Tramadol, fentanyl and sufentanil but not morphine block voltage-operated sodium channels

Pain

Volumn 126, Issue 1-3, 2006, Pages 234-244

  Haeseler, Gertrud ^a   Foadi, Nilufar ^a   Ahrens, Jörg ^a   Dengler, Reinhard ^a   Hecker, Hartmut ^a   Leuwer, Martin ^b  

^a HANNOVER MEDICAL SCHOOL   (Germany)

^b UNIVERSITY OF LIVERPOOL   (United Kingdom)

Author keywords

Local anesthetic like action; Opioids; Sodium channels; Voltage operated

Indexed keywords

FENTANYL; MORPHINE; SUFENTANIL; TRAMADOL; VOLTAGE GATED SODIUM CHANNEL;

ANESTHESIA MECHANISM; ANTINOCICEPTION; ARTICLE; CELL MEMBRANE DEPOLARIZATION; CONTROLLED STUDY; DRUG BINDING SITE; DRUG INHIBITION; DRUG POTENCY; DRUG RECEPTOR BINDING; EMBRYO; HUMAN; HUMAN CELL; HYPERPOLARIZATION; IC 50; NERVE FIBER; NERVE POTENTIAL; PREPULSE INHIBITION; PRIORITY JOURNAL; RECEPTOR AFFINITY; RECEPTOR BLOCKING; SODIUM CURRENT;

ANALGESICS, OPIOID; CELL LINE; ELECTRIC CONDUCTIVITY; FENTANYL; HUMANS; ION CHANNEL GATING; MORPHINE; NERVE TISSUE PROTEINS; SODIUM CHANNEL BLOCKERS; SODIUM CHANNELS; SUFENTANIL; TRAMADOL;

EID: 33750967055     PISSN: 03043959     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.pain.2006.07.003     Document Type: Article

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