메뉴 건너뛰기




Volumn 129, Issue 6, 2000, Pages 1183-1193

Characterization of [Nphe1]nociceptin(1-13)NH2, a new selective nociceptin receptor antagonist

Author keywords

Analgesia; Isolated tissues; Morphine; Mouse tail withdrawal assay; Native and recombinant receptors; Nociceptin; Nociceptin receptor antagonist

Indexed keywords

CYCLIC AMP; MORPHINE; NALOXONE; NOCICEPTIN; NOCICEPTIN RECEPTOR; PHENYL NOCICEPTIN; RECEPTOR BLOCKING AGENT; RECOMBINANT RECEPTOR; UNCLASSIFIED DRUG;

EID: 0034101842     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0703169     Document Type: Article
Times cited : (196)

References (48)
  • 2
    • 0032523346 scopus 로고    scopus 로고
    • Phe1psi(CH2-NH)Gly2nociceptin-(1-13)NH2 is an agonist of the nociceptin (ORL1) receptor
    • BUTOUR, J.L., MOISAND, C., MOLLEREAU, C. & MEUNIER, J.C. (1998). [Phe1psi(CH2-NH)Gly2]nociceptin-(1-13)NH2 is an agonist of the nociceptin (ORL1) receptor. Eur. J. Pharmacol., 349, R5-R6.
    • (1998) Eur. J. Pharmacol. , vol.349
    • Butour, J.L.1    Moisand, C.2    Mollereau, C.3    Meunier, J.C.4
  • 3
    • 0031694279 scopus 로고    scopus 로고
    • Pharmacological characterization of the nociceptin receptor binding hyperalgesia in the mouse tail withdrawal assay
    • CALO, G., RIZZI, A., MARZOLA, G., GUERRINI, R., SALVADORI, S., BEANI, L., REGOLI, D. & BIANCHI, C. (1998). Pharmacological characterization of the nociceptin receptor binding hyperalgesia in the mouse tail withdrawal assay. Br. J. Pharmacol., 125, 373-378.
    • (1998) Br. J. Pharmacol. , vol.125 , pp. 373-378
    • Calo, G.1    Rizzi, A.2    Marzola, G.3    Guerrini, R.4    Salvadori, S.5    Beani, L.6    Regoli, D.7    Bianchi, C.8
  • 4
    • 0032408286 scopus 로고    scopus 로고
    • Reverse physiology: Discovery of the novel neuropeptide, orphanin FQ/nociceptin
    • CIVELLI, O., NOTHACKER, H.P. & REINSCHEID, R. (1998). Reverse physiology: discovery of the novel neuropeptide, orphanin FQ/nociceptin. Crit. Rev. Neurobiol., 12, 163-176.
    • (1998) Crit. Rev. Neurobiol. , vol.12 , pp. 163-176
    • Civelli, O.1    Nothacker, H.P.2    Reinscheid, R.3
  • 5
    • 0030462638 scopus 로고    scopus 로고
    • Nociceptin receptor coupling to a potassium conductance in rat locus coeruleus neurones in vitro
    • CONNOR, M., VAUGHAN, C.W., CHIENG, B. & CHRISTIE, M.J. (1996a). Nociceptin receptor coupling to a potassium conductance in rat locus coeruleus neurones in vitro. Br. J. Pharmacol., 119, 1614-1618.
    • (1996) Br. J. Pharmacol. , vol.119 , pp. 1614-1618
    • Connor, M.1    Vaughan, C.W.2    Chieng, B.3    Christie, M.J.4
  • 6
    • 0029665959 scopus 로고    scopus 로고
    • The effect of nociceptin on Ca2+ channel current and intracellular Ca2+ in the SH-SY5Y human neuroblastoma cell line
    • CONNOR, M., YEO, A. & HENDERSON, G. (1996b). The effect of nociceptin on Ca2+ channel current and intracellular Ca2+ in the SH-SY5Y human neuroblastoma cell line. Br. J. Pharmacol., 118, 205-207.
    • (1996) Br. J. Pharmacol. , vol.118 , pp. 205-207
    • Connor, M.1    Yeo, A.2    Henderson, G.3
  • 7
