Synthesis and structure-activity relationships of thieno[2,3-d]pyrimidine-2,4-dione derivatives as potent GnRH receptor antagonists

Bioorganic and Medicinal Chemistry Letters

Volumn 13, Issue 20, 2003, Pages 3617-3622

  Guo, Zhiqiang ^a   Chen, Yongsheng ^a   Wu, Dongpei ^a   Zhu, Yun Fei ^a   Struthers, R Scott ^a   Saunders, John ^a   Xie, Qiu ^a   Chen, Chen ^a  

^a NEUROCRINE BIOSCIENCES INC   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

GONADORELIN ANTAGONIST; GONADORELIN RECEPTOR; THIENO[2,3 D]PYRIMIDINE DERIVATIVE;

ARTICLE; BINDING AFFINITY; CELL STRAIN; DRUG BINDING; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; EMBRYO; HUMAN; HUMAN CELL; HYDROPHOBICITY; REPRODUCTION; STRUCTURE ACTIVITY RELATION;

EID: 0141851351     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(03)00746-7     Document Type: Article

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