 112-122
    • Perez, D.M.1    Hwa, J.2    Gaivin, R.3    Mathur, M.4    Brown, E.5    Graham, R.M.6
  • 280
    • 0025297549 scopus 로고
    • 1-adrenoceptor subtypes in the regulation of arterial blood pressure
    • 1-adrenoceptor subtypes in the regulation of arterial blood pressure. Eur J Pharmacol 180:381-386.
    • (1990) Eur J Pharmacol , vol.180 , pp. 381-386
    • Piascik, M.T.1    Butler, B.T.2    Pruitt, T.A.3
  • 281
    • 0024987929 scopus 로고
    • 1-Adrenoceptor subtypes and the regulation of peripheral hemodynamics in the conscious rat
    • 1-Adrenoceptor subtypes and the regulation of peripheral hemodynamics in the conscious rat. Eur J Pharmacol 180:273-278.
    • (1990) Eur J Pharmacol , vol.180 , pp. 273-278
    • Piascik, M.T.1    Kusiak, J.W.2    Barron, K.W.3
  • 282
    • 0027732754 scopus 로고
    • EE the regulation of regional hemodynamics by alpha-1 adrenoceptor subtypes in the conscious rat
    • Piascik MT, Smith MS, Barron KW, Soltis (1993): EE The regulation of regional hemodynamics by alpha-1 adrenoceptor subtypes in the conscious rat. J Pharmacol Exp Ther 267:1250-1255.
    • (1993) J Pharmacol Exp Ther , vol.267 , pp. 1250-1255
    • Piascik, M.T.1    Smith, M.S.2    Barron, K.W.3    Soltis4
  • 284
    • 0017094668 scopus 로고
    • Pharmacodynamic actions of midodrine, a new α-adrenergic stimulating agent, and its main metabolite, ST 1059
    • Pittner H, Stormann J, Enzenhofer R (1976): Pharmacodynamic actions of midodrine, a new α-adrenergic stimulating agent, and its main metabolite, ST 1059. Arzneim-Forsch/Drug Res 26:2145-2154.
    • (1976) Arzneim-Forsch/Drug Res , vol.26 , pp. 2145-2154
    • Pittner, H.1    Stormann, J.2    Enzenhofer, R.3
  • 285
    • 0028227967 scopus 로고
    • A comparison of postspace-flight orthostatic intolerance to vasovagal syncope and autonomie failure and the potential use of the alpha agonist midodrine for these conditions
    • Piwinski SE, Jankovic J, McElligott MA (1994): A comparison of postspace-flight orthostatic intolerance to vasovagal syncope and autonomie failure and the potential use of the alpha agonist midodrine for these conditions. J Clin Pharmacol 34:466-471.
    • (1994) J Clin Pharmacol , vol.34 , pp. 466-471
    • Piwinski, S.E.1    Jankovic, J.2    McElligott, M.A.3
  • 287
    • 0027176259 scopus 로고
    • Structure-activity relationships in 1,4-benzodioxan-related compounds. 4. Effect of aryl and alkyl substituants at position 3 on α-adrenoceptor blocking activity
    • Quaglia W, Pigini M, Tayebati SK, Piergentili A, Giannella M, Marucci G, Melchiorre C (1993): Structure-activity relationships in 1,4-benzodioxan-related compounds. 4. Effect of aryl and alkyl substituants at position 3 on α-adrenoceptor blocking activity. J Med Chem 36:1520-1528.
    • (1993) J Med Chem , vol.36 , pp. 1520-1528
    • Quaglia, W.1    Pigini, M.2    Tayebati, S.K.3    Piergentili, A.4    Giannella, M.5    Marucci, G.6    Melchiorre, C.7
  • 288
    • 0029915978 scopus 로고    scopus 로고
    • Structure-activity relationships in 1,4-benzodioxan-related compounds. 5. Effects of modification of the side chain on α-adrenoceptor blocking activity
    • Quaglia W, Giannella M, Marucci G, Piergentili A, Pigini M, Tayebati SK, Melchiorre C (1996): Structure-activity relationships in 1,4-benzodioxan-related compounds. 5. Effects of modification of the side chain on α-adrenoceptor blocking activity. II Farmaco 51:27-32.
