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Bioorganic and Medicinal Chemistry Letters

Volumn 12, Issue 5, 2002, Pages 779-782

Synthesis and activity of a new methoxytetrahydropyran derivative as dual cyclooxygenase-2/5-lipoxygenase inhibitor

(12) Barbey, Sabine a Goossens, Laurence b Taverne, Thierry b Cornet, Joséphine b Choesmel, Valérie a Rouaud, Céline a Gimeno, Gilles a Yannic Arnoult, Sylvie a Michaux, Catherine c Charlier, Caroline c Houssin, Raymond b Hénichart, Jean Pierre b

a Laboratoires Innothera (France)

b Faculté des Sciences Pharmaceutiques et Biologiques Université de Lille (France)

c UNIVERSITY OF NAMUR (Belgium)

Author keywords

[No Author keywords available]

Indexed keywords

ANTIINFLAMMATORY AGENT; ARACHIDONATE 5 LIPOXYGENASE; CYCLOOXYGENASE 2 INHIBITOR; ENZYME INHIBITOR; TETRAHYDROPYRAN DERIVATIVE;

ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DRUG ACTIVITY; DRUG POTENCY; DRUG SYNTHESIS; ENZYME INHIBITION; IN VITRO STUDY; IN VIVO STUDY; INFLAMMATION; MALE; NONHUMAN; PHARMACOPHORE; RAT; STRUCTURE ACTIVITY RELATION;

ANIMALS; ARACHIDONATE 5-LIPOXYGENASE; CELLS, CULTURED; CYCLOOXYGENASE 2; CYCLOOXYGENASE 2 INHIBITORS; CYCLOOXYGENASE INHIBITORS; DINOPROSTONE; GRANULOCYTES; INHIBITORY CONCENTRATION 50; ISOENZYMES; LIPOXYGENASE INHIBITORS; MALE; MONOCYTES; OSTEOSARCOMA; PROSTAGLANDIN-ENDOPEROXIDE SYNTHASES; PYRAZOLES; RATS; RATS, WISTAR; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONES;

SIGANUS;

EID: 0037060906 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/S0960-894X(02)00013-6 Document Type: Article

Times cited : (81)

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