The ratio of constitutive androstane receptor to pregnane X receptor determines the activity of guggulsterone against the Cyp2b10 promoter

Journal of Pharmacology and Experimental Therapeutics

Volumn 314, Issue 1, 2005, Pages 120-127

  Ding, Xunshan ^a   Staudinger, Jeff L ^a  

^a UNIVERSITY OF KANSAS   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CELL NUCLEUS RECEPTOR; CONSTITUTIVE ANDROSTANE RECEPTOR; CYTOCHROME P450 2B10; GUGGULSTERONE; OXIDOREDUCTASE; PREGNANE X RECEPTOR; UNCLASSIFIED DRUG;

AGONIST; ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; ASSAY; CIRCADIAN RHYTHM; CRYSTAL STRUCTURE; DRUG ACTIVITY; DRUG MECHANISM; DRUG METABOLISM; ETHNIC GROUP; GENE EXPRESSION; GENE REPRESSION; INHIBITION KINETICS; LIVER CELL; MOLECULAR MECHANICS; MOUSE; NONHUMAN; NUCLEOTIDE SEQUENCE; POPULATION; PRIORITY JOURNAL; PROMOTER REGION; PROTEIN EXPRESSION; TWO HYBRID SYSTEM;

ANIMALS; ARYL HYDROCARBON HYDROXYLASES; BLOTTING, NORTHERN; CELLS, CULTURED; GENE EXPRESSION; GENES, REPORTER; LUCIFERASES; MICE; MICE, KNOCKOUT; PLASMIDS; PREGNENEDIONES; PROMOTER REGIONS (GENETICS); RECEPTORS, CYTOPLASMIC AND NUCLEAR; RECEPTORS, STEROID; REVERSE TRANSCRIPTASE POLYMERASE CHAIN REACTION; STEROID HYDROXYLASES; TRANSCRIPTION FACTORS; TRANSFECTION;

EID: 23044477294     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: 10.1124/jpet.105.085225     Document Type: Article

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