    • (1996) II Farmaco , vol.51 , pp. 27-32
    • Quaglia, W.1    Giannella, M.2    Marucci, G.3    Piergentili, A.4    Pigini, M.5    Tayebati, S.K.6    Melchiorre, C.7
  • 289
    • 0029886182 scopus 로고    scopus 로고
    • 1A-adrenoceptor antagonist for the treatment of symptomatic benign prostatic hyperplasia
    • 1A-adrenoceptor antagonist for the treatment of symptomatic benign prostatic hyperplasia. Drugs Today 32:259-268.
    • (1996) Drugs Today , vol.32 , pp. 259-268
    • Rabasseda, X.1    Fitzpatrick, J.M.2
  • 290
    • 0029609313 scopus 로고
    • A comparison of the effects of doxazosin and terazosin on the spontaneous sympathetic drive to the bladder and related organs in anaesthetized cats
    • Ramage AG, Wyllie MG (1995): A comparison of the effects of doxazosin and terazosin on the spontaneous sympathetic drive to the bladder and related organs in anaesthetized cats. Eur J Pharmacol 294:645-650.
    • (1995) Eur J Pharmacol , vol.294 , pp. 645-650
    • Ramage, A.G.1    Wyllie, M.G.2
  • 292
    • 0027174307 scopus 로고
    • 1-adrenoceptor occupancy decreases relaxing potency of nifedipine by increasing myosin light chain phosphorylation
    • 1-adrenoceptor occupancy decreases relaxing potency of nifedipine by increasing myosin light chain phosphorylation. Circ Res 72:1308-1316.
    • (1993) Circ Res , vol.72 , pp. 1308-1316
    • Ratz, P.J.1
  • 295
    • 0025320531 scopus 로고
    • 1-adrenoceptor-mediated second messenger responses in rat cerebral cortex slices
    • 1-adrenoceptor-mediated second messenger responses in rat cerebral cortex slices. Br J Pharmacol 100:3-4.
    • (1990) Br J Pharmacol , vol.100 , pp. 3-4
    • Robinson, J.P.1    Kendall, D.A.2
  • 299
    • 0028886201 scopus 로고
    • REM sleep inhibition by desipramine: Evidence for an α-1 adrenergic mechanism
    • Ross RJ, Gresch PJ, Ball WA, Sanford LD, Morrison AR (1995): REM sleep inhibition by desipramine: Evidence for an α-1 adrenergic mechanism. Brain Res 701:129-134.
    • (1995) Brain Res , vol.701 , pp. 129-134
    • Ross, R.J.1    Gresch, P.J.2    Ball, W.A.3    Sanford, L.D.4    Morrison, A.R.5
  • 301
    • 0019972619 scopus 로고
    • Receptor interactions of imidazolines. IX. Cirazoline is an alpha-1 adrenergic agonist and an alpha-2 adrenergic antagonist
    • Ruffolo RR Jr, Waddell JE (1982): Receptor interactions of imidazolines. IX. Cirazoline is an alpha-1 adrenergic agonist and an alpha-2 adrenergic antagonist. J Pharmacol Exp Ther 222:29-36.
    • (1982) J Pharmacol Exp Ther , vol.222 , pp. 29-36
    • Ruffolo Jr., R.R.1    Waddell, J.E.2
  • 302
    • 0021171287 scopus 로고
    • Possible relationship between receptor reserve and the differential antagonism of alpha-1 and alpha-2 adrenoceptor-mediated pressor responses by calcium channel antagonists in the pithed rat
    • Ruffolo RR Jr, Morgan EL, Messick K (1984): Possible relationship between receptor reserve and the differential antagonism of alpha-1 and alpha-2 adrenoceptor-mediated pressor responses by calcium channel antagonists in the pithed rat. J Pharmacol Exp Ther 230:587-594.
