SCOPUS 정보 검색 플랫폼

Volumn 58, Issue 16, 2002, Pages 3111-3128

The mono-functionalization of symmetrical polyamines

(3) Bender, John A a Meanwell, Nicholas A a Wang, Tao a

Author keywords

Acylation; Alkylation; Arylation; Aza macrocycles; Cyclam; Cyclen; Desymmetrization; Diamines; Piperazines; Regiocontrol

Indexed keywords

1,1' [1,4 PHENYLENEBIS(METHYLENE)]BIS(1,4,8,11 TETRAAZACYCLOTETRADECANE); ANTIINFECTIVE AGENT; AZIRIDINE DERIVATIVE; BUSPIRONE; CIPROFLOXACIN; EPOXIDE; ETHYLENEDIAMINE; HALIDE; MACROCYCLIC COMPOUND; PIPERANOMETOZINE; POLYAMINE DERIVATIVE; TOLUENESULFONIC ACID DERIVATIVE;

ACYLATION; ALKYLATION; AMINATION; CHEMICAL REACTION; CLINICAL TRIAL; HUMAN; HUMAN IMMUNODEFICIENCY VIRUS INFECTION; METHODOLOGY; MICHAEL ADDITION; ORGANIC CHEMISTRY; PRIORITY JOURNAL; REVIEW; STOICHIOMETRY; SYNTHESIS;

HUMAN IMMUNODEFICIENCY VIRUS;

EID: 0037090376 PISSN: 00404020 EISSN: None Source Type: Journal
DOI: 10.1016/S0040-4020(02)00165-5 Document Type: Review

Times cited : (49)

References (84)

1
- 0021348257
- (1984) Drugs , vol.27 , pp. 6-44
- Holmes, B.¹ Brogden, R.N.² Heel, R.C.³ Speight, T.M.⁴ Avery, G.S.⁵

2
- 0025650293
- (1990) Drugs , vol.40 , pp. 762-781
- Campoli-Richards, D.M.¹ Buckley, M.M.² Fitton, A.³

3
- 77953469244
- (1980) Anal. Profiles Drug Subst. , vol.9 , pp. 543-581
- Post, A.¹ Warren, R.J.² Zarembo, J.E.³

4
- 0023875893
- (1988) Drugs , vol.35 , pp. 373-447
- Campoli-Richards, D.M.¹ Monk, J.P.² Price, A.³ Benfield, P.⁴ Todd, P.A.⁵ Ward, A.⁶

5
- 0031016120
- (1997) Drugs , vol.53 , pp. 281-298
- Fulton, B.¹ Goa, K.L.²

6
- 0014573535
- (1969) J. Med. Chem. , vol.12 , pp. 876-881
- Wu, Y.-H.¹ Smith, K.R.² Rayburn, J.W.³ Kissel, J.W.⁴

7
- 0027165519
- (1993) Cardiovasc. Drug Rev. , vol.11 , pp. 1-11
- Feldman, A.M.¹

8
- 0035806208
- (2001) Tetrahedron , vol.57 , pp. 4801-4815
- Lee, S.H.¹ Cheong, C.S.²

9
- 0033214304
- (1999) J. Org. Chem. , vol.64 , pp. 7661-7662
- Wang, T.¹ Zhang, Z.² Meanwell, N.A.³

10
- 0000582870
- (2000) Synthesis , pp. 361-363
- Lai, L.-L.¹ Wang, E.² Luh, B.-J.³

11
- 0034921421
- (2001) Synthesis , pp. 1471-1478
- Picard, C.¹ Arnaud, N.² Tisnes, P.³

12
- 33750309194
- (1995) Angew. Chem., Int. Ed. Engl. , vol.34 , pp. 259-281
- Trost, B.M.¹

13
- 0031829003
- (1998) Synth. Commun. , pp. 2659-2664
- Fu, X.¹ Gong, C.² Ma, X.³ Wen, S.⁴

14
- 0023598499
- (1987) Yakugaku Zasshi , vol.107 , pp. 732-737
- Yokoo, N.¹ Hattori, E.² Hirata, M.³ Watanabe, K.⁴ Sato, F.⁵ Nagakura, M.⁶ Fujii, S.⁷

15
- 0028783526
- (1995) Arch. Pharm. (Weinheim) , vol.328 , pp. 654-658
- Corsano, S.¹ Strappaghetti, G.² Scapicchi, R.³ Lucacchin, A.⁴ Senatore, G.⁵

16
- 0008813327
- (1985) Collect. Czech. Chem. Commun. , vol.50 , pp. 1201-1211
- Kafka, S.¹ Cermak, J.² Novak, T.³ Pudil, F.⁴ Viden, I.⁵ Ferles, M.⁶

