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Volumn 58, Issue 32, 2002, Pages 6413-6432

Chemical synthesis and biological evaluation of novel epothilone B and trans-12,13-cyclopropyl epothilone B analogues

(10) Nicolaou, K C a,b Ritzén, Andreas a,b Namoto, Kenji a,b Buey, Rubén M c Díaz, J Fernando c Andreu, José M c Wartmann, Markus d Altmann, Karl Heinz d O'Brate, Aurora e Giannakakou, Paraskevi e

a SCRIPPS RESEARCH INSTITUTE (United States)

b UNIVERSITY OF CALIFORNIA (United States)

c CENTRO DE INVESTIGACIONES BIOLÓGICAS (Spain)

d NOVARTIS PHARMA AG (Switzerland)

e EMORY UNIVERSITY SCHOOL OF MEDICINE (United States)

Author keywords

Antitumor agents; Chemical synthesis; Epothilones; Structure activity relationships

Indexed keywords

CYCLOPROPANE DERIVATIVE; EPOTHILONE A; EPOTHILONE B; EPOTHILONE DERIVATIVE; MACROCYCLIC COMPOUND; ORGANOTIN COMPOUND; PACLITAXEL; VINYL DERIVATIVE;

ANTINEOPLASTIC ACTIVITY; ARTICLE; CHEMICAL REACTION; CONTROLLED STUDY; DRUG BINDING SITE; DRUG CYTOTOXICITY; DRUG SCREENING; DRUG SYNTHESIS; HUMAN; HUMAN CELL; MICROTUBULE ASSEMBLY; NOZAKI HIYAMA KISHI COUPLING REACTION; PRIORITY JOURNAL; STILLE REACTION; YAMAGUSHI REACTION;

EID: 18544369875 PISSN: 00404020 EISSN: None Source Type: Journal
DOI: 10.1016/S0040-4020(02)00655-5 Document Type: Article

Times cited : (56)

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