    • (1984) J Pharmacol Exp Ther , vol.230 , pp. 587-594
    • Ruffolo Jr., R.R.1    Morgan, E.L.2    Messick, K.3
  • 304
    • 0029113808 scopus 로고
    • α- And β-Adrenoceptors: From the gene to the clinic. 2. Structure-activity relationships and therapeutic applications
    • Ruffolo RR Jr, Bondinell WE, Hieble JP (1995a): α- and β-Adrenoceptors: From the gene to the clinic. 2. Structure-activity relationships and therapeutic applications. J Med Chem 38:3415-3444.
    • (1995) J Med Chem , vol.38 , pp. 3415-3444
    • Ruffolo Jr., R.R.1    Bondinell, W.E.2    Hieble, J.P.3
  • 306
    • 0028174149 scopus 로고
    • 1-adrenoceptors in rat myocardial tissue after alkylation with phenoxybenzamine
    • 1-adrenoceptors in rat myocardial tissue after alkylation with phenoxybenzamine. Eur J Pharmacol 266:35-42.
    • (1994) Eur J Pharmacol , vol.266 , pp. 35-42
    • Sallés, J.1    Gascón, S.2    Ivorra, D.3    Badia, A.4
  • 307
    • 0030431042 scopus 로고    scopus 로고
    • Alpha-1 adrenoceptor subtypes involved in mediating adrenergically induced antinatriuresis and antidiuresis in two kidney, one clip Goldblatt and deoxycorticosterone acetatesalt hypertensive rats
    • Sattar MA, Johns EJ (1996): Alpha-1 adrenoceptor subtypes involved in mediating adrenergically induced antinatriuresis and antidiuresis in two kidney, one clip Goldblatt and deoxycorticosterone acetatesalt hypertensive rats. J Pharmacol Exp Ther 277:245-252.
    • (1996) J Pharmacol Exp Ther , vol.277 , pp. 245-252
    • Sattar, M.A.1    Johns, E.J.2
  • 309
    • 0019723906 scopus 로고
    • Midodrine: A new agent in the management of idiopathic orthostatic hypotension and Shy-Drager syndrome
    • Schirger A, Sheps SG, Thomas JE, Fealey RD (1981): Midodrine: A new agent in the management of idiopathic orthostatic hypotension and Shy-Drager syndrome, Mayo Clin Proc 56:429-433.
    • (1981) Mayo Clin Proc , vol.56 , pp. 429-433
    • Schirger, A.1    Sheps, S.G.2    Thomas, J.E.3    Fealey, R.D.4
  • 310
    • 0030069240 scopus 로고    scopus 로고
    • 1A-adrenoceptor antagonist: Analysis of a multicentre, open-label study assessing the long-term efficacy and safety in patients with benign prostatic obstruction (symptomatic BPH)
    • European Tamsulosin Study Group
    • 1A-adrenoceptor antagonist: Analysis of a multicentre, open-label study assessing the long-term efficacy and safety in patients with benign prostatic obstruction (symptomatic BPH). Eur Urol 29:145-154.
    • (1996) Eur Urol , vol.29 , pp. 145-154
    • Schulman, C.C.1    Cortvriend, J.2    Jonas, U.3    Lock, T.M.T.W.4    Vaage, S.5    Speakman, M.J.6
  • 311
    • 0025868331 scopus 로고
    • Differences between full and partial α-adrenoceptor agonists in eliciting phasic and tonic types of responses in the longitudinal smooth muscle of the rat portal vein
    • Schwietert HR, Wilhelm D, Wilffert B, van Zwieten PA (1991): Differences between full and partial α-adrenoceptor agonists in eliciting phasic and tonic types of responses in the longitudinal smooth muscle of the rat portal vein. Naunyn-Schmiedeberg Arch Pharmacol 344:206-212.
