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note
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Analogy to conditions successfully used for arylation of imidazoles and benzimidazoles in ref 12c.
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33
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33845263579
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note
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3/heptane.
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34
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33751210583
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The only two known related examples of C-H homocoupling of heterocycles: (a) a Cu-mediated dimerization of benzothiazole: Chodowska-Palicka, J.; Nilsson, M. Synthesis 1974, 128-129.
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(b) Recently described Pd-catalyzed dimerization of bromothiophenes in the presence of AgF: Takahashi, M.; Masui, K.; Sekiguchi, H.; Kobayashi, N.; Mori, A.; Funahashi, M.; Tamaoki, N. J. Am. Chem. Soc. 2006, 128, 10930-10933.
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Tamaoki, N.7
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