A potent and highly selective nonpeptidyl nociceptin/orphanin FQ receptor (ORL1) antagonist: J-113397

European Journal of Pharmacology

Volumn 387, Issue 3, 2000, Pages R17-R18

  Ozaki, Satoshi ^a   Kawamoto, Hiroshi ^a   Itoh, Yoshiki ^a   Miyaji, Mitsuru ^a   Iwasawa, Yoshikazu ^a   Ohta, Hisashi ^a  

^a TAIHO PHARMACEUTICAL CO LTD   (Japan)

Author keywords

Nociceptin orphanin FQ; Opioid; ORL1 receptor

Indexed keywords

1 (1 CYCLOOCTYLMETHYL 3 HYDROXYMETHYL 4 PIPERIDYL) 3 ETHYL 1,3 DIHYDRO 2H BENZIMIDAZOL 2 ONE; DELTA OPIATE RECEPTOR; FORSKOLIN; KAPPA OPIATE RECEPTOR; MU OPIATE RECEPTOR; NOCICEPTIN; NOCICEPTIN RECEPTOR; OPIATE ANTAGONIST; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CHO CELL; DOSE RESPONSE; DRUG INHIBITION; DRUG RECEPTOR BINDING; DRUG STRUCTURE; NOCICEPTION; NONHUMAN; PRIORITY JOURNAL; RECEPTOR AFFINITY;

ANIMALS; BENZIMIDAZOLES; CHO CELLS; CRICETINAE; CYCLIC AMP; DOSE-RESPONSE RELATIONSHIP, DRUG; FORSKOLIN; PIPERIDINES; RECEPTORS, OPIOID;

EID: 0033969588     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-2999(99)00822-5     Document Type: Article

References (7)

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