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Volumn 10, Issue 4, 2002, Pages 929-934

Novel steroidal vinyl fluorides as inhibitors of steroid C17(20) lyase

(9) Burkhart, Joseph P a Weintraub, Philip M a Gates, Cynthia A a Resvick, Robert J a Vaz, Roy J a Friedrich, Dirk a Angelastro, Michael R a Bey, Philippe a Peet, Norton P a

a SANOFI (France)

Author keywords

[No Author keywords available]

Indexed keywords

20 FLUOROPREGNA 5,17(20) DIENE 3,21 DIOL; 20 FLUOROPREGNA 5,17(20)DIEN 3 OL; ALKENE DERIVATIVE; LYASE INHIBITOR; ORGANOFLUORINE DERIVATIVE; PREGNENOLONE DERIVATIVE; STEROID 17,20 LYASE; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; CONTROLLED STUDY; DRUG DESIGN; DRUG STRUCTURE; DRUG SYNTHESIS; ENANTIOMER; ENZYME INHIBITION; IN VITRO STUDY; MALE; MONKEY; NONHUMAN; NUCLEAR MAGNETIC RESONANCE; STRUCTURE ACTIVITY RELATION; TESTIS;

ANIMALS; DOSE-RESPONSE RELATIONSHIP, DRUG; ENZYME INHIBITORS; MACACA FASCICULARIS; PREGNENOLONE; STEROID 17-ALPHA-HYDROXYLASE; STEROIDS, FLUORINATED; STRUCTURE-ACTIVITY RELATIONSHIP; VINYL COMPOUNDS;

EID: 0036172443 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/S0968-0896(01)00354-6 Document Type: Article

Times cited : (35)

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