Identification of structures within GABAA receptor α subunits that regulate the agonist action of pentobarbital

Journal of Pharmacology and Experimental Therapeutics

Volumn 318, Issue 3, 2006, Pages 1094-1101

  Drafts, Brandon C ^a   Fisher, Janet L ^a  

^a UNIVERSITY OF SOUTH CAROLINA SCHOOL OF MEDICINE   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

4 AMINOBUTYRIC ACID; 4 AMINOBUTYRIC ACID A RECEPTOR; 4 AMINOBUTYRIC ACID A RECEPTOR STIMULATING AGENT; ETOMIDATE; PENTOBARBITAL; PROPOFOL; RECEPTOR SUBUNIT; 4 AMINOBUTYRIC ACID RECEPTOR STIMULATING AGENT; PROTEIN SUBUNIT;

ALLOSTERISM; AMINO TERMINAL SEQUENCE; ANIMAL CELL; ANIMAL EXPERIMENT; ARTICLE; CHIMERA; CONTROLLED STUDY; DRUG ACTIVATION; DRUG EFFICACY; DRUG IDENTIFICATION; DRUG INHIBITION; DRUG MECHANISM; DRUG STRUCTURE; ELECTROPHYSIOLOGY; FIBROBLAST; MOUSE; MUTATION; NONHUMAN; PATCH CLAMP; PRIORITY JOURNAL; PROTEIN DOMAIN; ANIMAL; CELL LINE; CHEMISTRY; DRUG POTENTIATION; STRUCTURE ACTIVITY RELATION;

ALLOSTERIC REGULATION; ANIMALS; CELL LINE; ETOMIDATE; GABA AGONISTS; GAMMA-AMINOBUTYRIC ACID; MICE; PENTOBARBITAL; PROTEIN SUBUNITS; RECEPTORS, GABA-A; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 33747598041     PISSN: 00223565     EISSN: 15210103     Source Type: Journal    
DOI: 10.1124/jpet.106.104844     Document Type: Article

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