Binding of [3H](2S,1'S,2'S)-2-(9-xanthylmethyl)-2-(2'-carboxycyclopropyl) glycine ([3H]LY341495) to cell membranes expressing recombinant human group III metabotropic glutamate receptor subtypes

Naunyn-Schmiedeberg's Archives of Pharmacology

Volumn 362, Issue 6, 2000, Pages 546-554

  Wright, R A ^a   Arnold, M B ^a   Wheeler, W J ^a   Ornstein, P L ^a   Schoepp, D D ^a  

^a ELI LILLY AND COMPANY   (United States)

Author keywords

Group III mGlu receptors; LY341495; Metabotropic glutamate receptors; Radioligand; Receptor binding

Indexed keywords

2 AMINO 2 (2 CARBOXYCYCLOPROPYL) 3 (XANTHEN 9 YL)PROPIONIC ACID; METABOTROPIC RECEPTOR; RECEPTOR SUBTYPE; AMINO ACID; AMINO ACID RECEPTOR BLOCKING AGENT; METABOTROPIC RECEPTOR 4; METABOTROPIC RECEPTOR 6; METABOTROPIC RECEPTOR 7; METABOTROPIC RECEPTOR 8; RECOMBINANT PROTEIN; TRITIUM; XANTHENE DERIVATIVE;

ARTICLE; BINDING AFFINITY; COMPETITIVE INHIBITION; ENZYME ACTIVITY; HUMAN; HUMAN CELL; LIGAND BINDING; MEMBRANE BINDING; NEUROTRANSMITTER RELEASE; PROTEIN PROTEIN INTERACTION; RECEPTOR BINDING; SECOND MESSENGER; SEQUENCE HOMOLOGY; SYNAPTIC TRANSMISSION; BINDING COMPETITION; BIOSYNTHESIS; CELL MEMBRANE; CLASSIFICATION; ENZYME SPECIFICITY; GENETICS; KINETICS; METABOLISM; RADIOASSAY;

AMINO ACIDS; BINDING, COMPETITIVE; CELL MEMBRANE; EXCITATORY AMINO ACID ANTAGONISTS; HUMANS; KINETICS; RADIOLIGAND ASSAY; RECEPTORS, METABOTROPIC GLUTAMATE; RECOMBINANT PROTEINS; SUBSTRATE SPECIFICITY; TRITIUM; XANTHENES;

EID: 0033625834     PISSN: 00281298     EISSN: None     Source Type: Journal    
DOI: 10.1007/s002100000305     Document Type: Article

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