    • (1991) Naunyn-Schmiedeberg Arch Pharmacol , vol.344 , pp. 206-212
    • Schwietert, H.R.1    Wilhelm, D.2    Wilffert, B.3    Van Zwieten, P.A.4
  • 312
    • 0027288774 scopus 로고
    • Adrenoceptors as models for G protein-coupled receptors: Structure, function and regulation
    • Schwinn DA (1993): Adrenoceptors as models for G protein-coupled receptors: Structure, function and regulation. Br J Anaesth 71:77-85.
    • (1993) Br J Anaesth , vol.71 , pp. 77-85
    • Schwinn, D.A.1
  • 316
    • 0026652997 scopus 로고
    • Effect of the optical isomers of YM-12617 on increased intra-urethral pressure induced by phenylephrine in anaesthetized dogs
    • Shihasaki M, Sudoh K, Inagaki O, Uchida W, Honda K (1992): Effect of the optical isomers of YM-12617 on increased intra-urethral pressure induced by phenylephrine in anaesthetized dogs. J Anton Pharmacol 12:263-268.
    • (1992) J Anton Pharmacol , vol.12 , pp. 263-268
    • Shihasaki, M.1    Sudoh, K.2    Inagaki, O.3    Uchida, W.4    Honda, K.5
  • 318
    • 0019488885 scopus 로고
    • Comparison of pre- And post-synaptic α-adrenoceptor blocking effects of E-643 in the isolated vas deferens of the rat
    • Shoji T (1981): Comparison of pre- and post-synaptic α-adrenoceptor blocking effects of E-643 in the isolated vas deferens of the rat. Jap J Pharmacol 31:361-368.
    • (1981) Jap J Pharmacol , vol.31 , pp. 361-368
    • Shoji, T.1
  • 319
    • 12644259518 scopus 로고
    • 1-adrenoceptor agonist action of chloroethylclonidine in the rat anococcygeus muscle
    • 1-adrenoceptor agonist action of chloroethylclonidine in the rat anococcygeus muscle. Br J Pharmacol 110 (Suppl):125.
    • (1993) Br J Pharmacol , vol.110 , Issue.SUPPL. , pp. 125
    • Sithers, A.J.1    Marshall, R.W.2    Spriggs, L.B.3
  • 322
    • 0025104014 scopus 로고
    • 1-adrenoceptor antagonist) and the role of α-adrenoceptor stimulation and blockade on atrioventricular conduction
    • 1-adrenoceptor antagonist) and the role of α-adrenoceptor stimulation and blockade on atrioventricular conduction. J Cardiovasc Pharmacol 16:824-830.
    • (1990) J Cardiovasc Pharmacol , vol.16 , pp. 824-830
    • Spiers, J.P.1    Harron, D.W.G.2    Wilson, R.3    Allen, J.D.4
  • 323
    • 0007009119 scopus 로고
    • Stereoselective discrimination of serotoninergic 5HT-1A and 5HT-1B binding sites using the enantiomers of spiroxatrine and WB-4101
    • Stanisic D, Hancock AA, Meyer M, DeBernardis JF (1988): Stereoselective discrimination of serotoninergic 5HT-1A and 5HT-1B binding sites using the enantiomers of spiroxatrine and WB-4101. FASEB J 2:A-1399.
    • (1988) FASEB J , vol.2
    • Stanisic, D.1    Hancock, A.A.2    Meyer, M.3    DeBernardis, J.F.4
  • 325
    • 0016198717 scopus 로고
    • Comparison of the effects of clonidine on pre- And post-synaptic adrenoceptors in the rabbit pulmonary artery
    • Starke K, Montel J, Gayk W, Merker R (1974): Comparison of the effects of clonidine on pre- and post-synaptic adrenoceptors in the rabbit pulmonary artery. Naunyn-Schmiedeberg Arch Pharmacol 285:133-150.
