메뉴 건너뛰기




Volumn 72, Issue 22, 2003, Pages 2429-2449

5-HT2A and 5-HT2C receptors and their atypical regulation properties

Author keywords

5 HT2A 2C receptors; Agonists; Antagonists; Antidepressants; Antipsychotics; Regulation

Indexed keywords

2 CHLORO 11 (3 DIMETHYLAMINOPROPYLIDENE)MORPHANTHRIDINE; 2,3,3A,12B TETRAHYDRO 3 METHYL 1H DIBENZO[B,F]OXEPINO[10,11 C]PYRROLE; AMITRIPTYLINE; ANTIDEPRESSANT AGENT; CITALOPRAM; CLOMIPRAMINE; CLORGYLINE; CYPROHEPTADINE; DESIPRAMINE; DOSULEPIN; EPLIVANSERIN; FLUOXETINE; IMIPRAMINE; IPRINDOLE; KETANSERIN; MAPROTILINE; METERGOLINE; METHYSERGIDE; MONOAMINE OXIDASE INHIBITOR; NEUROLEPTIC AGENT; PARGYLINE; PAROXETINE; PHENELZINE; RITANSERIN; SEROTONIN 2 ANTAGONIST; SEROTONIN 2A AGONIST; SEROTONIN 2C AGONIST; SERTRALINE; TRANYLCYPROMINE; TRICYCLIC ANTIDEPRESSANT AGENT; UNINDEXED DRUG; ZIMELDINE; GUANINE NUCLEOTIDE BINDING PROTEIN; SEROTONIN 2A RECEPTOR; SEROTONIN 2C RECEPTOR; SEROTONIN AGONIST; SEROTONIN ANTAGONIST; SEROTONIN RECEPTOR;

EID: 0037453204     PISSN: 00243205     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0024-3205(03)00141-3     Document Type: Short Survey
Times cited : (187)

References (163)
  • 4
    • 0033837453 scopus 로고    scopus 로고
    • 2A receptor mRNA levels and binding sites in rat frontal cortex by the agonist DOI and the antagonist mianserin
    • 2A receptor mRNA levels and binding sites in rat frontal cortex by the agonist DOI and the antagonist mianserin. Neuropharmacology. 39(11):2000;1996-2005.
    • (2000) Neuropharmacology , vol.39 , Issue.11 , pp. 1996-2005
    • Anji, A.1    Kumari, M.2    Sullivan Hanley, N.R.3    Bryan, G.L.4    Hensler, J.G.5
  • 5
    • 0035051189 scopus 로고    scopus 로고
    • The role of protein kinase C in the regulation of serotonin-2A receptor expression
    • Anji A., Sullivan Hanley N.R., Kumari M., Hensler J.G. The role of protein kinase C in the regulation of serotonin-2A receptor expression. Journal of Neurochemistry. 77(2):2001;589-597.
    • (2001) Journal of Neurochemistry , vol.77 , Issue.2 , pp. 589-597
    • Anji, A.1    Sullivan Hanley, N.R.2    Kumari, M.3    Hensler, J.G.4
  • 6
    • 0034604706 scopus 로고    scopus 로고
    • 2C receptor PDZ recognition motif prevents receptor phosphorylation and delays resensitization of receptor responses
    • 2C receptor PDZ recognition motif prevents receptor phosphorylation and delays resensitization of receptor responses. Journal of Biological Chemistry. 275(31):2000;23620-23626.
    • (2000) Journal of Biological Chemistry , vol.275 , Issue.31 , pp. 23620-23626
    • Backstrom, J.R.1    Price, R.D.2    Reasoner, D.T.3    Sanders-Bush, E.4
  • 7
    • 0031040711 scopus 로고    scopus 로고
    • Effects of selective serotonin reuptake inhibitors on platelet serotonin parameters in major depressive disorder
    • Bakish D., Cavazzoni P., Chudzik J., Ravindran A., Hrdina P.D. Effects of selective serotonin reuptake inhibitors on platelet serotonin parameters in major depressive disorder. Biological Psychiatry. 41:1997;184-190.
    • (1997) Biological Psychiatry , vol.41 , pp. 184-190
    • Bakish, D.1    Cavazzoni, P.2    Chudzik, J.3    Ravindran, A.4    Hrdina, P.D.5
  • 8
    • 0017767136 scopus 로고
    • Development of beta-adrenergic receptor subsensitivity by antidepressants
    • Banerjee S.P., Kung L.S., Riggi S.J., Chanda S.K. Development of beta-adrenergic receptor subsensitivity by antidepressants. Nature. 268(5619):1977;455-456.
    • (1977) Nature , vol.268 , Issue.5619 , pp. 455-456
    • Banerjee, S.P.1    Kung, L.S.2    Riggi, S.J.3    Chanda, S.K.4
  • 9
    • 0028000662 scopus 로고
    • A highly conserved tyrosine residue in G protein-coupled receptors is required for agonist-mediated beta 2-adrenergic receptor sequestration
    • Barak L.S., Tiberi M., Freedman N.J., Kwatra M.M., Lefkowitz R.J., Caron M.G. A highly conserved tyrosine residue in G protein-coupled receptors is required for agonist-mediated beta 2-adrenergic receptor sequestration. Journal of Biological Chemistry. 269:1994;2790-2795.
    • (1994) Journal of Biological Chemistry , vol.269 , pp. 2790-2795
    • Barak, L.S.1    Tiberi, M.2    Freedman, N.J.3    Kwatra, M.M.4    Lefkowitz, R.J.5    Caron, M.G.6
  • 10
    • 0020677878 scopus 로고
    • On the mode of action of imipramine: Relationship between serotonergic axon terminal function and down-regulation of beta-adrenergic receptors
    • Barbaccia M.L., Brunello N., Chuang D.M., Costa E. On the mode of action of imipramine: relationship between serotonergic axon terminal function and down-regulation of beta-adrenergic receptors. Neuropharmacology. 22:1983;373-383.
