[3H]ac-RYYRWK-NH2, a novel specific radioligand for the nociceptin/orphanin FQ receptor

Naunyn-Schmiedeberg's Archives of Pharmacology

Volumn 362, Issue 6, 2000, Pages 538-545

  Thomsen, C ^a   Valsborg, J S ^a   Platou, J ^a   Martin, J ^a   Foged, C ^a   Johansen, N L ^a   Olsen, U B ^a   Madsen, K ^a  

^a H LUNDBECK A S   (Denmark)

Author keywords

Autoradiography; Hexapeptide radioligand; Nociceptin receptor; ORL1; Orphanin FQ; Receptor binding

Indexed keywords

CAM 6369; NOCICEPTIN RECEPTOR; OLIGOPEPTIDE; OPIATE PEPTIDE; OPIATE RECEPTOR; TRITIUM; DYNORPHIN A; HEXAPEPTIDE; NOCICEPTIN;

AMYGDALOID NUCLEUS; ANIMAL; ARTICLE; AUTORADIOGRAPHY; BINDING COMPETITION; BINDING SITE; BRAIN CORTEX; CELL MEMBRANE; DRUG POTENTIATION; ENZYME SPECIFICITY; FEMALE; HAMSTER; HUMAN; HYPOTHALAMUS; KINETICS; METABOLISM; RADIOASSAY; RAT; SPRAGUE DAWLEY RAT; ANIMAL CELL; BRAIN MEMBRANE; COMPETITIVE INHIBITION; ENZYME ACTIVITY; LIGAND BINDING; NONHUMAN; PROTEIN DOMAIN; PROTEIN FAMILY; RECEPTOR AFFINITY; RECEPTOR BINDING; STRUCTURE ACTIVITY RELATION;

AMYGDALA; ANIMALS; AUTORADIOGRAPHY; BINDING SITES; BINDING, COMPETITIVE; CELL MEMBRANE; CEREBRAL CORTEX; CRICETINAE; FEMALE; HUMANS; HYPOTHALAMUS; KINETICS; OLIGOPEPTIDES; OPIOID PEPTIDES; RADIOLIGAND ASSAY; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, OPIOID; SUBSTRATE SPECIFICITY; TRITIUM;

EID: 0033625833     PISSN: 00281298     EISSN: None     Source Type: Journal    
DOI: 10.1007/s002100000307     Document Type: Article

References (21)

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