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Bioorganic and Medicinal Chemistry Letters

Volumn 15, Issue 12, 2005, Pages 3096-3101

Carbonic anhydrase inhibitors. Inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, IX, and XII with Schiff's bases incorporating chromone and aromatic sulfonamide moieties, and their zinc complexes

(6) Puccetti, Luca a Fasolis, Giuseppe a Vullo, Daniela b Chohan, Zahid H c Scozzafava, Andrea b Supuran, Claudiu T b

a Ospedale San Lazzaro (Italy)

b UNIVERSITY OF FLORENCE (Italy)

c BAHAUDDIN ZAKARIYA UNIVERSITY (Pakistan)

Author keywords

[No Author keywords available]

Indexed keywords

ACETAZOLAMIDE; CARBONATE DEHYDRATASE; CARBONATE DEHYDRATASE I; CARBONATE DEHYDRATASE II; CARBONATE DEHYDRATASE INHIBITOR; CHROMONE DERIVATIVE; DICLOFENAMIDE; ETHOXZOLAMIDE; INDISULAM; MAFENIDE; METHAZOLAMIDE; PROTEIN SUBUNIT; SCHIFF BASE; SULFAGUANIDINE; SULFANILAMIDE; SULFONAMIDE; ZINC COMPLEX;

ARTICLE; CHEMICAL REACTION; CYTOSOL; ENZYME INHIBITION; PHYSIOLOGY; STRUCTURE ACTIVITY RELATION; SUBSTITUTION REACTION;

ANTIGENS, NEOPLASM; ANTINEOPLASTIC AGENTS; CARBONIC ANHYDRASE I; CARBONIC ANHYDRASE II; CARBONIC ANHYDRASE INHIBITORS; CARBONIC ANHYDRASES; CELL MEMBRANE; CHROMONES; CYTOSOL; HUMANS; ISOENZYMES; MOLECULAR STRUCTURE; NERVE TISSUE PROTEINS; SCHIFF BASES; STRUCTURE-ACTIVITY RELATIONSHIP; SULFONAMIDES; ZINC COMPOUNDS;

EID: 19944394215 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2005.04.055 Document Type: Article

Times cited : (120)

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