    • (1983) Neuropharmacology , vol.22 , pp. 373-383
    • Barbaccia, M.L.1    Brunello, N.2    Chuang, D.M.3    Costa, E.4
  • 11
    • 0027332129 scopus 로고
    • 1C receptor density and mRNA levels in choroid plexus epithelial cells after treatment with mianserin and (-)-1-(4-Bromo-2,5-dimethoxyphenyl)-2-aminopropane
    • 1C receptor density and mRNA levels in choroid plexus epithelial cells after treatment with mianserin and (-)-1-(4-Bromo-2,5-dimethoxyphenyl)-2-aminopropane. Molecular Pharmacology. 44:1993;725-730.
    • (1993) Molecular Pharmacology , vol.44 , pp. 725-730
    • Barker, E.L.1    Sanders-Bush, E.2
  • 13
    • 0027421854 scopus 로고
    • Chronic treatment with fluvoxamine increases extracellular serotonin in frontal cortex but not in raphe nuclei
    • Bel N., Artigas F. Chronic treatment with fluvoxamine increases extracellular serotonin in frontal cortex but not in raphe nuclei. Synapse. 15(3):1993;243-245.
    • (1993) Synapse , vol.15 , Issue.3 , pp. 243-245
    • Bel, N.1    Artigas, F.2
  • 16
    • 0018361822 scopus 로고
    • Adrenergic and serotonergic receptor binding in rat brain after chronic desmethylimipramine treatment
    • Bergstrom D.A., Kellar K.J. Adrenergic and serotonergic receptor binding in rat brain after chronic desmethylimipramine treatment. Journal of Pharmacology and Experimental Therapeutics. 209(2):1979;256-261.
    • (1979) Journal of Pharmacology and Experimental Therapeutics , vol.209 , Issue.2 , pp. 256-261
    • Bergstrom, D.A.1    Kellar, K.J.2
  • 27
    • 0028081958 scopus 로고
    • 2 receptors and the abundances of 5-HT receptor and transporter mRNA in the cortex, hippocampus and dorsal raphe of three strains of rat
    • 2 receptors and the abundances of 5-HT receptor and transporter mRNA in the cortex, hippocampus and dorsal raphe of three strains of rat. Brain Research. 638:1994;311-324.
    • (1994) Brain Research , vol.638 , pp. 311-324
    • Burnet, P.W.1    Michelson, D.2    Smith, M.A.3    Gold, P.W.4    Sternberg, E.M.5
  • 28
    • 0024540787 scopus 로고
    • Imipramine and tetrabenazine: Effects on monoamine receptor binding sites and phosphoinositide hydrolysis
    • Butler P.D., Edwards E., Barkai A.I. Imipramine and tetrabenazine: Effects on monoamine receptor binding sites and phosphoinositide hydrolysis. European Journal of Pharmacology. 160:1989;93-100.
    • (1989) European Journal of Pharmacology , vol.160 , pp. 93-100
    • Butler, P.D.1    Edwards, E.2    Barkai, A.I.3
  • 31
    • 0030943091 scopus 로고    scopus 로고
    • Neurotransmitter aberrations in schizophrenia: New perspectives and therapeutic implications
    • Carlsson A., Hansson L.O., Waters N., Carlsson M.L. Neurotransmitter aberrations in schizophrenia: new perspectives and therapeutic implications. Life Sciences. 61:1997;75-94.
    • (1997) Life Sciences , vol.61 , pp. 75-94
    • Carlsson, A.1    Hansson, L.O.2    Waters, N.3    Carlsson, M.L.4
  • 32
    • 0027431521 scopus 로고
    • Behavioural and biochemical evidence that glucocorticoids are not involved in DOI-elicited 5-HT2 receptor down-regulation
    • Chaouloff F., Baudrie V., Coupry I. Behavioural and biochemical evidence that glucocorticoids are not involved in DOI-elicited 5-HT2 receptor down-regulation. European Journal of Pharmacology. 249(1):1993;117-120.
    • (1993) European Journal of Pharmacology , vol.249 , Issue.1 , pp. 117-120
    • Chaouloff, F.1    Baudrie, V.2    Coupry, I.3
  • 34
    • 0029619094 scopus 로고
    • 2) receptor binding sites in cerebellar granule neurons: Involvement of calcium influx and a calmodulin-dependent pathway
    • 2) receptor binding sites in cerebellar granule neurons: involvement of calcium influx and a calmodulin-dependent pathway. Journal of Pharmacology and Experimental Therapeutics. 275:1995;674-680.
    • (1995) Journal of Pharmacology and Experimental Therapeutics , vol.275 , pp. 674-680
    • Chen, H.1    Li, H.2    Chuang, D.3
  • 37
    • 0021024834 scopus 로고
    • 2 receptor binding during combined administration of tricyclic antidepressant drugs and alpha 2 antagonists
    • 2 receptor binding during combined administration of tricyclic antidepressant drugs and alpha 2 antagonists. Neuropharmacology. 22:1983;1203-1209.
    • (1983) Neuropharmacology , vol.22 , pp. 1203-1209
    • Crews, F.T.1    Scott, J.A.2    Shorstein, N.H.3
  • 38
    • 0018146337 scopus 로고
    • Presynaptic alpha-receptor subsensitivity after long-term antidepressant treatment
    • Crews F.T., Smith C.B. Presynaptic alpha-receptor subsensitivity after long-term antidepressant treatment. Science. 202(4365):1978;322-324.
    • (1978) Science , vol.202 , Issue.4365 , pp. 322-324
    • Crews, F.T.1    Smith, C.B.2
  • 39
    • 0021894160 scopus 로고
    • 1 receptor binding in cortex of rat after chronic administration of dothiepin. Application of the Woolf plot to analysis of binding parameters
    • 1 receptor binding in cortex of rat after chronic administration of dothiepin. Application of the Woolf plot to analysis of binding parameters. Neuropharmacology. 24:1985;275-278.
    • (1985) Neuropharmacology , vol.24 , pp. 275-278
    • Diggory, G.L.1    Buckett, W.R.2
  • 40
    • 0024380377 scopus 로고
    • Effects of imipramine and serotonin-2 agonists and antagonists on serotonin-2 and beta-adrenergic receptors following noradrenergic or serotonergic denervation
    • Eison A.S., Eison M.S., Yocca F.D., Gianutsos G. Effects of imipramine and serotonin-2 agonists and antagonists on serotonin-2 and beta-adrenergic receptors following noradrenergic or serotonergic denervation. Life Sciences. 44(19):1989;1419-1427.
