-
1
-
-
79960245915
-
Cross-coupling reactions of organoboranes: An easy way to construct C-C bonds (Nobel Lecture)
-
pmid: 21618370
-
A. Suzuki, Cross-coupling reactions of organoboranes: An easy way to construct C-C bonds (Nobel Lecture). Angew. Chem. Int. Ed. 50, 6722-6737 (2011). doi: 10.1002/ anie.201101379; pmid: 21618370
-
(2011)
Angew. Chem. Int. Ed.
, vol.50
, pp. 6722-6737
-
-
Suzuki, A.1
-
2
-
-
84958231622
-
Synthesis and applications of boronic acid-containing polymers: From materials to medicine
-
pmid: 26367140
-
W. L. A. Brooks, B. S. Sumerlin, Synthesis and applications of boronic acid-containing polymers: From materials to medicine. Chem. Rev. 116, 1375-1397 (2016). doi: 10.1021/acs.chemrev.5b00300; pmid: 26367140
-
(2016)
Chem. Rev.
, vol.116
, pp. 1375-1397
-
-
Brooks, W.L.A.1
Sumerlin, B.S.2
-
3
-
-
84874051877
-
Exploiting the reversible covalent bonding of boronic acids: Recognition, sensing, and assembly
-
pmid: 23148559
-
S. D. Bull et al., Exploiting the reversible covalent bonding of boronic acids: Recognition, sensing, and assembly. Acc. Chem. Res. 46, 312-326 (2013). doi: 10.1021/ar300130w; pmid: 23148559
-
(2013)
Acc. Chem. Res.
, vol.46
, pp. 312-326
-
-
Bull, S.D.1
-
4
-
-
79952191452
-
Boronic acids in medicinal chemistry: Anticancer, antibacterial and antiviral applications
-
P. C. Trippier, C. McGuigan, Boronic acids in medicinal chemistry: Anticancer, antibacterial and antiviral applications. MedChemComm 1, 183 (2010). doi: 10.1039/ c0md00119h
-
(2010)
MedChemComm
, vol.1
, pp. 183
-
-
Trippier, P.C.1
McGuigan, C.2
-
5
-
-
85051780817
-
The future of boron in medicinal chemistry: Therapeutic and diagnostic applications
-
J. Schwarz, Ed. (Springer)
-
A. Draganov, D. Wang, B. Wang, The future of boron in medicinal chemistry: Therapeutic and diagnostic applications. In Atypical Elements in Drug Design, J. Schwarz, Ed. (Springer, 2014), pp. 1-27. doi: 10.1007/7355-2014-65
-
(2014)
Atypical Elements in Drug Design
, pp. 1-27
-
-
Draganov, A.1
Wang, D.2
Wang, B.3
-
6
-
-
84874353612
-
Carboxylic acid (bio) isosteres in drug design
-
pmid: 23361977
-
C. Ballatore, D. M. Huryn, A. B. Smith 3rd, Carboxylic acid (bio) isosteres in drug design. ChemMedChem 8, 385-395 (2013). doi: 10.1002/cmdc.201200585; pmid: 23361977
-
(2013)
ChemMedChem
, vol.8
, pp. 385-395
-
-
Ballatore, C.1
Huryn, D.M.2
Smith, A.B.3
-
7
-
-
84865088209
-
Boron containing compounds as protease inhibitors
-
pmid: 22519511
-
R. Smoum, A. Rubinstein, V. M. Dembitsky, M. Srebnik, Boron containing compounds as protease inhibitors. Chem. Rev. 112, 4156-4220 (2012). doi: 10.1021/cr608202m; pmid: 22519511
-
(2012)
Chem. Rev.
, vol.112
, pp. 4156-4220
-
-
Smoum, R.1
Rubinstein, A.2
Dembitsky, V.M.3
Srebnik, M.4
-
9
-
-
17644381216
-
Recent advances in organic synthesis using transition metal-catalyzed hydroborations
-
C. M. Vogels, S. A. Westcott, Recent advances in organic synthesis using transition metal-catalyzed hydroborations. Curr. Org. Chem. 9, 687-699 (2005). doi: 10.2174/ 1385272053765060
-
(2005)
Curr. Org. Chem.
