Partial to complete antagonism by putative antagonists at the wild-type α(2c)-adrenoceptor based on kinetic analyses of agonist: Antagonist interactions

British Journal of Pharmacology

Volumn 131, Issue 7, 2000, Pages 1385-1390

  Pauwels, P J ^a   Colpaert, F C ^a  

^a INSTITUT DE RECHERCHE PIERRE FABRE   (France)

Author keywords

Agonist:antagonist interactions; Recombinant human (2C) adrenoceptor; Silent antagonist

Indexed keywords

2 (2 ETHOXY 1,4 BENZODIOXAN 2 YL) 2 IMIDAZOLINE; 2 (2 METHOXY 1,4 BENZODIOXAN 2 YL) 2 IMIDAZOLINE; 6 CHLORO 2,3,4,5 TETRAHYDRO 3 METHYL 1H 3 BENZAZEPINE; ADRENALIN; ALPHA 2 ADRENERGIC RECEPTOR; ALPHA 2 ADRENERGIC RECEPTOR BLOCKING AGENT; ALPHA 2 ADRENERGIC RECEPTOR STIMULATING AGENT; BRIMONIDINE; CHIMERIC PROTEIN; CLONIDINE; IDAZOXAN; MEDETOMIDINE; OXYMETAZOLINE; TALIPEXOLE;

ARTICLE; CALCIUM TRANSPORT; CHIMERA; CHO CELL; DRUG ANTAGONISM; PRIORITY JOURNAL; RECEPTOR INTRINSIC ACTIVITY; STRUCTURE ANALYSIS;

EID: 0033638153     PISSN: 00071188     EISSN: None     Source Type: Journal    
DOI: 10.1038/sj.bjp.0703726     Document Type: Article

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