    • (1989) Life Sciences , vol.44 , Issue.19 , pp. 1419-1427
    • Eison, A.S.1    Eison, M.S.2    Yocca, F.D.3    Gianutsos, G.4
  • 43
    • 0030593035 scopus 로고    scopus 로고
    • Role of beta-arrestin in mediating agonist-promoted G protein-coupled receptor internalization
    • Ferguson S.S., Downey W.E. III, Colapietro A.M., Barak L.S., Menard L., Caron M.G. Role of beta-arrestin in mediating agonist-promoted G protein-coupled receptor internalization. Science. 271:1996;363-366.
    • (1996) Science , vol.271 , pp. 363-366
    • Ferguson, S.S.1    Downey W.E. III2    Colapietro, A.M.3    Barak, L.S.4    Menard, L.5    Caron, M.G.6
  • 44
    • 0021074927 scopus 로고
    • 2), alpha 2-adrenergic. imipramine and dopaminergic receptors in brain
    • 2), alpha 2-adrenergic. imipramine and dopaminergic receptors in brain. Neuropharmacology. 22:1983;1257-1267.
    • (1983) Neuropharmacology , vol.22 , pp. 1257-1267
    • Ferris, R.M.1    Beaman, O.J.2
  • 47
    • 0028283115 scopus 로고
    • Uptake inhibitors increase extracellular serotonin concentration measured by brain microdialysis
    • Fuller R.W. Uptake inhibitors increase extracellular serotonin concentration measured by brain microdialysis. Life Sciences. 55:1994;163-167.
    • (1994) Life Sciences , vol.55 , pp. 163-167
    • Fuller, R.W.1
  • 49
    • 0027989702 scopus 로고
    • Agonist-induced internalization of the substance P (NK1) receptor expressed in epithelial cells
    • Garland A.M., Grady E.F., Payan D.G., Vigna S.R., Bunnett N.W. Agonist-induced internalization of the substance P (NK1) receptor expressed in epithelial cells. Biochemical Journal. 303(Pt 1):1994;177-186.
    • (1994) Biochemical Journal , vol.303 , pp. 177-186
    • Garland, A.M.1    Grady, E.F.2    Payan, D.G.3    Vigna, S.R.4    Bunnett, N.W.5
  • 50
    • 0021241901 scopus 로고
    • Comparison of iprindole.imipramine and mianserin action on brain serotonergic and beta adrenergic receptors
    • Gandolfi O., Barbaccia M.L., Costa E. Comparison of iprindole.imipramine and mianserin action on brain serotonergic and beta adrenergic receptors. Journal of Pharmacology and Experimental Therapeutics. 229:1984;782-786.
    • (1984) Journal of Pharmacology and Experimental Therapeutics , vol.229 , pp. 782-786
    • Gandolfi, O.1    Barbaccia, M.L.2    Costa, E.3
  • 52
    • 0028176097 scopus 로고
    • 2 and beta-adrenergic receptor regulation in rat brain following chronic treatment with desipramine and fluoxetine alone and in combination
    • 2 and beta-adrenergic receptor regulation in rat brain following chronic treatment with desipramine and fluoxetine alone and in combination. Journal of Neurochemistry. 62:1994;2262-2268.
    • (1994) Journal of Neurochemistry , vol.62 , pp. 2262-2268
    • Goodnough, D.B.1    Baker, G.B.2
  • 54
    • 0021285237 scopus 로고
    • 2 receptor-mediated head-twitch behaviour following antidepressant treatment to mice
    • 2 receptor-mediated head-twitch behaviour following antidepressant treatment to mice. Britisch Journal of Pharmacology. 83(1):1984;235-242.
    • (1984) Britisch Journal of Pharmacology , vol.83 , Issue.1 , pp. 235-242
    • Goodwin, G.M.1    Green, A.R.2    Johnson, P.3
  • 55
    • 0028290841 scopus 로고
    • Differential effects of N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ) on various 5-HT receptor binding sites in the rat brain
    • Gozlan H., Laporte A.M., Thibault S., Schechter L.E., Bolanos F., Hamon M. Differential effects of N-ethoxycarbonyl-2-ethoxy-1,2-dihydroquinoline (EEDQ) on various 5-HT receptor binding sites in the rat brain. Neuropharmacology. 33(3-4):1994;423-431.
    • (1994) Neuropharmacology , vol.33 , Issue.3-4 , pp. 423-431
    • Gozlan, H.1    Laporte, A.M.2    Thibault, S.3    Schechter, L.E.4    Bolanos, F.5    Hamon, M.6
  • 56
    • 0035891883 scopus 로고    scopus 로고
    • 2A receptors by agonists and antagonists
    • 2A receptors by agonists and antagonists. Brain Research Bulletins. 56(5):2001;441-451.
    • (2001) Brain Research Bulletins , vol.56 , Issue.5 , pp. 441-451
    • Gray, J.A.1    Roth, B.L.2
  • 61
    • 0021025617 scopus 로고
    • Unusual acute effects of antidepressants and neuroleptics on S2-serotonergic receptors
    • Helmeste D.M., Tang S.W. Unusual acute effects of antidepressants and neuroleptics on S2-serotonergic receptors. Life Sciences. 33:1983;2527-2533.
    • (1983) Life Sciences , vol.33 , pp. 2527-2533
    • Helmeste, D.M.1    Tang, S.W.2
  • 63
    • 0028183684 scopus 로고
    • Lack of 5-HT1A autoreceptor desensitisation following chronic citalopram treatment, as determined by in vivo microdialysis
    • Hjorth S., Auerbach S.B. Lack of 5-HT1A autoreceptor desensitisation following chronic citalopram treatment, as determined by in vivo microdialysis. Neuropharmacology. 33(3-4):1994;331-334.
    • (1994) Neuropharmacology , vol.33 , Issue.3-4 , pp. 331-334
    • Hjorth, S.1    Auerbach, S.B.2
  • 64
    • 0027290988 scopus 로고
    • 2 receptors in rat brain: An autoradiographic study
    • 2 receptors in rat brain: an autoradiographic study. Synapse. 14:1993;324-331.
