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Current Medicinal Chemistry

Volumn 7, Issue 10, 2000, Pages 1081-1100

Recent advances in the design and synthesis of SH2 inhibitors of Src, Grb2 and ZAP-70

(1) Vu, C B a

a BIOGEN (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ACETOPHENONE; AMIDE; BENZAMIDE DERIVATIVE; GROWTH RECEPTOR BOUND PROTEIN 2; HYDROXYLAMINE; OXADIAZOLE DERIVATIVE; PHOSPHATASE; PHOSPHOTYROSINE; PROPYLAMINE; PROTEIN TYROSINE KINASE; PROTEIN TYROSINE KINASE INHIBITOR; PYRIDINE DERIVATIVE; THIAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL MODEL; CANCER RESEARCH; CRYSTAL STRUCTURE; DRUG DESIGN; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME ACTIVITY; ENZYME INHIBITION; ENZYME LINKED IMMUNOSORBENT ASSAY; IMMUNOSUPPRESSIVE TREATMENT; KNOCKOUT MOUSE; MEMBRANE PERMEABILITY; MITOGENESIS; MOUSE; NONHUMAN; NUCLEAR MAGNETIC RESONANCE; OSTEOLYSIS; PROTEIN BINDING; PROTEIN PHOSPHORYLATION; PROTEIN PROTEIN INTERACTION; PROTEIN STRUCTURE; REVERSED PHASE HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; REVIEW; SEQUENCE HOMOLOGY; SIGNAL TRANSDUCTION; X RAY CRYSTALLOGRAPHY;

EID: 0033826421 PISSN: 09298673 EISSN: None Source Type: Journal
DOI: 10.2174/0929867003374390 Document Type: Review

Times cited : (44)

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