, vol.9
, pp. 687-699
-
-
Vogels, C.M.1
Westcott, S.A.2
-
10
-
-
84863469858
-
Nickel-catalyzed coupling reactions of alkyl electrophiles, including unactivated tertiary halides, to generate carbon-boron bonds
-
pmid: 22668072
-
A. S. Dudnik, G. C. Fu, Nickel-catalyzed coupling reactions of alkyl electrophiles, including unactivated tertiary halides, to generate carbon-boron bonds. J. Am. Chem. Soc. 134, 10693-10697 (2012). doi: 10.1021/ja304068t; pmid: 22668072
-
(2012)
J. Am. Chem. Soc.
, vol.134
, pp. 10693-10697
-
-
Dudnik, A.S.1
Fu, G.C.2
-
11
-
-
84903977425
-
Iron-catalyzed borylation of alkyl electrophiles
-
pmid: 24955892
-
T. C. Atack, R. M. Lecker, S. P. Cook, Iron-catalyzed borylation of alkyl electrophiles. J. Am. Chem. Soc. 136, 9521-9523 (2014). doi: 10.1021/ja505199u; pmid: 24955892
-
(2014)
J. Am. Chem. Soc.
, vol.136
, pp. 9521-9523
-
-
Atack, T.C.1
Lecker, R.M.2
Cook, S.P.3
-
12
-
-
84910003839
-
Iron-catalyzed borylation of alkyl, allyl, and aryl halides: Isolation of an iron(I) boryl complex
-
R. B. Bedford et al., Iron-catalyzed borylation of alkyl, allyl, and aryl halides: Isolation of an iron(I) boryl complex. Organometallics 33, 5940-5943 (2014). doi: 10.1021/ om500847j
-
(2014)
Organometallics
, vol.33
, pp. 5940-5943
-
-
Bedford, R.B.1
-
13
-
-
84855464257
-
Alkylboronic esters from copper-catalyzed borylation of primary and secondary alkyl halides and pseudohalides
-
pmid: 22135233
-
C.-T. Yang et al., Alkylboronic esters from copper-catalyzed borylation of primary and secondary alkyl halides and pseudohalides. Angew. Chem. Int. Ed. 51, 528-532 (2012). doi: 10.1002/anie.201106299; pmid: 22135233
-
(2012)
Angew. Chem. Int. Ed.
, vol.51
, pp. 528-532
-
-
Yang, C.-T.1
-
14
-
-
84856693018
-
Copper(I)-catalyzed boryl substitution of unactivated alkyl halides
-
pmid: 22260229
-
H. Ito, K. Kubota, Copper(I)-catalyzed boryl substitution of unactivated alkyl halides. Org. Lett. 14, 890-893 (2012). doi: 10.1021/ol203413w; pmid: 22260229
-
(2012)
Org. Lett.
, vol.14
, pp. 890-893
-
-
Ito, H.1
Kubota, K.2
-
16
-
-
0001307257
-
A simple preparation of boronic esters from organolithium reagents and selected trialkoxyboranes
-
A simple preparation of boronic esters from organolithium reagents and selected trialkoxyboranes. Organometallics 2, 1316-1319 (1983). doi: 10.1021/om50004a009
-
(1983)
Organometallics
, vol.2
, pp. 1316-1319
-
-
-
17
-
-
67650566923
-
Efficient C-B bond formation promoted by N-heterocyclic carbenes: Synthesis of tertiary and quaternary B-substituted carbons through metal-free catalytic boron conjugate additions to cyclic and acyclic a,b-unsaturated carbonyls
-
pmid: 19432440
-
K. S. Lee, A. R. Zhugralin, A. H. Hoveyda, Efficient C-B bond formation promoted by N-heterocyclic carbenes: Synthesis of tertiary and quaternary B-substituted carbons through metal-free catalytic boron conjugate additions to cyclic and acyclic a,b-unsaturated carbonyls. J. Am. Chem. Soc. 131, 7253-7255 (2009). doi: 10.1021/ja902889s; pmid: 19432440
-
(2009)