    • (1993) Synapse , vol.14 , pp. 324-331
    • Hrdina, P.D.1    Vu, T.B.2
  • 65
    • 0027984917 scopus 로고
    • Differential effects of chronic antidepressant treatment on 5-HT1C receptor binding sites in Wistar rat brain
    • Hulihan-Giblin B.A., Park Y.D., Aulakh C.S. Differential effects of chronic antidepressant treatment on 5-HT1C receptor binding sites in Wistar rat brain. European Journal of Pharmacology. 263(1-2):1994;213-216.
    • (1994) European Journal of Pharmacology , vol.263 , Issue.1-2 , pp. 213-216
    • Hulihan-Giblin, B.A.1    Park, Y.D.2    Aulakh, C.S.3
  • 66
    • 0021368802 scopus 로고
    • Biochemical effects and drug levels in rats after long-term treatment with the specific 5-HT-uptake inhibitor, citalopram
    • Hyttel J., Overo K.F., Arnt J. Biochemical effects and drug levels in rats after long-term treatment with the specific 5-HT-uptake inhibitor, citalopram. Psychopharmacology (Berl). 83(1):1984;20-27.
    • (1984) Psychopharmacology (Berl) , vol.83 , Issue.1 , pp. 20-27
    • Hyttel, J.1    Overo, K.F.2    Arnt, J.3
  • 67
    • 0028018469 scopus 로고
    • Chronic treatment with citalopram facilitates the effect of a challenge dose on cortical serotonin output: Role of presynaptic 5-HT1A receptors
    • Invernizzi R., Bramante M., Samanin R. Chronic treatment with citalopram facilitates the effect of a challenge dose on cortical serotonin output: role of presynaptic 5-HT1A receptors. European Journal of Pharmacology. 260(2-3):1994;243-246.
    • (1994) European Journal of Pharmacology , vol.260 , Issue.2-3 , pp. 243-246
    • Invernizzi, R.1    Bramante, M.2    Samanin, R.3
  • 69
    • 0031594813 scopus 로고    scopus 로고
    • 5-Hydroxytryptamine2A serotonin receptors in the primate cerebral cortex: Possible site of action of hallucinogenic and antipsychotic drugs in pyramidal cell apical dendrites
    • Jakab R., Goldman-Rakic P. 5-Hydroxytryptamine2A serotonin receptors in the primate cerebral cortex: possible site of action of hallucinogenic and antipsychotic drugs in pyramidal cell apical dendrites. Proceedings of the National Acadamie of Sciences U S A. 95:1998;735-740.
    • (1998) Proceedings of the National Acadamie of Sciences U S A , vol.95 , pp. 735-740
    • Jakab, R.1    Goldman-Rakic, P.2
  • 73
    • 0021963089 scopus 로고
    • 5-Hydroxytryptamine-stimulated inositol phospholipid hydrolysis in rat cerebral cortex slices: Pharmacological characterization and effects of antidepressants
    • Kendall D.A., Nahorski S.R. 5-Hydroxytryptamine-stimulated inositol phospholipid hydrolysis in rat cerebral cortex slices: pharmacological characterization and effects of antidepressants. Journal of Pharmacology and Experimental Therapeutics. 233(2):1985;473-479.
    • (1985) Journal of Pharmacology and Experimental Therapeutics , vol.233 , Issue.2 , pp. 473-479
    • Kendall, D.A.1    Nahorski, S.R.2
  • 74
    • 0020471321 scopus 로고
    • The inf1uence of sex hormones on antidepressant-induced alterations in neurotransmitter receptor binding
    • Kendall D.A., Stancel G.M., Enna S.J. The inf1uence of sex hormones on antidepressant-induced alterations in neurotransmitter receptor binding. Journal of Neurosciences. 2:1982;354-360.
    • (1982) Journal of Neurosciences , vol.2 , pp. 354-360
    • Kendall, D.A.1    Stancel, G.M.2    Enna, S.J.3
  • 78
    • 0024723668 scopus 로고
    • 2 receptor density induced by repeated treatment with 5-HT uptake inhibitor or 5-HT agonist]
    • 2 receptor density induced by repeated treatment with 5-HT uptake inhibitor or 5-HT agonist]. Yakubutsu Seishin Kodo. 9:1989;289-292.
    • (1989) Yakubutsu Seishin Kodo , vol.9 , pp. 289-292
    • Kubota, M.1    Ueno, K.2    Yamano, M.3    Kitagawa, H.4
  • 79
    • 0028783676 scopus 로고
    • 2C receptors after chronic treatment with clozapine, chlorpromazine and three putative atypical antipsychotic drugs
    • 2C receptors after chronic treatment with clozapine, chlorpromazine and three putative atypical antipsychotic drugs. Neuropsychopharmacology. 13:1995;139-150.
    • (1995) Neuropsychopharmacology , vol.13 , pp. 139-150
    • Kuoppamaki, M.1    Palvimaki, E.P.2    Hietala, J.3    Syvalahti, E.4
  • 80
    • 0027371938 scopus 로고
    • Chronic clozapine treatment decreases 5-hydroxytryptamine1C receptor density in the rat choroid plexus: Comparison with haloperidol
    • Kuoppamaki M., Seppala T., Syvalahti E., Hietala J. Chronic clozapine treatment decreases 5-hydroxytryptamine1C receptor density in the rat choroid plexus: comparison with haloperidol. Journal of Pharmacology and Experimental Therapeutics. 264(3):1993;1262-1267.
    • (1993) Journal of Pharmacology and Experimental Therapeutics , vol.264 , Issue.3 , pp. 1262-1267
    • Kuoppamaki, M.1    Seppala, T.2    Syvalahti, E.3    Hietala, J.4
  • 82
    • 0030967614 scopus 로고    scopus 로고
    • Arrestin/clathrin interaction: Localization of the clathrin binding domain of nonvisual arrestins to the carboxy terminus
    • Krupnick J.G., Goodman O.B., Keen J.H., Benovic J.L. Arrestin/clathrin interaction: localization of the clathrin binding domain of nonvisual arrestins to the carboxy terminus. Journal of Biological and Chemistry. 274:1997;15011-15016.
