Recent development in the field of dual COX / 5-LOX inhibitors

Mini-Reviews in Medicinal Chemistry

Volumn 4, Issue 6, 2004, Pages 633-638

  Julémont, Fabien ^a   Dogné, Jean Michel ^a   Pirotte, Bernard ^a   de Leval, Xavier ^a  

^a UNIVERSITY OF LIÈGE   (Belgium)

Author keywords

Cancer; Cyclooxygenases; Dual inhibitors; Inflammation; Leukotrienes

Indexed keywords

6 [[3 FLUORO 5 (3,4,5,6 TETRAHYDRO 4 METHOXY 2H PYRAN 4 YL)]PHENOXYMETHYL] 1 METHYL 2 QUINOLONE; ARACHIDONIC ACID; CELECOXIB; DARBUFELONE; DIPEPTIDASE; ENZYME INHIBITOR; FENAMIC ACID DERIVATIVE; GAMMA GLUTAMYLTRANSFERASE; HYDROLASE; HYDROXYUREA; INDOMETACIN DERIVATIVE; LEUKOTRIENE DERIVATIVE; LICOFELONE; LIPOXYGENASE; LIPOXYGENASE INHIBITOR; N [5 (4 FLUOROPHENOXY) 2 THIENYL]METHANESULFONAMIDE; NONSTEROID ANTIINFLAMMATORY AGENT; PROSTAGLANDIN; PROSTAGLANDIN E2; PROSTAGLANDIN H2; PROSTAGLANDIN SYNTHASE; PROSTAGLANDIN SYNTHASE INHIBITOR; PROSTANOID; PYRROLIZINE DERIVATIVE; R 380; SULFONAMIDE; TEBUFELONE; TEPOXALIN; THROMBOXANE; UNCLASSIFIED DRUG; UNINDEXED DRUG;

ANTIINFLAMMATORY ACTIVITY; ARACHIDONIC ACID METABOLISM; CARCINOGENESIS; CLINICAL TRIAL; COLON CANCER; DRUG SAFETY; DRUG STRUCTURE; DRUG TARGETING; ENZYME ACTIVITY; ENZYME INHIBITION; GASTROINTESTINAL SYMPTOM; HUMAN; INFLAMMATION; NONHUMAN; PROSTATE CANCER; PROTEIN TARGETING; SHORT SURVEY; SIGNAL TRANSDUCTION; STRUCTURE ANALYSIS;

EID: 3242715817     PISSN: 13895575     EISSN: None     Source Type: Journal    
DOI: 10.2174/1389557043403747     Document Type: Short Survey

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