    • (1974) Naunyn-Schmiedeberg Arch Pharmacol , vol.285 , pp. 133-150
    • Starke, K.1    Montel, J.2    Gayk, W.3    Merker, R.4
  • 331
    • 1842395865 scopus 로고
    • 1-Adrenoceptor subtype affinities of tamsulosin metabolites
    • 1-Adrenoceptor subtype affinities of tamsulosin metabolites. Br J Pharmacol 116:207P.
    • (1995) Br J Pharmacol , vol.116
    • Taguchi, K.1    Michel, M.C.2
  • 336
    • 0028170803 scopus 로고
    • 1-adrenoceptor subtypes in human prostate: Comparison with those in rat vas deferens and spleen
    • 1-adrenoceptor subtypes in human prostate: Comparison with those in rat vas deferens and spleen. Eur J Pharmacol 265:61-66.
    • (1994) Eur J Pharmacol , vol.265 , pp. 61-66
    • Teng, D.-M.1    Guh, J.-H.2    Ko, F.-N.3
  • 337
    • 0029656277 scopus 로고
    • 1-adrenoceptors in the reduction of external carotid blood flow induced by buspirone and ipsapirone in the dog
    • 1-adrenoceptors in the reduction of external carotid blood flow induced by buspirone and ipsapirone in the dog. Life Sci 58:63-73.
    • (1995) Life Sci , vol.58 , pp. 63-73
    • Terrón, J.A.1    Ramirez-San Juan, E.2    Hong, E.3    Villalón, C.M.4
  • 343
    • 12644310322 scopus 로고    scopus 로고
    • Functional antagonistic activity of Rec 15/2739, a novel alpha-1 antagonist selective for the lower urinary tract, on noradrenaline-induced contraction of human prostate and mesenteric artery
    • Testa R, Guarneri L, Taddei C, Poggesi E, Angelico P , Sartani A, Leonards A, Gofrit ON, Meretyk S, Gaine M (1996): Functional antagonistic activity of Rec 15/2739, a novel alpha-1 antagonist selective for the lower urinary tract, on noradrenaline-induced contraction of human prostate and mesenteric artery. J Pharmacol Exp Ther 277:1237-1246.
    • (1996) J Pharmacol Exp Ther , vol.277 , pp. 1237-1246
    • Testa, R.1    Guarneri, L.2    Taddei, C.3    Poggesi, E.4    Angelico, P.5    Sartani, A.6    Leonards, A.7    Gofrit, O.N.8    Meretyk, S.9    Gaine, M.10
  • 344
    • 0026507061 scopus 로고
    • 1-adrenoceptor antagonist activity of the anti-arrhythmic drug, abanoquil (UK-52,046), without reduction in blood pressure in man
    • 1-adrenoceptor antagonist activity of the anti-arrhythmic drug, abanoquil (UK-52,046), without reduction in blood pressure in man. Br J Clin Pharmacol 33:405-409.
    • (1992) Br J Clin Pharmacol , vol.33 , pp. 405-409
    • Tham, T.C.I.1    Guy, S.2    Shanks, S.G.3    Harror, D.W.G.4
  • 348
    • 0029417102 scopus 로고
    • 1-adrenoceptor agonist, SDZ NV1-085, behaves as a potent, competitive antagonist of 5-hydroxytryptamine-induced contraction of rat aorta
    • 1-adrenoceptor agonist, SDZ NV1-085, behaves as a potent, competitive antagonist of 5-hydroxytryptamine-induced contraction of rat aorta. Eur J Pharmacol 287:309-312.
    • (1995) Eur J Pharmacol , vol.287 , pp. 309-312
    • Van der Graaf, P.H.1    Apaydin, S.2    Saxena, P.R.3
  • 350
    • 0030056471 scopus 로고    scopus 로고
    • 1-adrenoceptor antagonists on noradrenaline-mediated contraction of rat small mesenteric artery
    • 1-adrenoceptor antagonists on noradrenaline-mediated contraction of rat small mesenteric artery. Br J Pharmacol 118:1308-1316.
