Indexed keywords
2 (3,5 DIMETHYLPHENYL)TRYPTAMINE DERIVATIVE;
3 (N BENZYL N METHYLAMINOMETHYL) 7 (2,6 DIFLUOROBENZYL) 4,7 DIHYDRO 2 (4 ISOBUTYRYLAMINOPHENYL) 4 OXOTHIENO[2,3 B]PYRIDINE 5 CARBOXYLIC ACID ISOPROPYL ESTER;
GONADORELIN ANTAGONIST;
GONADORELIN RECEPTOR;
NITROGEN;
TRYPTAMINE DERIVATIVE;
UNCLASSIFIED DRUG;
ARTICLE;
BINDING AFFINITY;
DRUG RECEPTOR BINDING;
DRUG STRUCTURE;
DRUG SYNTHESIS;
ISOMER;
NONHUMAN;
RAT;
ANIMALS;
BINDING SITES;
DRUG DESIGN;
FEMALE;
HORMONE ANTAGONISTS;
HUMANS;
INHIBITORY CONCENTRATION 50;
MOLECULAR STRUCTURE;
RATS;
RECEPTORS, LHRH;
TRYPTAMINES;
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-
1
-
-
0015218538
-
-
(1971)
Science
, vol.173
, pp. 1036
-
-
Schally, A.V.1
Arimura, A.2
Kastin, A.J.3
Matsuo, H.4
Baba, Y.5
Reddin, T.W.6
Nair, R.M.G.7
Debeljuk, L.8
White, W.F.9
-
4
-
-
85047684169
-
-
(2000)
Mol. Endocrinol.
, vol.14
, pp. 671
-
-
Cui, J.1
Smith, R.G.2
Mount, G.R.3
Lo, J.-L.4
Yu, J.5
Walsh, T.F.6
Singh, S.B.7
DeVita, R.J.8
Goulet, M.T.9
Schaeffer, J.M.10
Cheng, K.11
-
5
-
-
0029135443
-
-
(1995)
J. Biol. Chem.
, vol.270
, pp. 18853
-
-
Zhou, W.1
Rodic, V.2
Kitanovic, S.3
Flanagan, C.A.4
Chi, L.5
Weinstein, H.6
Maayani, S.7
Millar, R.P.8
Sealfon, S.C.9
-
8
-
-
0005357704
-
-
Filicori, M.; Flamigni, C., Ed.; Parthenon Publishing: Carnforth, UK
-
(1998)
Ovul. Induct. Update '98, Proc. World Conf., 2nd, Meeting Date 1997
, pp. 107-113
-
-
Behre, H.M.1
Nordhoff, V.2
Nieschlag, E.3
-
9
-
-
15444355594
-
-
(1998)
J. Med. Chem.
, vol.41
, pp. 4190
-
-
Cho, N.1
Harada, M.2
Imaeda, T.3
Imada, T.4
Matsumoto, H.5
Hayase, Y.6
Sasaki, S.7
Furuya, S.8
Suzuki, N.9
Okuobo, S.10
Ogi, K.11
Endo, S.12
Onda, H.13
Fujino, M.14
-
10
-
-
0033530102
-
-
(1999)
Bioorg. Med. Chem. Lett.
, vol.9
, pp. 2615
-
-
DeVita, R.J.1
Hollings, D.D.2
Goulet, M.T.3
Wyvratt, M.J.4
Fisher, M.H.5
Lo, J.-L.6
Yang, Y.T.7
Cheng, K.8
Smith, R.G.9
-
11
-
-
0033530138
-
-
(1999)
Bioorg. Med. Chem. Lett.
, vol.9
, pp. 2621
-
-
DeVita, R.J.1
Goulet, M.T.2
Wyvratt, M.J.3
Fisher, M.H.4
Lo, J.-L.5
Yang, Y.T.6
Cheng, K.7
Smith, R.G.8
-
12
-
-
0034611086
-
-
(2000)
Bioorg. Med. Chem. Lett.
, vol.10
, pp. 443
-
-
Walsh, T.F.1
Toupence, R.B.2
Young, J.R.3
Huang, S.X.4
Ujjainwalla, F.5
DeVita, R.J.6
Goulet, M.T.7
Wyvratt M.J., Jr.8
Fisher, M.H.9
Lo, J.-L.10
Ren, N.11
Yudkovitz, J.B.12
Yang, Y.T.13
Cheng, K.14
Smith, R.G.15
-
13
-
-
0034618152
-
-
(2000)
Bioorg. Med. Chem. Lett.
, vol.10
, pp. 1723
-
-
Young, J.R.1
Huang, S.X.2
Chen, I.3
Walsh, T.F.4
DeVita, R.J.5
Goulet, M.T.6
Wyvratt M.J., Jr.7
Fisher, M.H.8
Lo, J.9
Ren, N.10
Yudkovitz, J.B.11
Yang, Y.T.12
Cheng, K.13
Smith, R.G.14
-
14
-
-
0035866652
-
-
(2001)
J. Med. Chem.
, vol.44
, pp. 917
-
-
DeVita, R.J.1
Walsh, T.F.2
Young, J.R.3
Jiang, J.4
Ujjainwalla, F.5
Toupence, R.B.6
Parikh, M.7
Huang, S.X.8
Fair, J.A.9
Goulet, M.T.10
Wyvratt, M.J.11
Lo, J.-L.12
Ren, N.13
Yudkovitz, J.B.14
Yang, Y.T.15
Cheng, K.16
Cui, J.17
Mount, G.18
Rohrer, S.P.19
Schaeffer, J.M.20
Rhodes, L.21
Drisko, J.E.22
McGowan, E.23
MacIntyre, D.E.24
Vincent, S.25
Carlin, J.R.26
Cameron, J.27
Smith, R.G.28
more..
-
15
-
-
0035952261
-
-
(2001)
Bioorg. Med. Chem. Lett.
, vol.11
, pp. 509
-
-
Chu, L.1
Hutchins, J.E.2
Weber, A.E.3
Lo, J.-L.4
Yang, Y.T.5
Cheng, K.6
Smith, R.G.7
Fisher, M.H.8
Wyvratt, M.J.9
Goulet, M.T.10
-
16
-
-
0035952296
-
-
(2001)
Bioorg. Med. Chem. Lett.
, vol.11
, pp. 515
-
-
Chu, L.1
Lo, J.-L.2
Yang, Y.T.3
Cheng, K.4
Smith, R.G.5
Fisher, M.H.6
Wyvratt, M.J.7
Goulet, M.T.8
-
17
-
-
0005280155
-
-
note
-
-
-
-
18
-
-
0005279844
-
-
note
-
-
-
-
19
-
-
0005281092
-
-
note
-
-
-
-
20
-
-
0035938412
-
-
(2001)
Bioorg. Med. Chem. Lett.
, vol.11
, pp. 1077
-
-
Lin, P.1
Parikh, M.2
Lo, J.-L.3
Yang, Y.T.4
Cheng, K.5
Smith, R.G.6
Fisher, M.H.7
Wyvratt, M.J.8
Goulet, M.T.9
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