J. Am. Chem. Soc.
, vol.131
, pp. 7253-7255
-
-
Lee, K.S.1
Zhugralin, A.R.2
Hoveyda, A.H.3
-
18
-
-
76349094490
-
Enantioselective conjugate borylation
-
pmid: 20077553
-
J. A. Schiffner, K. M?ther, M. Oestreich, Enantioselective conjugate borylation. Angew. Chem. Int. Ed. 49, 1194-1196 (2010). doi: 10.1002/anie.200906521; pmid: 20077553
-
(2010)
Angew. Chem. Int. Ed.
, vol.49
, pp. 1194-1196
-
-
Schiffner, J.A.1
Mther, K.2
Oestreich, M.3
-
19
-
-
84967262800
-
Synthesis of a-aminoboronic acids
-
pmid: 26853637
-
P. Andrés, G. Ballano, M. I. Calaza, C. Cativiela, Synthesis of a-aminoboronic acids. Chem. Soc. Rev. 45, 2291-2307 (2016). doi: 10.1039/C5CS00886G; pmid: 26853637
-
(2016)
Chem. Soc. Rev.
, vol.45
, pp. 2291-2307
-
-
Andrés, P.1
Ballano, G.2
Calaza, M.I.3
Cativiela, C.4
-
20
-
-
44449138158
-
Asymmetric coppercatalyzed synthesis of a-amino boronate esters from N-tertbutanesulfinyl aldimines
-
pmid: 18461938
-
M. A. Beenen, C. An, J. A. Ellman, Asymmetric coppercatalyzed synthesis of a-amino boronate esters from N-tertbutanesulfinyl aldimines. J. Am. Chem. Soc. 130, 6910-6911 (2008). doi: 10.1021/ja800829y; pmid: 18461938
-
(2008)
J. Am. Chem. Soc.
, vol.130
, pp. 6910-6911
-
-
Beenen, M.A.1
An, C.2
Ellman, J.A.3
-
21
-
-
77349125577
-
C-H activation for the construction of C-B bonds
-
pmid: 20028025
-
I. A. Mkhalid, J. H. Barnard, T. B. Marder, J. M. Murphy, J. F. Hartwig, C-H activation for the construction of C-B bonds. Chem. Rev. 110, 890-931 (2010). doi: 10.1021/cr900206p; pmid: 20028025
-
(2010)
Chem. Rev.
, vol.110
, pp. 890-931
-
-
Mkhalid, I.A.1
Barnard, J.H.2
Marder, T.B.3
Murphy, J.M.4
Hartwig, J.F.5
-
23
-
-
84964558188
-
A general alkyl-alkyl cross-coupling enabled by redox-active esters and alkylzinc reagents
-
pmid: 27103669
-
T. Qin et al., A general alkyl-alkyl cross-coupling enabled by redox-active esters and alkylzinc reagents. Science 352, 801-805 (2016). doi: 10.1126/science.aaf6123; pmid: 27103669
-
(2016)
Science
, vol.352
, pp. 801-805
-
-
Qin, T.1
-
24
-
-
84959450281
-
Practical Ni-catalyzed aryl-alkyl cross-coupling of secondary redox-active esters
-
pmid: 26835704
-
J. Cornella et al., Practical Ni-catalyzed aryl-alkyl cross-coupling of secondary redox-active esters. J. Am. Chem. Soc. 138, 2174-2177 (2016). doi: 10.1021/jacs.6b00250; pmid: 26835704
-
(2016)
J. Am. Chem. Soc.
, vol.138
, pp. 2174-2177
-
-
Cornella, J.1
-
25
-
-
84979074178
-
Nickel-catalyzed cross-coupling of redox-active esters with boronic acids
-
pmid: 27380912
-
J. Wang et al., Nickel-catalyzed cross-coupling of redox-active esters with boronic acids. Angew. Chem. Int. Ed. 55, 9676-9679 (2016). doi: 10.1002/anie.201605463; pmid: 27380912
-
(2016)
Angew. Chem. Int. Ed.