    • (1996) Br J Pharmacol , vol.118 , pp. 1308-1316
    • Van der Graaf, P.H.1    Shankley, N.P.2    Black, J.W.3
  • 351
    • 0028879397 scopus 로고
    • Vascular alpha-l adrenergic receptor subtypes in the regulation of arterial blood pressure
    • Vargas HM, Gorman AJ (1995): Vascular alpha-l adrenergic receptor subtypes in the regulation of arterial blood pressure. Life Sci 57:2291-2308.
    • (1995) Life Sci , vol.57 , pp. 2291-2308
    • Vargas, H.M.1    Gorman, A.J.2
  • 354
    • 0023010594 scopus 로고
    • The cardiovascular effects of trimazosin and prazosin in the rabbit
    • Vincent J, Hamilton CA, Reid JL (1986): The cardiovascular effects of trimazosin and prazosin in the rabbit. Clin Exp Pharmacol Physiol 13:593-608.
    • (1986) Clin Exp Pharmacol Physiol , vol.13 , pp. 593-608
    • Vincent, J.1    Hamilton, C.A.2    Reid, J.L.3
  • 357
    • 0019778150 scopus 로고
    • 3H]WB-4101) to multiple sites in human brain
    • 3H]WB-4101) to multiple sites in human brain. Biochem Pharmacol 30:3115-3120.
    • (1981) Biochem Pharmacol , vol.30 , pp. 3115-3120
    • Weinreich, P.1    Seeman, P.2
  • 359
    • 0027477729 scopus 로고
    • Alfuzosin: A review of its pharmacodynamic and pharmacokinetic properties, and therapeutic potential in benign prostatic hyperplasia
    • Wilde MI, Fitton A, McTavish D (1993): Alfuzosin: A review of its pharmacodynamic and pharmacokinetic properties, and therapeutic potential in benign prostatic hyperplasia. Drugs 45:410-429.
    • (1993) Drugs , vol.45 , pp. 410-429
    • Wilde, M.I.1    Fitton, A.2    McTavish, D.3
  • 362
    • 0027501466 scopus 로고
    • Pharmacology of 2-amino-l,4-dihydro-4-(2-{4-[4-(2-methoxyphenyl)-l-piperazinyl] butylsulfinyl} phenyl) -6-methyl-5-nitro-3-pyridine carboxylic acid methyl ester (XB513), a novel calcium agonist with alpha-1 adrenergic receptor antagonistic property
    • Wong PC, Aldrich PE, Chiu AT, Earl RA, Hart SD, Johnson AL, Ma P, McCall DE, Price WA Jr, Smith RD, Wexler RR, Timmermans PBMWM (1993): Pharmacology of 2-amino-l,4-dihydro-4-(2-{4-[4-(2-methoxyphenyl)-l-piperazinyl] butylsulfinyl} phenyl) -6-methyl-5-nitro-3-pyridine carboxylic acid methyl ester (XB513), a novel calcium agonist with alpha-1 adrenergic receptor antagonistic property. J Pharmacol Exp Ther 265:1088-1095.
    • (1993) J Pharmacol Exp Ther , vol.265 , pp. 1088-1095
    • Wong, P.C.1    Aldrich, P.E.2    Chiu, A.T.3    Earl, R.A.4    Hart, S.D.5    Johnson, A.L.6    Ma, P.7    McCall, D.E.8    Price Jr., W.A.9    Smith, R.D.10    Wexler, R.R.11    Timmermans, P.B.M.W.M.12
  • 363
    • 12644300651 scopus 로고    scopus 로고
    • 1-AR) with chloroethylclonidine (CEC): A kinetic analysis
    • 1-AR) with chloroethylclonidine (CEC): A kinetic analysis. FASEB J 10:A418.