    • (1997) Journal of Biological and Chemistry , vol.274 , pp. 15011-15016
    • Krupnick, J.G.1    Goodman, O.B.2    Keen, J.H.3    Benovic, J.L.4
  • 84
    • 0029045445 scopus 로고
    • Serotonergic antagonists differentially inhibit spontaneous activity and decrease ligand binding capacity of the rat 5-hydroxytryptamine type 2C receptor in Sf9 cells
    • Labrecque J., Fargin A., Bouvier M., Chidiac P., Dennis M. Serotonergic antagonists differentially inhibit spontaneous activity and decrease ligand binding capacity of the rat 5-hydroxytryptamine type 2C receptor in Sf9 cells. Molecular Pharmacology. 48:1995;150-159.
    • (1995) Molecular Pharmacology , vol.48 , pp. 150-159
    • Labrecque, J.1    Fargin, A.2    Bouvier, M.3    Chidiac, P.4    Dennis, M.5
  • 86
    • 0021218659 scopus 로고
    • Loxapine and clozapine decrease serotonin (S2) but do not elevate dopamine (D2) receptor numbers in the rat brain
    • Lee T., Tang S.W. Loxapine and clozapine decrease serotonin (S2) but do not elevate dopamine (D2) receptor numbers in the rat brain. Psychiatry Research. 12(4):1984;277-285.
    • (1984) Psychiatry Research , vol.12 , Issue.4 , pp. 277-285
    • Lee, T.1    Tang, S.W.2
  • 87
    • 0025350916 scopus 로고
    • Role of phosphorylation in desensitisation of the β-adrenoreceptor
    • Lefkowitz R.J., Hausdorff W.P., Caron M.G. Role of phosphorylation in desensitisation of the β-adrenoreceptor. TIPS. 11:1990;190-194.
    • (1990) TIPS , vol.11 , pp. 190-194
    • Lefkowitz, R.J.1    Hausdorff, W.P.2    Caron, M.G.3
  • 91
    • 0023255094 scopus 로고
    • Differential regulation of dopamine-D2 and serotonin-S2 receptors by chronic treatment with the serotonin-S2 antagonists, ritanserin, and setoperone
    • S.G. et al. Dahl. Berlin, Heidelberg: Springer Verlag
    • Leysen J.E., Van Gompel P., Gommeren W., Laduron P.M. Differential regulation of dopamine-D2 and serotonin-S2 receptors by chronic treatment with the serotonin-S2 antagonists, ritanserin, and setoperone. Dahl S.G.et al. Clinical pharmacology in Psychiatry. 1987;214-224 Springer Verlag, Berlin, Heidelberg.
    • (1987) Clinical pharmacology in Psychiatry , pp. 214-224
    • Leysen, J.E.1    Van Gompel, P.2    Gommeren, W.3    Laduron, P.M.4
  • 92
    • 0022595471 scopus 로고
    • Down-regulation of serotonin-S2 receptor sites in rat brain by chronic treatment with the serotonin-S2 antagonists ritanserin and setoperone
    • Leysen J.E., Van Gompel P., Gommeren W., Woestenborghs R., Janssen P. Down-regulation of serotonin-S2 receptor sites in rat brain by chronic treatment with the serotonin-S2 antagonists ritanserin and setoperone. Psychopharmacology. 88:1986;434-444.
    • (1986) Psychopharmacology , vol.88 , pp. 434-444
    • Leysen, J.E.1    Van Gompel, P.2    Gommeren, W.3    Woestenborghs, R.4    Janssen, P.5
  • 96
    • 0029089951 scopus 로고
    • 2A receptor-mediated excitatory effects of serotonin on interneurons in rat piriform cortex
    • 2A receptor-mediated excitatory effects of serotonin on interneurons in rat piriform cortex. Synapse. 21(2):1995;123-130.
    • (1995) Synapse , vol.21 , Issue.2 , pp. 123-130
    • Marek, G.J.1    Aghajanian, G.K.2
  • 97
    • 0024429166 scopus 로고
    • 2 receptor density in rat cerebral cortex
    • 2 receptor density in rat cerebral cortex. Life Sciences. 45:1989;1397-1406.
    • (1989) Life Sciences , vol.45 , pp. 1397-1406
    • Matsubara, S.1    Meltzer, H.Y.2
  • 100
    • 0030609874 scopus 로고    scopus 로고
    • Synergistic regulation of beta2-adrenergic receptor sequestration: Intracellular complement of beta-adrenergic receptor kinase and beta-arrestin determine kinetics of internalization
    • Menard L., Ferguson S.S., Zhang J., Lin F.T., Lefkowitz R.J., Caron M.G., Barak L.S. Synergistic regulation of beta2-adrenergic receptor sequestration: Intracellular complement of beta-adrenergic receptor kinase and beta-arrestin determine kinetics of internalization. Molecular Pharmacology. 51:1997;800-808.
    • (1997) Molecular Pharmacology , vol.51 , pp. 800-808
    • Menard, L.1    Ferguson, S.S.2    Zhang, J.3    Lin, F.T.4    Lefkowitz, R.J.5    Caron, M.G.6    Barak, L.S.7
  • 102
    • 0021352730 scopus 로고
    • Reduction of serotonin-2 y receptors in rat cerebral cortex after subchronic administration of imipramine, chlorpromazine, and the combination thereof
    • Mikuni M., Meltzer H.Y. Reduction of serotonin-2 y receptors in rat cerebral cortex after subchronic administration of imipramine, chlorpromazine, and the combination thereof. Life Sciences. 34:1984;87-92.
    • (1984) Life Sciences , vol.34 , pp. 87-92
    • Mikuni, M.1    Meltzer, H.Y.2
  • 103
    • 0027329899 scopus 로고
    • 2 receptor immunoreactivity on cholinergic neurons of the pontomesencephalic tegmentum shown by double immunofluorescence
    • 2 receptor immunoreactivity on cholinergic neurons of the pontomesencephalic tegmentum shown by double immunofluorescence. Brain Research. 627(1):1993;49-54.