, vol.55
, pp. 9676-9679
-
-
Wang, J.1
-
26
-
-
84986230272
-
Redox-active esters in Fe-catalyzed C-C coupling
-
pmid: 27548696
-
F. Toriyama et al., Redox-active esters in Fe-catalyzed C-C coupling. J. Am. Chem. Soc. 138, 11132-11135 (2016). doi: 10.1021/jacs.6b07172; pmid: 27548696
-
(2016)
J. Am. Chem. Soc.
, vol.138
, pp. 11132-11135
-
-
Toriyama, F.1
-
27
-
-
85007124060
-
Nickel-catalyzed barton decarboxylation and Giese reactions: A practical take on classic transforms
-
pmid: 27981703
-
T. Qin et al., Nickel-catalyzed barton decarboxylation and Giese reactions: A practical take on classic transforms. Angew. Chem. Int. Ed. 56, 260-265 (2017). doi: 10.1002/ anie.201609662; pmid: 27981703
-
(2017)
Angew. Chem. Int. Ed.
, vol.56
, pp. 260-265
-
-
Qin, T.1
-
28
-
-
77955379578
-
Iron-catalyzed Suzuki-Miyaura coupling of alkyl halides
-
pmid: 20681696
-
T. Hatakeyama et al., Iron-catalyzed Suzuki-Miyaura coupling of alkyl halides. J. Am. Chem. Soc. 132, 10674-10676 (2010). doi: 10.1021/ja103973a; pmid: 20681696
-
(2010)
J. Am. Chem. Soc.
, vol.132
, pp. 10674-10676
-
-
Hatakeyama, T.1
-
29
-
-
84903176970
-
Expedient iron-catalyzed coupling of alkyl, benzyl and allyl halides with arylboronic esters
-
pmid: 24715587
-
R. B. Bedford et al., Expedient iron-catalyzed coupling of alkyl, benzyl and allyl halides with arylboronic esters. Chemistry 20, 7935-7938 (2014). doi: 10.1002/chem.201402174; pmid: 24715587
-
(2014)
Chemistry
, vol.20
, pp. 7935-7938
-
-
Bedford, R.B.1
-
30
-
-
79957759309
-
Design, synthesis, radiolabeling, and in vitro and in vivo evaluation of bridgehead iodinated analogues of N-2-[4-(2-methoxyphenyl)piperazin-1-yl]ethyl-N-(pyridin-2-yl)cyclohexanecarboxamide (WAY-100635) as potential SPECT ligands for the 5-HT1A receptor
-
pmid: 21520940
-
R. Al Hussainy et al., Design, synthesis, radiolabeling, and in vitro and in vivo evaluation of bridgehead iodinated analogues of N-2-[4-(2-methoxyphenyl)piperazin-1-yl]ethyl-N-(pyridin-2-yl)cyclohexanecarboxamide (WAY-100635) as potential SPECT ligands for the 5-HT1A receptor. J. Med. Chem. 54, 3480-3491 (2011). doi: 10.1021/jm1009956; pmid: 21520940
-
(2011)
J. Med. Chem.
, vol.54
, pp. 3480-3491
-
-
Al Hussainy, R.1
-
31
-
-
84966333678
-
Structure property relationships of carboxylic acid isosteres
-
pmid: 26967507
-
P. Lassalas et al., Structure property relationships of carboxylic acid isosteres. J. Med. Chem. 59, 3183-3203 (2016). doi: 10.1021/acs.jmedchem.5b01963; pmid: 26967507
-
(2016)
