SAR studies of novel 5-substituted 2-arylindoles as nonpeptidyl GnRH receptor antagonists

Bioorganic and Medicinal Chemistry Letters

Volumn 11, Issue 4, 2001, Pages 515-517

  Chu, Lin ^a   Lo, Jane Ling ^a   Yang, Yi Tien ^a   Cheng, Kang ^a   Smith, Roy G ^a   Fisher, Michael H ^a   Wyvratt, Matthew J ^a   Goulet, Mark T ^a  

^a MERCK RESEARCH LABORATORIES   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

GONADORELIN ANTAGONIST; GONADORELIN RECEPTOR;

ARTICLE; BINDING AFFINITY; DRUG POTENCY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; NONHUMAN; RAT; STRUCTURE ACTIVITY RELATION; STRUCTURE ANALYSIS;

ANIMALS; INDOLES; RATS; RECEPTORS, LHRH; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0035952296     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0960-894X(00)00708-3     Document Type: Article

References (6)