    • (1993) Brain Research , vol.627 , Issue.1 , pp. 49-54
    • Morilak, D.A.1    Ciaranello, R.D.2
  • 105
    • 0033573730 scopus 로고    scopus 로고
    • Epidermal growth factor (EGF)-induced up-regulation and agonist- and antagonist-induced desensitisation and internalization of A1 adenosine receptors in a pituitary-derived cel1 line
    • Navarro A., Zapata R., Canela E.I., Mallol J., Luis C., Franco R. Epidermal growth factor (EGF)-induced up-regulation and agonist- and antagonist-induced desensitisation and internalization of A1 adenosine receptors in a pituitary-derived cel1 line. Brain Research. 816:1999;47-57.
    • (1999) Brain Research , vol.816 , pp. 47-57
    • Navarro, A.1    Zapata, R.2    Canela, E.I.3    Mallol, J.4    Luis, C.5    Franco, R.6
  • 106
    • 0030855796 scopus 로고    scopus 로고
    • 2C receptors stably expressed in the human neuroblastoma cell line SH-SY5Y
    • 2C receptors stably expressed in the human neuroblastoma cell line SH-SY5Y. Journal of Neurochemistry. 69:1997;1031-1038.
    • (1997) Journal of Neurochemistry , vol.69 , pp. 1031-1038
    • Newton, R.A.1    Elliot, J.M.2
  • 108
    • 0031933295 scopus 로고    scopus 로고
    • Differential localisation of the metabotropic glutamate receptor mGluR1a and the ionotropic glutamate receptor GluR2/3 in neurons of the human cerebral cortex
    • Ong W.Y., Tan K.K., Garey L.J. Differential localisation of the metabotropic glutamate receptor mGluR1a and the ionotropic glutamate receptor GluR2/3 in neurons of the human cerebral cortex. Exp. Brain Res. 119:1998;367-374.
    • (1998) Exp. Brain Res. , vol.119 , pp. 367-374
    • Ong, W.Y.1    Tan, K.K.2    Garey, L.J.3
  • 109
    • 0032545503 scopus 로고    scopus 로고
    • Characterization of dominant negative arrestins that inhibit beta2-adrenergic receptor internalization by distinct mechanisms
    • Orsini M.J., Benovic J.L. Characterization of dominant negative arrestins that inhibit beta2-adrenergic receptor internalization by distinct mechanisms. Journal of Biological Chemistry. 273:1998;34616-34622.
    • (1998) Journal of Biological Chemistry , vol.273 , pp. 34616-34622
    • Orsini, M.J.1    Benovic, J.L.2
  • 110
    • 0025667832 scopus 로고
    • 2 receptor mediated phosphatidyl inositol hydrolysis by serotonin agonists in quiescent calf aortic smooth muscle cells
    • 2 receptor mediated phosphatidyl inositol hydrolysis by serotonin agonists in quiescent calf aortic smooth muscle cells. Life Sciences. 47:1990;2009-2019.
    • (1990) Life Sciences , vol.47 , pp. 2009-2019
    • Pauwels, P.J.1    Van Gompel, P.2    Leysen, J.E.3
  • 112
    • 0021686458 scopus 로고
    • The binding of serotonergic ligands to the porcine choroid plexus: Characterisation of a new type of serotonin recognition site
    • Pazos A., Hoyer D., Palacios J.M. The binding of serotonergic ligands to the porcine choroid plexus: characterisation of a new type of serotonin recognition site. European Journal of Pharmacology. 106:1984;539-546.
    • (1984) European Journal of Pharmacology , vol.106 , pp. 539-546
    • Pazos, A.1    Hoyer, D.2    Palacios, J.M.3
  • 113
    • 0029809349 scopus 로고    scopus 로고
    • Local infusion of the seotonin antagonist ritanserin or ICS205930 increases in vivo dopamine release in the rat medial frontal cortex
    • Pehek E.A. Local infusion of the seotonin antagonist ritanserin or ICS205930 increases in vivo dopamine release in the rat medial frontal cortex. Synapse. 24:1996;12-19.
    • (1996) Synapse , vol.24 , pp. 12-19
    • Pehek, E.A.1
  • 114
    • 0019793815 scopus 로고
    • Two distinct central serotonin receptors with different physiological functions
    • Peroutka S.J., Lebovitz R.M., Snyder S.H. Two distinct central serotonin receptors with different physiological functions. Science. 212:1981;827-829.
    • (1981) Science , vol.212 , pp. 827-829
    • Peroutka, S.J.1    Lebovitz, R.M.2    Snyder, S.H.3
  • 115
    • 0019122846 scopus 로고
    • Long-term antidepressant treatment decreases spiroperidol-labeled serotonin receptor binding
    • Peroutka S.J., Snyder S.H. Long-term antidepressant treatment decreases spiroperidol-labeled serotonin receptor binding. Science. 210:1980;88-90.
    • (1980) Science , vol.210 , pp. 88-90
    • Peroutka, S.J.1    Snyder, S.H.2
  • 116
    • 0019225887 scopus 로고
    • 2) receptors labeled with [3H]spiroperidol by chronic treatment with the antidepressant amitriptyline
    • 2) receptors labeled with [3H]spiroperidol by chronic treatment with the antidepressant amitriptyline. Journal of Pharmacology and Experimental Therapeutics. 215:1980;582-587.
    • (1980) Journal of Pharmacology and Experimental Therapeutics , vol.215 , pp. 582-587
    • Peroutka, S.J.1    Snyder, S.H.2
  • 117
    • 0032505683 scopus 로고    scopus 로고
    • Agonist and antagonist-dependent interna1ization of the human vasopressin V2 receptor
    • Pfeiffer R., Kirsch J., Fahrenholz F. Agonist and antagonist-dependent interna1ization of the human vasopressin V2 receptor. Experimental Cell Research. 244:1998;327-339.
    • (1998) Experimental Cell Research , vol.244 , pp. 327-339
    • Pfeiffer, R.1    Kirsch, J.2    Fahrenholz, F.3
  • 118
    • 0028986859 scopus 로고
    • Sequestration and recycling of beta 2-adrenergic receptors permit receptor resensitization
    • Pippig S., Andexinger S., Lohse M.J. Sequestration and recycling of beta 2-adrenergic receptors permit receptor resensitization. Molecular Pharmacology. 47(4):1995;666-676.