17
- 0026074336
- (1991) Tetrahedron Lett. , vol.32 , pp. 639-642
- Bernard, H.¹ Yaouanc, J.-J.² Clement, J.C.³ Des Abbayes, H.⁴ Handel, H.⁵

18
- 0032580321
- (1998) Tetrahedron Lett. , vol.39 , pp. 2659-2662
- Maillet, M.¹ Kwok, C.S.² Noujaim, A.A.³ Snieckus, V.⁴

19
- 0029041599
- (1995) J. Chem. Soc., Chem. Commun. , pp. 1233-1234
- Roignant, A.¹ Gardinier, I.² Bernard, H.³ Yaouanc, J.-J.⁴ Handel, H.⁵

20
- 33748214807
- (1991) Angew. Chem., Int. Ed. Engl. , vol.30 , pp. 560-561
- Filali, A.¹ Yaouanc, J.-J.² Handel, H.³

21
- 0031822843
- (1998) Synth. Commun. , vol.28 , pp. 2903-2906
- Guillaume, D.¹ Marshall, G.R.²

22
- 0027999746
- (1994) Tetrahedron Lett. , vol.35 , pp. 9075-9078
- Burguete, M.I.¹ Escuder, B.² Luis, S.V.³ Miravet, J.F.⁴ Garcia-Espana, E.⁵

23
- 0030716938
- (1997) Tetrahedron , vol.53 , pp. 16169-16176
- Burguete, M.I.¹ Escuder, B.² Frias, J.C.³ Luis, S.V.⁴ Miravet, J.F.⁵ Garcia-Espana, E.⁶

24
- 0002730009
- (1998) Chem. Commun. , pp. 1823-1824
- Burguete, M.I.¹ Garcia-Espana, E.² Luis, S.V.³ Miravet, J.F.⁴ Paya, L.⁵ Querol, M.⁶ Soriano, C.⁷

25
- 0035901340
- (2001) Tetrahedron , vol.57 , pp. 2385-2390
- Chubura, F.¹ Le Baccon, M.² Handel, H.³

26
- 0034062515
- (2000) Mol. Pharmacol. , vol.57 , pp. 833-839
- DeClerq, E.¹

27
- 0034899714
- (2001) Expert Opin. Ther. Patents , vol.11 , pp. 1245-1252
- Mastrolorenzo, A.¹ Scozzafava, A.² Supuran, C.T.³

28
- 0024510819
- (1989) Tetrahedron , vol.45 , pp. 219-226
- Helps, I.M.¹ Parker, D.² Morphy, J.R.³ Chapman, J.⁴

29
- 0000722487
- (1995) Bull. Chem. Soc. Jpn , vol.68 , pp. 2465-2469
- Tucker, J.H.R.¹ Shionoya, M.² Koike, T.³ Kimura, E.⁴

30
- 0031575618
- (1997) Tetrahedron Lett. , vol.38 , pp. 1261-1264
- De Koning, C.B.¹ Hancock, R.D.² Van Otterlo, W.A.³

31
- 9744268040
- (1995) J. Chem. Soc., Chem. Commun. , pp. 415-416
- De Sousa, A.S.¹ Hancock, R.D.²

32
- 0008810103
- (1991) Huaxue , vol.49 , pp. 267-270
- Le, C.-H.¹

33
- 0000360603
- (1990) Zh. Obshch. Khim. , vol.60 , pp. 2721-2725
- Bobylev, V.A.¹ Chechik, V.O.²

34
- 0024579002
- (1989) J. Med. Chem. , vol.32 , pp. 236-243
- Westerberg, D.A.¹ Carney, P.L.² Rogers, P.E.³ Kline, S.J.⁴ Johnson, D.K.⁵

35
- 0000494451
- (1999) J. Chem. Soc., Perkin Trans 1 , pp. 811-815
- Fensterbank, H.¹ Zhu, J.² Riou, D.³ Larpent, C.⁴

36
- 0008863329
- (1997) Chem. Lett. , pp. 275-376
- Matsuyama, H.¹ Itoh, N.² Yoshida, M.³ Kamigatra, N.⁴ Sasaki, S.⁵ Iyoda, M.⁶

37
- 0025191178
- (1990) Tetrahedron Lett. , vol.31 , pp. 839-840
- Pastor, S.¹ Togni, A.²

38
- 0028813685
- (1995) Tetrahedron , vol.51 , pp. 1197-1208
- Granier, C.¹ Guillard, R.²

39
- 0000680342
- (1988) Tetrahedron Lett. , vol.29 , pp. 1991-1992
- Pietrusiewicz, K.M.¹ Zablocka, M.²