    • 0030586364 scopus 로고    scopus 로고
    • The novel neuropeptide orphanin FQ fails to produce conditioned place preference or aversion
    • DEVINE, D.P., REINSCHEID, R.K., MONSMA, F.J., CIVELLI, O. & AKIL, H. (1996). The novel neuropeptide orphanin FQ fails to produce conditioned place preference or aversion. Brain Res., 727, 225-229.
    • (1996) Brain Res. , vol.727 , pp. 225-229
    • Devine, D.P.1    Reinscheid, R.K.2    Monsma, F.J.3    Civelli, O.4    Akil, H.5
  • 9
    • 0029901195 scopus 로고    scopus 로고
    • Inhibition of tachykinin release from peripheral endings of sensory nerves by nociceptin, a novel opioid peptide
    • GIULIANI, S. & MAGGI, C.A. (1996). Inhibition of tachykinin release from peripheral endings of sensory nerves by nociceptin, a novel opioid peptide. Br. J. Pharmacol., 118, 1567-1569.
    • (1996) Br. J. Pharmacol. , vol.118 , pp. 1567-1569
    • Giuliani, S.1    Maggi, C.A.2
  • 11
    • 0031006367 scopus 로고    scopus 로고
    • Address and message sequences for the nociceptin receptor: A structure-activity study of nociceptin-(1-13)-peptide amide
    • GUERRINI, R., CALO, G., RIZZI, A., BIANCHI, C., LAZARUS, L.H., SALVADORI, S., TEMUSSI, P.A. & REGOLI, D. (1997). Address and message sequences for the nociceptin receptor: a structure-activity study of nociceptin-(1-13)-peptide amide. J. Med. Chem., 40, 1789-1793.
    • (1997) J. Med. Chem. , vol.40 , pp. 1789-1793
    • Guerrini, R.1    Calo, G.2    Rizzi, A.3    Bianchi, C.4    Lazarus, L.H.5    Salvadori, S.6    Temussi, P.A.7    Regoli, D.8
  • 13
    • 0003274798 scopus 로고    scopus 로고
    • The new approach to opioid receptors
    • SA 5.3
    • HAMON, M. (1998). The new approach to opioid receptors. N.S. Arch. Pharmacol., 358 (Suppl 2), SA 5.3.
    • (1998) N.S. Arch. Pharmacol. , vol.358 , Issue.SUPPL. 2
    • Hamon, M.1
  • 14
    • 0033621642 scopus 로고    scopus 로고
    • 2 on nociceptin receptor mediated inhibition of cAMP formation in Chinese ovary cells stably expressing the recombinant human nociceptin receptor
    • 2 on nociceptin receptor mediated inhibition of cAMP formation in Chinese ovary cells stably expressing the recombinant human nociceptin receptor. Neurosci. Lett., 278, 109-112.
    • (2000) Neurosci. Lett. , vol.278 , pp. 109-112
    • Hashimoto, Y.1    Calo', G.2    Guerrini, R.3    Smith, G.4    Lambert, D.G.5
  • 15
    • 0023709280 scopus 로고    scopus 로고
    • Evidence that the kappa agonist U50488H has non-opioid actions
    • HAYES, A.G., BIRCH, P.P. & CAVICCHINI, E. (1998). Evidence that the kappa agonist U50488H has non-opioid actions. J. Pharm. Pharmacol., 40, 718-720.
    • (1998) J. Pharm. Pharmacol. , vol.40 , pp. 718-720
    • Hayes, A.G.1    Birch, P.P.2    Cavicchini, E.3
  • 16
    • 0030848732 scopus 로고    scopus 로고
    • Coupling of the cloned rat k-opioid receptor to adenylyl cyclase is dependent on receptor expression
    • HIRST, R.A., HIROTA, K., GRANDY, D.K. & LAMBERT, D.G. (1997). Coupling of the cloned rat k-opioid receptor to adenylyl cyclase is dependent on receptor expression. Neurosci. Lett., 232, 119-122.