J. Med. Chem.
, vol.59
, pp. 3183-3203
-
-
Lassalas, P.1
-
32
-
-
85003022498
-
A general, modular method for the catalytic asymmetric synthesis of alkylboronate esters
-
pmid: 27940868
-
J. Schmidt, J. Choi, A. T. Liu, M. Slusarczyk, G. C. Fu, A general, modular method for the catalytic asymmetric synthesis of alkylboronate esters. Science 354, 1265-1269 (2016). doi: 10.1126/science.aai8611; pmid: 27940868
-
(2016)
Science
, vol.354
, pp. 1265-1269
-
-
Schmidt, J.1
Choi, J.2
Liu, A.T.3
Slusarczyk, M.4
Fu, G.C.5
-
33
-
-
84973380029
-
Diverse asymmetric hydrofunctionalization of aliphatic internal alkenes through catalytic regioselective hydroboration
-
Y. Xi, J. F. Hartwig, Diverse asymmetric hydrofunctionalization of aliphatic internal alkenes through catalytic regioselective hydroboration. J. Am. Chem. Soc. 138, 6703-6706 (2016). doi: 10.1021/jacs.6b02478;pmid: 27167490
-
(2016)
J. Am. Chem. Soc.
, vol.138
, pp. 6703-6706
-
-
Xi, Y.1
Hartwig, J.F.2
-
34
-
-
34248385279
-
Organotrifluoroborates: Protected boronic acids that expand the versatility of the Suzuki coupling reaction
-
pmid: 17256882
-
G. A. Molander, N. Ellis, Organotrifluoroborates: Protected boronic acids that expand the versatility of the Suzuki coupling reaction. Acc. Chem. Res. 40, 275-286 (2007). doi: 10.1021/ ar050199q; pmid: 17256882
-
(2007)
Acc. Chem. Res.
, vol.40
, pp. 275-286
-
-
Molander, G.A.1
Ellis, N.2
-
35
-
-
84867338504
-
Direct stereospecific amination of alkyl and aryl pinacol boronates
-
pmid: 23002712
-
S. N. Mlynarski, A. S. Karns, J. P. Morken, Direct stereospecific amination of alkyl and aryl pinacol boronates. J. Am. Chem. Soc. 134, 16449-16451 (2012). doi: 10.1021/ja305448w; pmid: 23002712
-
(2012)
J. Am. Chem. Soc.
, vol.134
, pp. 16449-16451
-
-
Mlynarski, S.N.1
Karns, A.S.2
Morken, J.P.3
-
36
-
-
84903219214
-
Enantiospecific sp2-sp3 coupling of secondary and tertiary boronic esters
-
pmid: 24950327
-
A. Bonet, M. Odachowski, D. Leonori, S. Essafi, V. K. Aggarwal, Enantiospecific sp2-sp3 coupling of secondary and tertiary boronic esters. Nat. Chem. 6, 584-589 (2014). doi: 10.1038/ nchem.1971; pmid: 24950327
-
(2014)
Nat. Chem.
, vol.6
, pp. 584-589
-
-
Bonet, A.1
Odachowski, M.2
Leonori, D.3
Essafi, S.4
Aggarwal, V.K.5
-
37
-
-
84984865364
-
Selective and serial Suzuki-Miyaura reactions of polychlorinated aromatics with alkyl pinacol boronic esters
-
pmid: 27537216
-
S. Laulhé, J. M. Blackburn, J. L. Roizen, Selective and serial Suzuki-Miyaura reactions of polychlorinated aromatics with alkyl pinacol boronic esters. Org. Lett. 18, 4440-4443 (2016). doi: 10.1021/acs.orglett.6b02323; pmid: 27537216
-
(2016)
Org. Lett.
, vol.18
, pp. 4440-4443
-
-
Laulhé, S.1
Blackburn, J.M.2
Roizen, J.L.3
-
38
-
-
0037467698
-
Synthesis and biological activity of a-aminoboronic acids, amine-carboxyboranes and their derivatives
-
V. M. Dembitsky, M. Srebnik, Synthesis and biological activity of a-aminoboronic acids, amine-carboxyboranes and their derivatives. Tetrahedron 59, 579-593 (2003). doi: 10.1016/ S0040-4020(02)01618-6
-
(2003)
Tetrahedron
, vol.59
, pp. 579-593
-
-
Dembitsky, V.M.1
Srebnik, M.2
-
39
-
-
0037029807
-
Synthesis and evaluation of vancomycin and vancomycin aglycon analogues that bear modifications in the residue 3 asparagine
-
pmid: 11965380
-
J. J. McAtee, S. L. Castle, Q. Jin, D. L. Boger, Synthesis and evaluation of vancomycin and vancomycin aglycon analogues that bear modifications in the residue 3 asparagine. Bioorg. Med. Chem. Lett. 12, 1319-1322 (2002). doi: 10.1016/S0960-894X(02)00130-0; pmid: 11965380
-
(2002)
Bioorg. Med. Chem. Lett.