    • (1995) Molecular Pharmacology , vol.47 , Issue.4 , pp. 666-676
    • Pippig, S.1    Andexinger, S.2    Lohse, M.J.3
  • 119
    • 0025923909 scopus 로고
    • 2 receptors in rat cortex. Studies with a putative selective agonist and an antagonist
    • 2 receptors in rat cortex. Studies with a putative selective agonist and an antagonist. Biochemical Pharmacology. 42:1991;1099-1105.
    • (1991) Biochemical Pharmacology , vol.42 , pp. 1099-1105
    • Pranzatelli, M.R.1
  • 122
    • 0028920668 scopus 로고
    • Protein kinases that phosphorylate activated G protein-coupled receptors
    • Premont R.T., Inglese J., Lefkowitz R.J. Protein kinases that phosphorylate activated G protein-coupled receptors. FASEB J. 9:1995;175-182.
    • (1995) FASEB J. , vol.9 , pp. 175-182
    • Premont, R.T.1    Inglese, J.2    Lefkowitz, R.J.3
  • 125
    • 0027254653 scopus 로고
    • Multiple mechanisms of serotonin 5-HT2 receptor desensitisation
    • Rahman S., Neuman R.S. Multiple mechanisms of serotonin 5-HT2 receptor desensitisation. European Journal of Pharmacology. 238(2-3):1993;173-180.
    • (1993) European Journal of Pharmacology , vol.238 , Issue.2-3 , pp. 173-180
    • Rahman, S.1    Neuman, R.S.2
  • 134
    • 0028214689 scopus 로고
    • Increase in extracellular serotonin produced by uptake inhibitors is enhanced after chronic treatment with fluoxetine
    • Rutter J.J., Gundlah C., Auerbach S.B. Increase in extracellular serotonin produced by uptake inhibitors is enhanced after chronic treatment with fluoxetine. Neuroscience Letters. 171(1-2):1994;183-186.
    • (1994) Neuroscience Letters , vol.171 , Issue.1-2 , pp. 183-186
    • Rutter, J.J.1    Gundlah, C.2    Auerbach, S.B.3
  • 135
    • 0024372505 scopus 로고
    • Sertraline-induced desensitisation of the serotonin 5HT-2 receptor transmembrane signalling system
    • Sanders-Bush E., Breeding M., Knoth K., Tsutsumi M. Sertraline-induced desensitisation of the serotonin 5HT-2 receptor transmembrane signalling system. Psychopharmacology. 99:1989;64-69.
    • (1989) Psychopharmacology , vol.99 , pp. 64-69
    • Sanders-Bush, E.1    Breeding, M.2    Knoth, K.3    Tsutsumi, M.4
  • 136
    • 0023163413 scopus 로고
    • 5HT2 binding sites after mianserin: Comparison of loss of sites and brain levels of drug
    • Sanders-Bush E., Breeding M., Roznoski M. 5HT2 binding sites after mianserin: comparison of loss of sites and brain levels of drug. European Journal of Pharmacology. 133(2):1987;199-204.
    • (1987) European Journal of Pharmacology , vol.133 , Issue.2 , pp. 199-204
    • Sanders-Bush, E.1    Breeding, M.2    Roznoski, M.3
  • 137
    • 0031770955 scopus 로고    scopus 로고
    • Endogenous serotonin-2A and-3C receptors in balb/c-3T3 cells revealed in serotonin-free medium
    • Saucier C., Morris S.J., Albert P.R. Endogenous serotonin-2A and-3C receptors in balb/c-3T3 cells revealed in serotonin-free medium. Biochemical Pharmacology. 56:1998;1347-1357.
    • (1998) Biochemical Pharmacology , vol.56 , pp. 1347-1357
    • Saucier, C.1    Morris, S.J.2    Albert, P.R.3
  • 138
    • 0030910406 scopus 로고    scopus 로고
    • Identification of an endogenous 5-hydroxytryptamine2A receptor in NIH-3T3 cells: Agonist-induced downregulation involves decreases in receptor RNA and number
    • Saucier C., AIbert P.R. Identification of an endogenous 5-hydroxytryptamine2A receptor in NIH-3T3 cells: agonist-induced downregulation involves decreases in receptor RNA and number. Journal of Neurochemistry. 68(5):1997;1998-2011.
    • (1997) Journal of Neurochemistry , vol.68 , Issue.5 , pp. 1998-2011
    • Saucier, C.1    Aibert, P.R.2
  • 139
    • 0024213895 scopus 로고
    • Species dependence of adaptations at the pre- and postsynaptic serotonergic receptors following longterm antidepressant drug treatment
    • Schoups A.A., De Potter W.P. Species dependence of adaptations at the pre- and postsynaptic serotonergic receptors following longterm antidepressant drug treatment. Biochemical Pharmacology. 37:1988;4451-4460.
    • (1988) Biochemical Pharmacology , vol.37 , pp. 4451-4460
    • Schoups, A.A.1    De Potter, W.P.2
  • 141
    • 0022885986 scopus 로고
    • Phosphorylation/dephosphorylation of the beta-adrenergic receptor regulates its functional coupling to adenylate cyclase and subcellular distribution
    • Sibley D.R., Strasser R.H., Benovic J.L., Daniel K., Lefkowitz R.J. Phosphorylation/dephosphorylation of the beta-adrenergic receptor regulates its functional coupling to adenylate cyclase and subcellular distribution. Proceedings of the National Acadamie of Sciences U S A. 83(24):1986;9408-9412.
    • (1986) Proceedings of the National Acadamie of Sciences U S A , vol.83 , Issue.24 , pp. 9408-9412
    • Sibley, D.R.1    Strasser, R.H.2    Benovic, J.L.3    Daniel, K.4    Lefkowitz, R.J.5
  • 143
    • 0020158830 scopus 로고
    • A possible role of serotonin receptors in antidepressant drug action
    • Snyder S.H., Peroutka S.J. A possible role of serotonin receptors in antidepressant drug action. Pharmacopsychiatria. 15(4):1982;131-134.
