Receptor-assisted combinatorial chemistry: Thermodynamics and kinetics in drug discovery

Chemistry - A European Journal

Volumn 11, Issue 6, 2005, Pages 1708-1716

  Cheeseman, Jeremy D ^a   Corbett, Andrew D ^b   Gleason, James L ^a   Kazlauskas, Romas J ^c  

^a MCGILL UNIVERSITY   (Canada)

^b UNIVERSITÉ DE SHERBROOKE   (Canada)

^c UNIVERSITY OF MINNESOTA   (United States)

Author keywords

Combinatorial chemistry; Drug design; Inhibitors; Receptors; Template synthesis

Indexed keywords

REACTION KINETICS; STOICHIOMETRY; SYNTHESIS (CHEMICAL); THERMODYNAMICS;

COMBINATORIAL CHEMISTRY; DRUG DISCOVERY; PSEUDO-DYNAMIC LIBRARIES; RECEPTOR ASSISTANCE;

DRUG PRODUCTS;

RECEPTOR;

COMBINATORIAL CHEMISTRY; DRUG RESEARCH; DRUG SCREENING; DRUG SYNTHESIS; KINETICS; RECEPTOR ASSISTED COMBINATORIAL CHEMISTRY; REVIEW; STOICHIOMETRY; THERMODYNAMICS;

COMBINATORIAL CHEMISTRY TECHNIQUES; DRUG DESIGN; KINETICS; MOLECULAR CONFORMATION; PEPTIDE LIBRARY; RECEPTORS, DRUG; STRUCTURE-ACTIVITY RELATIONSHIP; THERMODYNAMICS;

EID: 15044347857     PISSN: 09476539     EISSN: None     Source Type: Journal    
DOI: 10.1002/chem.200400371     Document Type: Review

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