α2-adrenoceptor agonists stimulate high-affinity GTPase activity in a receptor subtype-selective manner

European Journal of Pharmacology

Volumn 374, Issue 1, 1999, Pages 137-146

  Jansson, Christian C ^a   Pohjanoksa, Katariina ^a   Lang, Jaana ^b   Wurster, Siegfried ^b   Savola, Juha Matti ^b   Scheinin, Mika ^a  

^a UNIVERSITY OF TURKU   (Finland)

^b ORION CORPORATION   (Finland)

Author keywords

2 adrenoceptor subtype; cAMP; CHO (Chinese hamster ovary) cell; GTPase assay; HEL (human erythroleukemia) cell; NG108 15 cell; Subtype selectivity

Indexed keywords

ADRENALIN; ALPHA 2 ADRENERGIC RECEPTOR STIMULATING AGENT; ALPHA 2A ADRENERGIC RECEPTOR; ALPHA 2B ADRENERGIC RECEPTOR; ALPHA 2C ADRENERGIC RECEPTOR; BRIMONIDINE; DEXMEDETOMIDINE; GUANOSINE TRIPHOSPHATASE; GUANOSINE TRIPHOSPHATE; OXYMETAZOLINE; ALPHA 2 ADRENERGIC RECEPTOR; BORDETELLA VIRULENCE FACTOR; CYCLIC AMP; PERTUSSIS TOXIN;

ANIMAL CELL; ARTICLE; CHO CELL; ENZYME ACTIVATION; GENETIC TRANSFECTION; NONHUMAN; PRIORITY JOURNAL; ANIMAL; BIOSYNTHESIS; CELL MEMBRANE; CLASSIFICATION; DRUG POTENTIATION; ENZYMOLOGY; HAMSTER; HUMAN; HYDROLYSIS; METABOLISM;

ANIMALS; CELL MEMBRANE; CHO CELLS; CRICETINAE; CYCLIC AMP; EPINEPHRINE; GTP PHOSPHOHYDROLASES; GUANOSINE TRIPHOSPHATE; HUMANS; HYDROLYSIS; PERTUSSIS TOXIN; RECEPTORS, ADRENERGIC, ALPHA-2; VIRULENCE FACTORS, BORDETELLA;

EID: 0032589056     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(99)00306-4     Document Type: Article

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