Characterization of the efflux transport of 17β-estradiol-D-17β-glucuronide from the brain across the blood-brain barrier

Journal of Pharmacology and Experimental Therapeutics

Volumn 298, Issue 1, 2001, Pages 316-322

  Sugiyama, Daisuke ^a   Kusuhara, Hiroyuki ^a   Shitara, Yoshihisa ^b   Abe, Takaaki ^c   Meier, Peter J ^d   Sekine, Takashi ^a   Endou, Hitoshi ^e   Suzuki, Hiroshi ^a   Sugiyama, Yuichi ^a  

^a UNIVERSITY OF TOKYO   (Japan)

^b KITASATO UNIVERSITY   (Japan)

^c TOHOKU UNIVERSITY SCHOOL OF MEDICINE   (Japan)

^d UNIVERSITY HOSPITAL ZURICH   (Switzerland)

^e KYORIN UNIVERSITY   (Japan)

Author keywords

[No Author keywords available]

Indexed keywords

17BETA ESTRADIOL DEXTRO 17BETA GLUCURONIDE; 4 AMINOHIPPURIC ACID; CARRIER PROTEIN; DIGOXIN; ESTRADIOL DERIVATIVE; ORGANIC ANION TRANSPORTER 1; ORGANIC ANION TRANSPORTER 2; PROBENECID; TAUROCHOLIC ACID; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL TISSUE; ANION TRANSPORT; ARTICLE; BINDING AFFINITY; BLOOD BRAIN BARRIER; CONTROLLED STUDY; DRUG BINDING; DRUG ELIMINATION; DRUG INHIBITION; DRUG UPTAKE; GENETIC TRANSFECTION; MALE; NONHUMAN; PRIORITY JOURNAL; RAT;

ANIMALS; ANION TRANSPORT PROTEINS; BLOOD-BRAIN BARRIER; BRAIN; CARRIER PROTEINS; DIGOXIN; ENZYME INHIBITORS; ESTRADIOL; GLUCURONATES; MALE; MICROINJECTIONS; ORGANIC ANION TRANSPORTERS, SODIUM-INDEPENDENT; P-AMINOHIPPURIC ACID; PROBENECID; RATS; RATS, WISTAR; TAUROCHOLIC ACID;

EID: 0034978374     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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