, vol.12
, pp. 1319-1322
-
-
McAtee, J.J.1
Castle, S.L.2
Jin, Q.3
Boger, D.L.4
-
40
-
-
0028245052
-
Design of orally active, non-peptidic inhibitors of human leukocyte elastase
-
pmid: 8176703
-
F. J. Brown et al., Design of orally active, non-peptidic inhibitors of human leukocyte elastase. J. Med. Chem. 37, 1259-1261 (1994). doi: 10.1021/jm00035a004; pmid: 8176703
-
(1994)
J. Med. Chem.
, vol.37
, pp. 1259-1261
-
-
Brown, F.J.1
-
41
-
-
9844256449
-
Orally active trifluoromethyl ketone inhibitors of human leukocyte elastase
-
pmid: 9379436
-
C. A. Veale et al., Orally active trifluoromethyl ketone inhibitors of human leukocyte elastase. J. Med. Chem. 40, 3173-3181 (1997). doi: 10.1021/jm970250z; pmid: 9379436
-
(1997)
J. Med. Chem.
, vol.40
, pp. 3173-3181
-
-
Veale, C.A.1
-
42
-
-
0028998059
-
Nonpeptidic inhibitors of human leukocyte elastase. 6. Design of a potent, intratracheally active, pyridone-based trifluoromethyl ketone
-
pmid: 7837235
-
P. R. Bernstein, B. C. Gomes, B. J. Kosmider, E. P. Vacek, J. C. Williams, Nonpeptidic inhibitors of human leukocyte elastase. 6. Design of a potent, intratracheally active, pyridone-based trifluoromethyl ketone. J. Med. Chem. 38, 212-215 (1995). doi: 10.1021/jm00001a028; pmid: 7837235
-
(1995)
J. Med. Chem.
, vol.38
, pp. 212-215
-
-
Bernstein, P.R.1
Gomes, B.C.2
Kosmider, B.J.3
Vacek, E.P.4
Williams, J.C.5
-
43
-
-
0029043448
-
Inhibition of human neutrophil elastase. 3. An orally active enol acetate prodrug
-
pmid: 7830264
-
J. P. Burkhart et al., Inhibition of human neutrophil elastase. 3. An orally active enol acetate prodrug. J. Med. Chem. 38, 223-233 (1995). doi: 10.1021/jm00002a003; pmid: 7830264
-
(1995)
J. Med. Chem.
, vol.38
, pp. 223-233
-
-
Burkhart, J.P.1
-
44
-
-
15144355533
-
Discovery and biological activity of orally active peptidyl trifluoromethyl ketone inhibitors of human neutrophil elastase
-
pmid: 9191965
-
P. D. Edwards et al., Discovery and biological activity of orally active peptidyl trifluoromethyl ketone inhibitors of human neutrophil elastase. J. Med. Chem. 40, 1876-1885 (1997). doi: 10.1021/jm960819g; pmid: 9191965
-
(1997)
J. Med. Chem.
, vol.40
, pp. 1876-1885
-
-
Edwards, P.D.1
-
46
-
-
0037421010
-
True interaction mode of porcine pancreatic elastase with FR136706, a potent peptidyl inhibitor
-
pmid: 12467609
-
T. Kinoshita, I. Nakanishi, A. Sato, T. Tada, True interaction mode of porcine pancreatic elastase with FR136706, a potent peptidyl inhibitor. Bioorg. Med. Chem. Lett. 13, 21-24 (2003). doi: 10.1016/S0960-894X(02)00852-1; pmid: 12467609
-
(2003)
Bioorg. Med. Chem. Lett.
