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Volumn 13, Issue 13, 2005, Pages 4200-4208

Synthesis of a C-terminally biotinylated macrocyclic peptide mimetic exhibiting high Grb2 SH2 domain-binding affinity

(8) Shi, Zhen Dan a Liu, Hongpeng b Zhang, Manchao b Worthy, Karen M c Bindu, Lakshman c Yang, Dajun b Fisher, Robert J c Burke Jr , Terrence R a

a NATIONAL CANCER INSTITUTE (United States)

b UNIVERSITY OF MICHIGAN MEDICAL SCHOOL (United States)

c SAIC FREDERICK INC (United States)

Author keywords

Biotin conjugate; Grb2 SH2 Domain; Macrocycle

Indexed keywords

18 (2 AMINO 2 OXOETHYL) 14 (1 NAPHTHALENYLMETHYL) 8,17,20 TRIOXO 10 [4 (PHOSPHONOMETHYL)PHENYL] 7,16,19 TRIAZASPIRO[5.14]EICOS 11 EN 9 ACETIC ACID; MACROCYCLIC COMPOUND; PEPTIDE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; BIOTINYLATION; CARBOXY TERMINAL SEQUENCE; DRUG BINDING; DRUG POTENCY; DRUG SCREENING; DRUG SPECIFICITY; DRUG SYNTHESIS; HUMAN; HUMAN CELL;

ADAPTOR PROTEINS, SIGNAL TRANSDUCING; ANTINEOPLASTIC AGENTS; BIOTINYLATION; BREAST NEOPLASMS; CYCLIZATION; FEMALE; GRB2 ADAPTOR PROTEIN; HUMANS; LIGANDS; MODELS, MOLECULAR; MOLECULAR MIMICRY; PEPTIDE FRAGMENTS; PHOSPHOTYROSINE; PROTEIN BINDING; RECEPTOR, ERBB-2; SRC HOMOLOGY DOMAINS; STRUCTURE-ACTIVITY RELATIONSHIP; TUMOR CELLS, CULTURED;

EID: 20344377158 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/j.bmc.2005.04.028 Document Type: Article

Times cited : (13)

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