Structural analysis of caspase-1 inhibitors derived from Tethering

Acta Crystallographica Section F: Structural Biology and Crystallization Communications

Volumn 61, Issue 5, 2005, Pages 451-458

  Fahr, Bruce T ^a   Sopko, Michelle M ^a   Lam, Joni W ^a   O'Brien, Tom ^a   Waal, Nathan D ^a   Pham, Phuongly ^a   Purkey, Hans E ^a   Raimundo, Brian C ^a   Romanowski, Michael J ^a  

^a Sunesis Pharmaceuticals Inc   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CYSTEINE PROTEINASE INHIBITOR; INTERLEUKIN 1; INTERLEUKIN 1BETA CONVERTING ENZYME; INTERLEUKIN 6;

ARTICLE; BINDING SITE; BLOOD; CHEMICAL STRUCTURE; CHEMISTRY; COMBINATORIAL CHEMISTRY; DRUG ANTAGONISM; DRUG DESIGN; DRUG EFFECT; ENZYMOLOGY; HUMAN; METABOLISM; METHODOLOGY; MONONUCLEAR CELL; PROTEIN BINDING; SOLUBILITY; X RAY CRYSTALLOGRAPHY;

BINDING SITES; CASPASE 1; COMBINATORIAL CHEMISTRY TECHNIQUES; CRYSTALLOGRAPHY, X-RAY; CYSTEINE PROTEINASE INHIBITORS; DRUG DESIGN; HUMANS; INTERLEUKIN-1; INTERLEUKIN-6; LEUKOCYTES, MONONUCLEAR; MODELS, MOLECULAR; PROTEIN BINDING; SOLUBILITY;

EID: 29544442944     PISSN: 17443091     EISSN: 17443091     Source Type: Journal    
DOI: 10.1107/S1744309105010109     Document Type: Article

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