    • (1997) Neurosci. Lett. , vol.232 , pp. 119-122
    • Hirst, R.A.1    Hirota, K.2    Grandy, D.K.3    Lambert, D.G.4
  • 17
    • 0031776122 scopus 로고    scopus 로고
    • Effects of C-terminal truncation of the recombinant delta opioid receptor on phospholipase C and anenylyl cyclase coupling
    • HIRST, R.A., SMART, D., DEVI, L.A. & LAMBERT, D.G. (1998). Effects of C-terminal truncation of the recombinant delta opioid receptor on phospholipase C and anenylyl cyclase coupling. J. Neurochem., 70, 2273-2278.
    • (1998) J. Neurochem. , vol.70 , pp. 2273-2278
    • Hirst, R.A.1    Smart, D.2    Devi, L.A.3    Lambert, D.G.4
  • 18
    • 0029013360 scopus 로고
    • Analysis of selective binding epitopes for the kappa opioid receptor antagonist norbinaltorphimine
    • HJORTH, S.A., THIRSTRUP, K., GRANDY, D.K. & SCHWARTZ, T.W. (1995). Analysis of selective binding epitopes for the kappa opioid receptor antagonist norbinaltorphimine. Mol. Pharmacol., 47, 1089-1094.
    • (1995) Mol. Pharmacol. , vol.47 , pp. 1089-1094
    • Hjorth, S.A.1    Thirstrup, K.2    Grandy, D.K.3    Schwartz, T.W.4
  • 20
    • 0029010943 scopus 로고
    • International Union of Pharmacology Committee on receptor nomenclature and drug classification X1 recommendation on terms and symbols in quantitative pharmacology
    • JENKINSON, D.H., BARNARD, E.A., HOYER, D., HUMPHREY, P.P.A., LEFF, P. & SHANKLEY, N.P. (1995). International Union of Pharmacology Committee on receptor nomenclature and drug classification X1 Recommendation on terms and symbols in quantitative pharmacology. Pharmacol. Rev., 47, 255-266.
    • (1995) Pharmacol. Rev. , vol.47 , pp. 255-266
    • Jenkinson, D.H.1    Barnard, E.A.2    Hoyer, D.3    Humphrey, P.P.A.4    Leff, P.5    Shankley, N.P.6
  • 21
    • 0033013383 scopus 로고    scopus 로고
    • Opioids: First lessons from knockout mice
    • KIEFFER, B.L. (1999). Opioids: first lessons from knockout mice. Trends Pharmacol. Sci., 20, 19-26.
    • (1999) Trends Pharmacol. Sci. , vol.20 , pp. 19-26
    • Kieffer, B.L.1
  • 22
    • 0030903527 scopus 로고    scopus 로고
    • Effects of sigma ligands on the nociceptin/orphanin FQ receptor co-expressed with the G-protein-activated K+ channel in Xenopus oocytes
    • KOBAYASHI, T., IKEDA, K., TOGASHI, S., ITOH, N. & KUMANISHI, T. (1997). Effects of sigma ligands on the nociceptin/orphanin FQ receptor co-expressed with the G-protein-activated K+ channel in Xenopus oocytes. Br. J. Pharmacol., 120, 986-987.
    • (1997) Br. J. Pharmacol. , vol.120 , pp. 986-987
    • Kobayashi, T.1    Ikeda, K.2    Togashi, S.3    Itoh, N.4    Kumanishi, T.5
  • 24
    • 0023850632 scopus 로고
    • Kappa-Opioid agonists produce antinociception after i.v. and i.e.v. But not intrathecal administration in the rat
    • LEIGHTON, G.E, RODRIGUEZ, R.E., HILL, R.G & HUGHES, J. (1988). kappa-Opioid agonists produce antinociception after i.v. and i.e.v. but not intrathecal administration in the rat. Br. J. Pharmacol., 93, 553-560.
    • (1988) Br. J. Pharmacol. , vol.93 , pp. 553-560
