Identification of an inhibitor-binding site to HIV-1 integrase with affinity acetylation and mass spectrometry

Proceedings of the National Academy of Sciences of the United States of America

Volumn 101, Issue 18, 2004, Pages 6894-6899

  Shkriabai, Nick ^a   Patil, Sachindra S ^b   Hess, Sonja ^c   Budihas, Scott R ^b   Craigie, Robert ^c   Burke Jr , Terrence R ^b   Le Grice, Stuart F J ^b   Kvaratskhelia, Mamuka ^a,d  

^a THE OHIO STATE UNIVERSITY WEXNER MEDICAL CENTER   (United States)

^b NATIONAL CANCER INSTITUTE   (United States)

^c NATIONAL INSTITUTE OF DIABETES AND DIGESTIVE AND KIDNEY DISEASES   (United States)

^d OHIO STATE UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ACETIC ACID DERIVATIVE; AMINO ACID; CYSTEINE; INTEGRASE; INTEGRASE INHIBITOR; LIGAND; LYSINE; PEPTIDE; PEPTIDE LIBRARY; POLYCYCLIC AROMATIC HYDROCARBON DERIVATIVE; PROTEIN; TYROSINE; VIRUS ENZYME;

ACETYLATION; AFFINITY ACETYLATION; ARTICLE; BINDING AFFINITY; BINDING SITE; CONTROLLED STUDY; ENZYME BINDING; ENZYME INHIBITION; HUMAN IMMUNODEFICIENCY VIRUS 1; LIGAND BINDING; LIGAND PROTEIN INTERACTION; MASS SPECTROMETRY; NONHUMAN; PRIORITY JOURNAL; PROTEIN PROTEIN INTERACTION;

ACETYLATION; BINDING SITES; ENZYME INHIBITORS; HIV INTEGRASE; HIV-1; PEPTIDES; SPECTROMETRY, MASS, MATRIX-ASSISTED LASER DESORPTION-IONIZATION;

HUMAN IMMUNODEFICIENCY VIRUS; HUMAN IMMUNODEFICIENCY VIRUS 1; RNA VIRUSES;

EID: 2342569518     PISSN: 00278424     EISSN: None     Source Type: Journal    
DOI: 10.1073/pnas.0400873101     Document Type: Article

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