Estrogen receptor (ER) modulators each induce distinct conformational changes in ER α and ER β

Proceedings of the National Academy of Sciences of the United States of America

Volumn 96, Issue 7, 1999, Pages 3999-4004

  Paige, Lisa A ^a   Christensen, Dale J ^a   Grøn, Hanne ^a   Norris, John D ^b   Gottlin, Elizabeth B ^a   Padilla, Karen M ^a   Chang, Ching Yi ^b   Ballas, Lawrence M ^a   Hamilton, Paul T ^a   McDonnell, Donald P ^b   Fowlkes, Dana M ^a  

^a Novalon Pharmaceutical Corporation   (United States)

^b DUKE UNIVERSITY MEDICAL CENTER   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

16ALPHA HYDROXYESTRONE; 4 HYDROXYTAMOXIFEN; CLOMIFENE; CONJUGATED ESTROGEN; DIETHYLSTILBESTROL; ESTRADIOL; ESTRIOL; ESTROGEN; ESTROGEN RECEPTOR; FULVESTRANT; NAFOXIDINE; RALOXIFENE; STREPTAVIDIN;

ARTICLE; BINDING SITE; CONFORMATIONAL TRANSITION; DRUG RECEPTOR BINDING; PRIORITY JOURNAL; PROTEIN CONFORMATION; RECEPTOR AFFINITY; RECEPTOR BLOCKING; RECEPTOR INTRINSIC ACTIVITY; STRUCTURE ACTIVITY RELATION;

AMINO ACID SEQUENCE; BINDING SITES; ESTRADIOL; ESTRADIOL CONGENERS; ESTRIOL; ESTROGEN ANTAGONISTS; ESTROGEN RECEPTOR ALPHA; ESTROGEN RECEPTOR BETA; ESTROGENS; HUMANS; MOLECULAR SEQUENCE DATA; PROTEIN CONFORMATION; RECEPTORS, ESTROGEN; SEQUENCE ALIGNMENT; SEQUENCE HOMOLOGY, AMINO ACID; TAMOXIFEN;

EID: 2642544810     PISSN: 00278424     EISSN: None     Source Type: Journal    
DOI: 10.1073/pnas.96.7.3999     Document Type: Article

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