A convenient, high-throughput assay for measuring the relative cell permeability of synthetic compounds

Nature Protocols

Volumn 2, Issue 1, 2007, Pages 23-30

  Yu, Peng ^a   Liu, Bo ^a   Kodadek, Thomas ^a  

^a UNIVERSITY OF TEXAS SOUTHWESTERN MEDICAL CENTER   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

DEXAMETHASONE; DEXAMETHASONE DERIVATIVE; DNA BINDING PROTEIN; GLUCOCORTICOID RECEPTOR; HYBRID PROTEIN; LUCIFERASE; PROTEIN VP16; GAL4 PROTEIN, S CEREVISIAE; ORGANIC COMPOUND; SACCHAROMYCES CEREVISIAE PROTEIN; TRANSCRIPTION FACTOR; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; CELL MEMBRANE PERMEABILITY; COMBINATORIAL LIBRARY; DRUG CONJUGATION; DRUG RECEPTOR BINDING; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; DRUG TRANSPORT; GENE EXPRESSION; HIGH THROUGHPUT SCREENING; IC 50; INTRACELLULAR TRANSPORT; MAMMAL CELL; PRIORITY JOURNAL; PROTEIN DOMAIN; QUANTITATIVE ANALYSIS; REPORTER GENE; COMBINATORIAL CHEMISTRY; CYTOLOGY; DRUG EFFECT; ENZYME ACTIVATION; METABOLISM; METHODOLOGY; PHYSIOLOGY;

MAMMALIA;

CELL MEMBRANE PERMEABILITY; COMBINATORIAL CHEMISTRY TECHNIQUES; CYTOLOGICAL TECHNIQUES; DEXAMETHASONE; ENZYME ACTIVATION; LUCIFERASES; ORGANIC CHEMICALS; SACCHAROMYCES CEREVISIAE PROTEINS; TRANSCRIPTION FACTORS;

EID: 34347273069     PISSN: 17542189     EISSN: 17502799     Source Type: Journal    
DOI: 10.1038/nprot.2007.1     Document Type: Article

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