    • (1982) Pharmacopsychiatria , vol.15 , Issue.4 , pp. 131-134
    • Snyder, S.H.1    Peroutka, S.J.2
  • 144
    • 0022580619 scopus 로고
    • In vivo regulation of the serotonin-2 receptor in rat brain
    • Stockmeier C.A., Kellar K.J. In vivo regulation of the serotonin-2
    • (1986) Life Sciences , vol.38 , Issue.2 , pp. 117-127
    • Stockmeier, C.A.1    Kellar, K.J.2
  • 145
    • 0020625373 scopus 로고
    • Effect of chronic antidepressant treatment and subsequent withdrawal on [3H]-5-hydroxytryptamine and [3H]-spiperone binding in rat frontal cortex and serotonin receptor mediated behaviour
    • Stolz J.F., Marsden C.A., Middlemiss D.N. Effect of chronic antidepressant treatment and subsequent withdrawal on [3H]-5-hydroxytryptamine and [3H]-spiperone binding in rat frontal cortex and serotonin receptor mediated behaviour. Psychopharmacology. 80:1983;150-155.
    • (1983) Psychopharmacology , vol.80 , pp. 150-155
    • Stolz, J.F.1    Marsden, C.A.2    Middlemiss, D.N.3
  • 146
    • 0027413354 scopus 로고
    • 2 receptors following chronic treatment with amperozide
    • 2 receptors following chronic treatment with amperozide. Journal of Receptor Research. 13:1993;379-392.
    • (1993) Journal of Receptor Research , vol.13 , pp. 379-392
    • Svartengren, J.O.1
  • 148
    • 0018263658 scopus 로고
    • Feedback inhibition of brain noradrenaline neurons by tricyclic antidepressants: Alpha-receptor mediation
    • Svensson T.H., Usdin T. Feedback inhibition of brain noradrenaline neurons by tricyclic antidepressants: alpha-receptor mediation. Science. 202(4372):1978;1089-1091.
    • (1978) Science , vol.202 , Issue.4372 , pp. 1089-1091
    • Svensson, T.H.1    Usdin, T.2
  • 149
    • 0030716407 scopus 로고    scopus 로고
    • Phosphorylation of phospholipase C-coupled receptors
    • Tobin A.B. Phosphorylation of phospholipase C-coupled receptors. Pharmacological Therapeutics. 75(2):1997;135-151.
    • (1997) Pharmacological Therapeutics , vol.75 , Issue.2 , pp. 135-151
    • Tobin, A.B.1
  • 150
    • 0029025072 scopus 로고
    • Chronic administration of the antidepressants phenelzine, despiramine, clomipramine, or matrotiline decreases binding to 5-hydroxytryptamine2A receptors without affecting benzodiazepine binding sites
    • Todd K.G., McManus D.J., Baker G.B. Chronic administration of the antidepressants phenelzine, despiramine, clomipramine, or matrotiline decreases binding to 5-hydroxytryptamine2A receptors without affecting benzodiazepine binding sites. Cellular and Molecular Neurobiology. 15(3):1995;361-370.
    • (1995) Cellular and Molecular Neurobiology , vol.15 , Issue.3 , pp. 361-370
    • Todd, K.G.1    McManus, D.J.2    Baker, G.B.3
  • 151
    • 0028235547 scopus 로고
    • Antagonist-mediated down-regulation of 5-hydroxytryptamine type 2 receptor gene expression: Modulation of transcription
    • Toth M., Shenk T. Antagonist-mediated down-regulation of 5-hydroxytryptamine type 2 receptor gene expression: Modulation of transcription. Molecular Pharmacology. 45:1994;1095-1100.
    • (1994) Molecular Pharmacology , vol.45 , pp. 1095-1100
    • Toth, M.1    Shenk, T.2
  • 153
  • 154
    • 0026510181 scopus 로고
    • Long-term administration of m-chlorophenylpiperazine (mCPP) to rats induces changes in serotonin receptor binding, dopamine levels and locomotor activity without altering prolactin and corticosterone secretion
    • Ulrichsen J., Partilla J.S., Dax E.M. Long-term administration of m-chlorophenylpiperazine (mCPP) to rats induces changes in serotonin receptor binding, dopamine levels and locomotor activity without altering prolactin and corticosterone secretion. Psychopharmacology (Berlin). 107(2-3):1992;229-235.
    • (1992) Psychopharmacology (Berlin) , vol.107 , Issue.2-3 , pp. 229-235
    • Ulrichsen, J.1    Partilla, J.S.2    Dax, E.M.3
  • 161
    • 0024560135 scopus 로고
    • Effects of acute and chronic treatments with clozapine and haloperidol on serotonin (5-HT2) and dopamine (D2) receptors in the rat brain
    • Wilmot C.A., Szczepanik A.M. Effects of acute and chronic treatments with clozapine and haloperidol on serotonin (5-HT2) and dopamine (D2) receptors in the rat brain. Brain Research. 487(2):1989;288-298.
    • (1989) Brain Research , vol.487 , Issue.2 , pp. 288-298
    • Wilmot, C.A.1    Szczepanik, A.M.2
  • 162
    • 0027404263 scopus 로고
    • Beta-adrenergic receptor sequestration. A potential mechanism of receptor resensitization
    • Yu S.S., Lefkowitz R.J., Hausdorff W.P. Beta-adrenergic receptor sequestration. A potential mechanism of receptor resensitization. Journal of Biological Chemistry. 268(1):1993;337-341.
    • (1993) Journal of Biological Chemistry , vol.268 , Issue.1 , pp. 337-341
    • Yu, S.S.1    Lefkowitz, R.J.2    Hausdorff, W.P.3
  • 163
    • 0030766471 scopus 로고    scopus 로고
    • A central role for beta-arrestins and clathrin-coated vesicle-mediated endocytosis in beta2-adrenergic receptor resensitization. Differential regulation of receptor resensitization in two distinct cell types
    • Zhang J., Barak L.S., Winkier K.E., Caron M.G., Ferguson S.S. A central role for beta-arrestins and clathrin-coated vesicle-mediated endocytosis in beta2-adrenergic receptor resensitization. Differential regulation of receptor resensitization in two distinct cell types. Journal of Biological Chemistry. 272:1997;27005-270014.
    • (1997) Journal of Biological Chemistry , vol.272 , pp. 27005-270014
    • Zhang, J.1    Barak, L.S.2    Winkier, K.E.3    Caron, M.G.4    Ferguson, S.S.5


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.