, vol.13
, pp. 21-24
-
-
Kinoshita, T.1
Nakanishi, I.2
Sato, A.3
Tada, T.4
-
47
-
-
84942837686
-
Neutrophil elastase inhibitors for the treatment of (cardio)pulmonary diseases: Into clinical testing with pre-adaptive pharmacophores
-
pmid: 26358162
-
F. von Nussbaum, V. M.-J. Li, Neutrophil elastase inhibitors for the treatment of (cardio)pulmonary diseases: Into clinical testing with pre-adaptive pharmacophores. Bioorg. Med. Chem. Lett. 25, 4370-4381 (2015). doi: 10.1016/j.bmcl.2015.08.049; pmid: 26358162
-
(2015)
Bioorg. Med. Chem. Lett.
, vol.25
, pp. 4370-4381
-
-
Von Nussbaum, F.1
Li, V.M.-J.2
-
48
-
-
84933525796
-
Freezing the bioactive conformation to boost potency: The identification of BAY 85-8501, a selective and potent inhibitor of human neutrophil elastase for pulmonary diseases
-
pmid: 26083237
-
F. von Nussbaum et al., Freezing the bioactive conformation to boost potency: The identification of BAY 85-8501, a selective and potent inhibitor of human neutrophil elastase for pulmonary diseases. ChemMedChem 10, 1163-1173 (2015). doi: 10.1002/cmdc.201500131; pmid: 26083237
-
(2015)
ChemMedChem
, vol.10
, pp. 1163-1173
-
-
Von Nussbaum, F.1
-
49
-
-
85020556278
-
-
F. O. Gombert et al., patent application WO2015096873 (2015).
-
(2015)
-
-
Gombert, F.O.1
-
50
-
-
85020589773
-
-
patent application WO2013037809
-
T. J. Blench et al., patent application WO2013037809 (2013).
-
(2013)
-
-
Blench, T.J.1
-
52
-
-
84885190072
-
The thermodynamic basis for the use of lipophilic efficiency (LipE) in enthalpic optimizations
-
pmid: 24054120
-
M. D. Shultz, The thermodynamic basis for the use of lipophilic efficiency (LipE) in enthalpic optimizations. Bioorg. Med. Chem. Lett. 23, 5992-6000 (2013). doi: 10.1016/j.bmcl.2013.08.030; pmid: 24054120
-
(2013)
Bioorg. Med. Chem. Lett.
, vol.23
, pp. 5992-6000
-
-
Shultz, M.D.1
-
53
-
-
79960260060
-
Unexpected tricovalent binding mode of boronic acids within the active site of a penicillin-binding protein
-
pmid: 21574608
-
A. Zervosen et al., Unexpected tricovalent binding mode of boronic acids within the active site of a penicillin-binding protein. J. Am. Chem. Soc. 133, 10839-10848 (2011). doi: 10.1021/ja200696y; pmid: 21574608
-
(2011)
J. Am. Chem. Soc.
, vol.133
, pp. 10839-10848
-
-
Zervosen, A.1
-
54
-
-
33644845743
-
Crystal structure of the boronic acid-based proteasome inhibitor bortezomib in complex with the yeast 20S proteasome
-
pmid: 16531229
-
M. Groll, C. R. Berkers, H. L. Ploegh, H. Ovaa, Crystal structure of the boronic acid-based proteasome inhibitor bortezomib in complex with the yeast 20S proteasome. Structure 14, 451-456 (2006). doi: 10.1016/j.str.2005.11.019; pmid: 16531229
-
(2006)
Structure
, vol.14
, pp. 451-456
-
-
Groll, M.1
Berkers, C.R.2
Ploegh, H.L.3
Ovaa, H.4
-
55
-
-
84856373151
-
Proteasome inhibitors: An expanding army attacking a unique target
-
pmid: 22284358
-
A. F. Kisselev, W. A. van der Linden, H. S. Overkleeft, Proteasome inhibitors: An expanding army attacking a unique target. Chem. Biol. 19, 99-115 (2012). doi: 10.1016/ j.chembiol.2012.01.003; pmid: 22284358
-
(2012)
Chem. Biol.
, vol.19
, pp. 99-115
-
-
Kisselev, A.F.1
Linden Der Van, W.A.2
Overkleeft, H.S.3
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