A novel pesticide-induced conformational state of the oestrogen receptor ligand-binding domain, detected by conformation-specific peptide binding

FEBS Letters

Volumn 579, Issue 2, 2005, Pages 541-548

  Sumbayev, Vadim V ^a   Bonefeld Jørgensen, Eva C ^a   Wind, Troels ^a   Andreasen, Peter A ^a  

^a AARHUS UNIVERSITY   (Denmark)

Author keywords

Endocrine disruptor; Oestrogen; Oestrogen receptor; Phage displayed peptide library

Indexed keywords

4 HYDROXYTAMOXIFEN; ESTRADIOL; ESTROGEN; ESTROGEN RECEPTOR; ETHYLENE DERIVATIVE; PESTICIDE;

ANIMAL CELL; ARTICLE; CHEMICAL INTERACTION; CONFORMATIONAL TRANSITION; CONTROLLED STUDY; HORMONE ACTION; LIGAND BINDING; NONHUMAN; PEPTIDE ANALYSIS; PRIORITY JOURNAL; PROTEIN BINDING; PROTEIN DOMAIN; PROTEIN INTERACTION; TRANSACTIVATION;

AMINO ACID SUBSTITUTION; ANIMALS; BINDING SITES; CHLORINE COMPOUNDS; CHO CELLS; CRICETINAE; CRICETULUS; DICHLORODIPHENYL DICHLOROETHYLENE; ESTRADIOL; ESTROGEN RECEPTOR ALPHA; ESTROGEN RECEPTOR BETA; GENES, REPORTER; LIGANDS; LUCIFERASES; PEPTIDES; PESTICIDES; PROTEIN STRUCTURE, TERTIARY; SELECTIVE ESTROGEN RECEPTOR MODULATORS; TAMOXIFEN; TRANS-ACTIVATION (GENETICS);

EID: 11844294719     PISSN: 00145793     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.febslet.2004.12.025     Document Type: Article

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