Testing the specificity of allosteric modulators of muscarinic receptors in phylogenetically closely related histamine H1-receptors

Naunyn-Schmiedeberg's Archives of Pharmacology

Volumn 361, Issue 2, 2000, Pages 107-112

  Franken, Christian ^b   Tränkle, Christian ^a   Mohr, Klaus ^a  

^a UNIVERSITY OF BONN   (Germany)

^b UNIVERSITY HOSPITAL ULM   (Germany)

Author keywords

Alcuronium; Allosteric modulation; Gallamine; Histamine H1 receptor; Mepyramine binding; Muscarinic acetylcholine M2 receptor; N methylscopolamine binding; W84

Indexed keywords

1,6 HEXAMETHYLENEBIS[DIMETHYL(3 PHTHALIMIDOPROPYL)AMMONIUM BROMIDE]; ALCURONIUM; GALLAMINE; HISTAMINE H1 RECEPTOR; MUSCARINIC M2 RECEPTOR;

ALLOSTERISM; ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; CONCENTRATION RESPONSE; DISSOCIATION CONSTANT; DRUG RECEPTOR BINDING; HEART; NONHUMAN; RECEPTOR SENSITIVITY; SWINE;

ALCURONIUM; ALLOSTERIC REGULATION; ANIMALS; BINDING SITES; GALLAMINE TRIETHIODIDE; GUINEA PIGS; N-METHYLSCOPOLAMINE; PHTHALIMIDES; PYRILAMINE; RECEPTORS, HISTAMINE H1; RECEPTORS, MUSCARINIC;

EID: 0043278941     PISSN: 00281298     EISSN: None     Source Type: Journal    
DOI: 10.1007/s002109900176     Document Type: Article

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