    • Leighton, G.E.1    Rodriguez, R.E.2    Hill, R.G.3    Hughes, J.4
  • 29
    • 0032796883 scopus 로고    scopus 로고
    • In vitro effects of nociceptin and [Phe1psi(Ch2-NH)Gly2]nociceptin(1-13)NH2 in the mouse and rat colon and the mouse vas deferens
    • MENZIES, J.R.W., GLEN, T., DAVIES, M.R.P., PATERSON, S.J. & CORBETT, A.D. (1999). In vitro effects of nociceptin and [Phe1psi(Ch2-NH)Gly2]nociceptin(1-13)NH2 in the mouse and rat colon and the mouse vas deferens. Eur. J. Pharmacol., 385, 217-223.
    • (1999) Eur. J. Pharmacol. , vol.385 , pp. 217-223
    • Menzies, J.R.W.1    Glen, T.2    Davies, M.R.P.3    Paterson, S.J.4    Corbett, A.D.5
  • 31
    • 0031553387 scopus 로고    scopus 로고
    • Nociceptin/orphanin FQ and the opioid receptor-like ORL1 receptor
    • MEUNIER, J.C. (1997). Nociceptin/orphanin FQ and the opioid receptor-like ORL1 receptor. Eur. J. Pharmacol., 340, 1-15.
    • (1997) Eur. J. Pharmacol. , vol.340 , pp. 1-15
    • Meunier, J.C.1
  • 35
    • 0032541091 scopus 로고    scopus 로고
    • Loss of antinociception induced by naloxone benzoylhydrazone in nociceptin receptor-knockout mice
    • NODA, Y., MAMIYA, T., NABESHIMA, T., NISHI, M., HIGASHIOKA, M. & TAKESHIMA, H. (1998). Loss of antinociception induced by naloxone benzoylhydrazone in nociceptin receptor-knockout mice. J. Biol. Chem., 273, 18047-18051.
    • (1998) J. Biol. Chem. , vol.273 , pp. 18047-18051
    • Noda, Y.1    Mamiya, T.2    Nabeshima, T.3    Nishi, M.4    Higashioka, M.5    Takeshima, H.6
  • 37
    • 0032588075 scopus 로고    scopus 로고
    • Comparison of the effects of the Phe1psi(CH2-NH)Gly2nociceptin(1-13)NH2 in rat brain, rat vas deferens and CHO cells expressing recombinant human nociceptin receptors
    • OKAWA, H., NICOL., B., BIGONI, R., HIRST, R.A., CALO, G., GUERRINI, R., ROWBOTHAM, D.J., SMART, D., MCKNIGHT, A.T. & LAMBERT, D.G. (1999). Comparison of the effects of the Phe1psi(CH2-NH)Gly2]nociceptin(1-13)NH2 in rat brain, rat vas deferens and CHO cells expressing recombinant human nociceptin receptors. Br. J. Pharmacol., 127, 123-130.
    • (1999) Br. J. Pharmacol. , vol.127 , pp. 123-130
    • Okawa, H.1    Nicol, B.2    Bigoni, R.3    Hirst, R.A.4    Calo, G.5    Guerrini, R.6    Rowbotham, D.J.7    Smart, D.8    McKnight, A.T.9    Lambert, D.G.10
  • 39
    • 0001580029 scopus 로고    scopus 로고
    • Pharmacological characterization of the nociceptin receptor mediating hyperphagia: Identification of a selective antagonist
    • in press
    • POLIDORI, C., CALO, G., CICCOCIOPPO, R., GUERRINI, R., REGOLI, D. & MASSI, M. (2000). Pharmacological characterization of the nociceptin receptor mediating hyperphagia: identification of a selective antagonist. Psychopharmacology, in press.
    • (2000) Psychopharmacology
    • Polidori, C.1    Calo, G.2    Ciccocioppo, R.3    Guerrini, R.4    Regoli, D.5    Massi, M.6
  • 42
    • 0031715554 scopus 로고    scopus 로고
    • Nociceptin inhibits noradrenaline release in the mouse brain cortex via presynaptic ORLI receptors