40
- 0001659332
- (1987) J. Org. Chem. , vol.52 , pp. 2592-2594
- Jacobson, A.R.¹ Makris, A.N.² Sayre, L.M.³

41
- 0001811914
- (1929) J. Chem. Soc. , pp. 39-51
- Moore, T.S.¹ Boyle, M.² Thorn, V.M.³

42
- 84970543232
- (1956) Aust. J. Chem. , vol.9 , pp. 397-405
- Cymerman-Craig, J.¹ Rogers, W.P.² Tate, M.E.³

43
- 0002783668
- (1976) Org. Prep. Proced. Int. , vol.8 , pp. 85-86
- Desai, M.¹ Watthey, J.W.H.² Zuckerman, M.³

44
- 84987478892
- (1984) Synthesis , pp. 1032-1033
- Atwell, G.J.¹ Denny, W.A.²

45
- 53349112702
- (1990) Synth. Commun. , vol.20 , pp. 2559-2564
- Krapcho, A.P.¹ Kuell, C.S.²

46
- 0002096853
- (1997) Synlett , pp. 1190-1192
- Guilard, R.¹ Bessmertnykh, A.G.² Beletskaya, I.P.³

47
- 0030841926
- (1997) Synthesis , pp. 759-763
- Kovacs, Z.¹ Sherry, A.D.²

48
- 0030932589
- (1997) Synth. Commun. , vol.27 , pp. 979-987
- Rabiet, F.¹ Denat, F.² Guilard, R.³

49
- 37049094242
- (1978) J. Chem. Soc., Chem. Commun. , pp. 471-472
- Barrett, A.G.M.¹ Lana, J.C.A.²

50
- 37049099720
- (1980) J. Chem. Soc., Chem. Commun. , pp. 300-301
- Barrett, A.G.M.¹ Lana, J.C.A.² Tograie, S.³

51
- 0008812936
- (1994) Bull. Korean Chem. Soc. , vol.15 , pp. 1025-1027
- Ham, J.-Y.¹ Kang, H.-S.²

52
- 0000582870
- (2000) Synthesis , pp. 361-363
- Lai, L.-L.¹ Wang, E.² Luh, B.-J.³

53
- 0000379540
- (2000) Heterocycles , vol.53 , pp. 529-533
- Chung, I.H.¹ Cha, K.S.² Seo, J.H.³ Kim, J.H.⁴ Chung, B.Y.⁵ Kim, C.S.⁶

54
- 84985079736
- (1986) J. Chin. Chem. Soc. , vol.33 , pp. 347-349
- Chen, L.-C.¹ Yang, S.-C.²

55
- 0001464057
- (1987) Synth. Commun. , vol.17 , pp. 1741-1748
- Rebelo, R.A.¹ Rezende, M.C.² Nome, F.³ Zucco, C.⁴

56
- 0026572458
- (1992) Synth. Commun. , vol.22 , pp. 1307-1318
- Kuswik-Rabiega, G.¹ Bruenger, F.W.² Miller, S.C.³

57
- 0029130012
- (1995) Tetrahedron Lett. , vol.36 , pp. 7357-7360
- Xu, D.¹ Prasad, K.² Repic, O.³ Blacklock, T.J.⁴

58
- 0030598007
- (1996) Tetrahedron Lett. , vol.37 , pp. 5301-5304
- Xu, D.¹ Mattner, P.G.² Prasad, K.³ Repic, O.⁴ Blacklock, T.J.⁵

59
- 0028072642
- (1994) Arch. Pharm. (Weinheim) , vol.327 , pp. 747-750
- Imming, P.¹ Yang, X.-G.²

60
- 0034921421
- (2001) Synthesis , pp. 1471-1478
- Picard, C.¹ Arnaud, N.² Tisnes, P.³

61
- 0042963065
- (1988) Synthesis , pp. 917-918
- Zaragoza-Dorwald, F.¹ Von Kiedrowski, G.²

62
- 0008837786
- Murthy, K. S. K; Weeratunga, G.; Zhou, T.; Guntoort, B. R. U.S. Patent 5,919, 931, July 6, 1999.