    • (1996) FASEB J , vol.10
    • Xiao, L.1    Makoid, M.2    Jeffries, W.B.3
  • 368
    • 0027446196 scopus 로고
    • Role of adrenoceptors in the proximal urethral function of female and male rabbits using an in vivo model of isovolumetric pressure generation
    • Yamaguchi T, Kitada S, Osada Y (1993): Role of adrenoceptors in the proximal urethral function of female and male rabbits using an in vivo model of isovolumetric pressure generation. Neurourol Urodyn 12:49-57.
    • (1993) Neurourol Urodyn , vol.12 , pp. 49-57
    • Yamaguchi, T.1    Kitada, S.2    Osada, Y.3
  • 369
    • 0028795596 scopus 로고
    • 1 adrenergic stimulation: A potential role for receptor mediated activation of sarcolemmal sodium-hydrogen exchange
    • 1 adrenergic stimulation: A potential role for receptor mediated activation of sarcolemmal sodium-hydrogen exchange. Cardiovasc Res 29:222-230.
    • (1995) Cardiovasc Res , vol.29 , pp. 222-230
    • Yasutake, M.1    Avkiran, M.2
  • 370
    • 0026610837 scopus 로고
    • 3H](o-ethoxyphenoxy)ethyl]amino]-propyl-2-methoxybenzenesulfonamide HCL, a potent and selective alpha-1 adrenoceptor radioligand
    • 3H](o-ethoxyphenoxy)ethyl]amino]-propyl]-2-methoxybenzenesulfonamide HCL, a potent and selective alpha-1 adrenoceptor radioligand. J Pharmacol Exp Ther 263:201-206.
    • (1992) J Pharmacol Exp Ther , vol.263 , pp. 201-206
    • Yazawa, H.1    Takanashi, M.2    Sudoh, K.3    Inagaki, O.4    Honda, K.5
  • 371
    • 0025335926 scopus 로고
    • Central sympathoinhibitory action of a new type of alpha-1 adrenoceptor antagonist, YM-617in rats
    • Yoshioka M, Togashi H, Abe M, Ikeda T, Matsumoto M, Saito H (1990): Central sympathoinhibitory action of a new type of alpha-1 adrenoceptor antagonist, YM-617in rats. J Pharmacol Exp Ther 253:427-431.
    • (1990) J Pharmacol Exp Ther , vol.253 , pp. 427-431
    • Yoshioka, M.1    Togashi, H.2    Abe, M.3    Ikeda, T.4    Matsumoto, M.5    Saito, H.6
  • 372
    • 0028058799 scopus 로고
    • The electrophysiological effects of dicentrine on the conduction system of rabbit heart
    • Young ML, Su MJ, Wu MH, Chen CC (1994): The electrophysiological effects of dicentrine on the conduction system of rabbit heart. Br J Pharmacol 113:69-76.
    • (1994) Br J Pharmacol , vol.113 , pp. 69-76
    • Young, M.L.1    Su, M.J.2    Wu, M.H.3    Chen, C.C.4
  • 375
    • 33749134608 scopus 로고    scopus 로고
    • Pharmacological studies on the potency and selectivity of BMY 7378 for alpha-1 adrenoceptor (AR) subtypes in pithed rat
    • Zhou L, Vargas HM (1996a): Pharmacological studies on the potency and selectivity of BMY 7378 for alpha-1 adrenoceptor (AR) subtypes in pithed rat. FASEB J 10:A425.
    • (1996) FASEB J , vol.10
    • Zhou, L.1    Vargas, H.M.2
  • 376
    • 0029949772 scopus 로고    scopus 로고
    • 1D-adrenoceptors have a role in the pressor response to phenylephrine in the pithed rat
    • 1D-adrenoceptors have a role in the pressor response to phenylephrine in the pithed rat. Eur J Pharmacol 305:173-176.
    • (1996) Eur J Pharmacol , vol.305 , pp. 173-176
    • Zhou, L.1    Vargas, H.M.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.