    • SCHLICKER, E., WERTHWEIN, S., KATHMANN, M. & BAUER, U. (1998). Nociceptin inhibits noradrenaline release in the mouse brain cortex via presynaptic ORLI receptors. N.S. Arch. Pharmacol., 358, 418-422.
    • (1998) N.S. Arch. Pharmacol. , vol.358 , pp. 418-422
    • Schlicker, E.1    Werthwein, S.2    Kathmann, M.3    Bauer, U.4
  • 43
    • 0030902326 scopus 로고    scopus 로고
    • The effects of recombinant rat mu opioid receptor activation in CHO cells on phospholipase C, [Ca2+ ]i and adenylyl cyclase
    • SMART, D., HIRST, R.A., HIROTA, K., GRANDY, D.K. & LAMBERT, D.G. (1997). The effects of recombinant rat mu opioid receptor activation in CHO cells on phospholipase C, [Ca2+ ]i and adenylyl cyclase. Br. J. Pharmacol., 120, 1165-1171.
    • (1997) Br. J. Pharmacol. , vol.120 , pp. 1165-1171
    • Smart, D.1    Hirst, R.A.2    Hirota, K.3    Grandy, D.K.4    Lambert, D.G.5
  • 45
    • 0031919105 scopus 로고    scopus 로고
    • Endogenous orphanin FQ: Evidence for a role in the modulation of electroacupuncture analgesia and the development of tolerance to analgesia produced by morphine and electroacupuncture
    • TIAN, J.H., ZHANG, W., FANG, Y., XU, W., GRANDY, D.K. & HAN, J.S. (1998). Endogenous orphanin FQ: evidence for a role in the modulation of electroacupuncture analgesia and the development of tolerance to analgesia produced by morphine and electroacupuncture. Br. J. Pharmacol., 124, 21-26.
    • (1998) Br. J. Pharmacol. , vol.124 , pp. 21-26
    • Tian, J.H.1    Zhang, W.2    Fang, Y.3    Xu, W.4    Grandy, D.K.5    Han, J.S.6
  • 46
    • 0031450208 scopus 로고    scopus 로고
    • Partial loss of tolerance liability to morphine analgesia in mice lacking the nociceptin receptor gene
    • UEDA, H., YAMAGUCHI, T., TOKUYAMA, S., INOUE, M., NISHI, M. & TAKESHIMA, H. (1997). Partial loss of tolerance liability to morphine analgesia in mice lacking the nociceptin receptor gene. Neurosci. Lett., 237, 136-138.
    • (1997) Neurosci. Lett. , vol.237 , pp. 136-138
    • Ueda, H.1    Yamaguchi, T.2    Tokuyama, S.3    Inoue, M.4    Nishi, M.5    Takeshima, H.6
  • 47
    • 0032546651 scopus 로고    scopus 로고
    • Phe1psi(CH2-NH)Gly2-nociceptin-(1-13)NH2, a proposed antagonist of the nociceptin receptor, is a potent and stable agonist in the rat spinal cord
    • XU, I.S., WIESENFELD-HALLIN, Z. & XU, X.J. (1998). [Phe1psi(CH2-NH)Gly2]-nociceptin-(1-13)NH2, a proposed antagonist of the nociceptin receptor, is a potent and stable agonist in the rat spinal cord. Neurosci. Lett., 249, 127-130.
    • (1998) Neurosci. Lett. , vol.249 , pp. 127-130
    • Xu, I.S.1    Wiesenfeld-Hallin, Z.2    Xu, X.J.3
  • 48
    • 0030777654 scopus 로고    scopus 로고
    • Orphanin FQ potentiates formalin-induced pain behavior and antagonizes morphine analgesia in rats
    • ZHU, C.B., CAO, X.D., XU, S.F. & WU, G.C. (1997). Orphanin FQ potentiates formalin-induced pain behavior and antagonizes morphine analgesia in rats. Neurosci. Lett., 235, 37-40.
    • (1997) Neurosci. Lett. , vol.235 , pp. 37-40
    • Zhu, C.B.1    Cao, X.D.2    Xu, S.F.3    Wu, G.C.4


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.