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Proceedings of the National Academy of Sciences of the United States of America

Volumn 98, Issue 22, 2001, Pages 12718-12723

SCH-C (SCH 351125), an orally bioavailable, small molecule antagonist of the chemokine receptor CCR5, is a potent inhibitor of HIV-1 infection in vitro and in vivo

(25) Strizki, Julie M a Xu, Serena a Wagner, Nicole E a Wojcik, Lisa a Liu, Jia a Hou, Yan a Endres, Michael a,f Palani, Anandan a Shapiro, Sherry a Clader, John W a Greenlee, William J a Tagat, Jayaram R a McCombie, Stuart a Cox, Kathleen a Fawzi, Ahmad B a Chou, Chuan Chu a Pugliese Sivo, Catherine a Davies, Liza a Moreno, Mary E b Ho, David D c more..

a MERCK RESEARCH LABORATORIES (United States)

b UNIVERSITY OF CALIFORNIA (United States)

c ROCKEFELLER UNIVERSITY (United States)

d UNIVERSITY HOSPITAL ZURICH (Switzerland)

e WEILL CORNELL MEDICAL COLLEGE (United States)

f MEDAREX INC (United States)

Author keywords

[No Author keywords available]

Indexed keywords

4 [(4 BROMOPHENYL)(ETHOXYIMINO)METHYL] 1' [(2,4 DIMETHYL 3 PYRIDINYL)CARBONYL] 4' METHYL 1,4' BIPIPERIDINE; CHEMOKINE RECEPTOR CCR5; CHEMOKINE RECEPTOR CCR5 ANTAGONIST; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL MODEL; ANTIVIRAL ACTIVITY; ARTICLE; ASTROCYTOMA; CONTROLLED STUDY; DRUG BIOAVAILABILITY; DRUG HALF LIFE; DRUG POTENCY; HUMAN; HUMAN CELL; HUMAN IMMUNODEFICIENCY VIRUS 1; HUMAN IMMUNODEFICIENCY VIRUS INFECTION; MOUSE; NONHUMAN; PRIORITY JOURNAL; RECEPTOR BINDING; SIGNAL TRANSDUCTION; VIRUS INHIBITION; VIRUS REPLICATION;

ACQUIRED IMMUNODEFICIENCY SYNDROME; ANIMALS; ANTI-HIV AGENTS; CYCLIC N-OXIDES; HIV-1; HUMANS; MACACA FASCICULARIS; MALE; MICE; MICE, SCID; PIPERIDINES; PYRIDINES; RANTES; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, CCR5;

ANIMALIA; HUMAN IMMUNODEFICIENCY VIRUS; HUMAN IMMUNODEFICIENCY VIRUS 1; PRIMATES; RNA VIRUSES; RODENTIA;

EID: 0035940445 PISSN: 00278424 EISSN: None Source Type: Journal
DOI: 10.1073/pnas.221375398 Document Type: Article

Times cited : (324)

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