63
- 0032567392
- (1998) J. Org. Chem. , vol.63 , pp. 10015-10017
- Chou, W.-C.¹ Tan, C.-W.² Chen, S.-F.³ Ku, H.⁴

64
- 0033597262
- (1999) Tetrahedron Lett. , vol.40 , pp. 3419-3422
- Chou, W.-C.¹ Chou, M.-C.² Lu, Y.-Y.³ Chen, S.-F.⁴

65
- 0033214304
- (1999) J. Org. Chem. , vol.64 , pp. 7661-7662
- Wang, T.¹ Zhang, Z.² Meanwell, N.A.³

66
- 0023288071
- (1987) J. Mol. Catal. , vol.39 , pp. 233-236
- Jenner, G.¹ Bitsi, G.² Schleiffer, E.³

67
- 0345476938
- (1999) J. Org. Chem. , vol.64 , pp. 9201-9205
- Kihlberg, T.¹ Långström, B.²

68
- 0008832982
- (1990) Sulfur Lett. , vol.11 , pp. 201-207
- Lei, L.¹ Senning, A.²

69
- 0000626110
- (1951) J. Am. Chem. Soc. , vol.73 , pp. 3100-3125
- Bent, R.L.¹ Dessloch, J.C.² Dunnebier, F.C.³ Fassett, D.W.⁴ Glass, D.B.⁵ James, T.H.⁶ Julian, D.B.⁷ Ruby, W.R.⁸ Snell, J.M.⁹ Sterner, J.H.¹⁰ Thirtle, J.R.¹¹ Vittum, P.W.¹² Weissberger, A.¹³

70
- 0032752508
- (1999) J. Med. Chem. , vol.42 , pp. 4794-4803
- Lagu, B.¹ Tian, D.² Nagarathnam, D.³ Marzabadi, M.R.⁴ Wong, W.C.⁵ Miao, S.W.⁶ Zhang, F.⁷ Sun, W.⁸ Chiu, G.⁹ Fang, J.¹⁰ Forray, C.¹¹ Chang, R.S.L.¹² Ransom, R.W.¹³ Chen, T.B.¹⁴ O'Malley, S.¹⁵ Zhang, K.¹⁶ Vyas, K.P.¹⁷ Gluchowski, C.¹⁸

71
- 0025726861
- (1991) J. Med. Chem. , vol.34 , pp. 1155-1161
- Hagen, S.E.¹ Domagala, J.M.² Heifetz, C.L.³ Johnson, J.⁴

72
- 0033618356
- (1999) Tetrahedron Lett. , vol.40 , pp. 5655-5659
- Hepperle, M.¹ Eckert, J.² Gala, D.³

73
- 0033618313
- (1999) Tetrahedron Lett. , vol.40 , pp. 5661-5665
- Eckert, J.¹ Chan, T.-M.² Osterman, R.M.³ Lambert, J.B.⁴ Gala, D.⁵

74
- 0034650425
- (2000) Tetrahedron Lett. , vol.41 , pp. 313-316
- Beletskaya, I.P.¹ Artamkina, G.A.² Ivushkin, V.A.³ Guilard, R.⁴

75
- 0030600196
- (1996) Tetrahedron Lett. , vol.37 , pp. 4463-4466
- Zhao, S.-H.¹ Miller, A.K.² Berger, J.³ Flippin, L.A.⁴

76
- 0032079256
- (1998) Tetrahedron , vol.54 , pp. 4811-4818
- Morita, S.¹ Kitano, K.² Matsubara, J.³ Ohtani, T.⁴ Kawano, Y.⁵ Otsubo, K.⁶ Uchida, M.⁷

77
- 0031592580
- (1997) Tetrahedron Lett. , vol.38 , pp. 2287-2290
- Beletskaya, I.P.¹ Bessmertnykh, A.G.² Guilard, R.³

78
- 0032826764
- (1999) Synlett , pp. 1459-1461
- Beletskaya, I.P.¹ Bessmertnykh, A.G.² Guilard, R.³

79
- 0001038733
- (1998) Acc. Chem. Res. , vol.31 , pp. 805-818
- Wolfe, J.P.¹ Wahaw, S.² Marcoux, J.-F.³ Buchwald, S.L.⁴

80
- 0032541260
- (1998) Angew. Chem., Int. Ed. Engl. , vol.37 , pp. 2046-2067
- Hartwig, J.F.¹

81
- 0024532177
- (1989) J. Med. Chem. , vol.32 , pp. 42-46
- Morikawa, A.¹ Sone, T.² Asano, T.³

82
- 0024492468
- (1989) J. Med. Chem. , vol.32 , pp. 46-50
- Morikawa, A.¹ Sone, T.² Asano, T.³

83
- 0034177625
- (2000) Heterocycles , vol.53 , pp. 797-804
- Varlet, D.¹ Fourmaintraux, E.² Depreux, P.³ Lesieur, D.⁴

84
- 0037039904
- (2002) J. Org. Chem. , vol.67 , pp. 674-683
- Salvatore, R.N.¹ Nagle, A.S.² Jung, K.Y.³

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.