-
2
-
-
45849092587
-
Preparation, characterization and in vitro evaluation of solid dispersions containing docetaxel
-
Chen J, Qiu L, Hu M, et al. Preparation, characterization and in vitro evaluation of solid dispersions containing docetaxel. Drug Dev Ind Pharm 2008;34:588-94.
-
(2008)
Drug Dev Ind Pharm
, vol.34
, pp. 588-594
-
-
Chen, J.1
Qiu, L.2
Hu, M.3
-
3
-
-
80054697562
-
Pharmaceutical development and preliminary clinical testing of an oral solid dispersion formulation of docetaxel (ModraDoc001)
-
Moes JJ, Koolen SL, Huitema AD, et al. Pharmaceutical development and preliminary clinical testing of an oral solid dispersion formulation of docetaxel (ModraDoc001). Int J Pharm 2011;420: 244-50.
-
(2011)
Int J Pharm
, vol.420
, pp. 244-250
-
-
Moes, J.J.1
Koolen, S.L.2
Huitema, A.D.3
-
4
-
-
11244321887
-
Oral bioavailability of docetaxel in combination with OC144-093 (ONT-093)
-
Kuppens IE, Bosch TM, van Maanen MJ, et al. Oral bioavailability of docetaxel in combination with OC144-093 (ONT-093). Cancer Chemother Pharmacol 2005;55:72-8.
-
(2005)
Cancer Chemother Pharmacol
, vol.55
, pp. 72-78
-
-
Kuppens, I.E.1
Bosch, T.M.2
Van Maanen, M.J.3
-
5
-
-
54349088541
-
Preparation and characterization of a submicron lipid emulsion of docetaxel: Submicron lipid emulsion of docetaxel
-
Gao K, Sun J, Liu K, et al. Preparation and characterization of a submicron lipid emulsion of docetaxel: submicron lipid emulsion of docetaxel. Drug Dev Ind Pharm 2008;34:1227-37.
-
(2008)
Drug Dev Ind Pharm
, vol.34
, pp. 1227-1237
-
-
Gao, K.1
Sun, J.2
Liu, K.3
-
6
-
-
71549157438
-
Absence of both cytochrome P450 3A and P-glycoprotein dramatically increases docetaxel oral bioavailability and risk of intestinal toxicity
-
van Waterschoot RA, Lagas JS, Wagenaar E, et al. Absence of both cytochrome P450 3A and P-glycoprotein dramatically increases docetaxel oral bioavailability and risk of intestinal toxicity. Cancer Res 2009;69:8996-9002.
-
(2009)
Cancer Res
, vol.69
, pp. 8996-9002
-
-
Van Waterschoot, R.A.1
Lagas, J.S.2
Wagenaar, E.3
-
7
-
-
0036829187
-
Low systemic exposure of oral docetaxel in mice resulting from extensive first-pass metabolism is boosted by ritonavir
-
Bardelmeijer HA, Ouwehand M, Buckle T, et al. Low systemic exposure of oral docetaxel in mice resulting from extensive first-pass metabolism is boosted by ritonavir. Cancer Res 2002;62:6158-64
-
(2002)
Cancer Res
, vol.62
, pp. 6158-6164
-
-
Bardelmeijer, H.A.1
Ouwehand, M.2
Buckle, T.3
-
8
-
-
84983608244
-
-
FDA/CDER
-
Sanofi-Aventis. Taxotere (docetaxel) injection. FDA/CDER; 2011. Available from: http://www.accessdata.fda.gov/drugsatfda_docs/label/2014/020449s073lbl.pdf.
-
(2011)
Sanofi-Aventis. Taxotere (Docetaxel) Injection
-
-
-
9
-
-
77954805866
-
Solid dispersion as an approach for bioavailability enhancement of poorly water-soluble drug ritonavir
-
Sinha S, Ali M, Baboota S, et al. Solid dispersion as an approach for bioavailability enhancement of poorly water-soluble drug ritonavir. AAPS PharmSciTech 2010;11:518-27.
-
(2010)
AAPS Pharmscitech
, vol.11
, pp. 518-527
-
-
Sinha, S.1
Ali, M.2
Baboota, S.3
-
10
-
-
84896705229
-
Influence of different polymers on crystallization tendency and dissolution behavior of cilnidipine in solid dispersions
-
Chen C, Xie X, Li Y, et al. Influence of different polymers on crystallization tendency and dissolution behavior of cilnidipine in solid dispersions. Drug Dev Ind Pharm 2014;40:441-51.
-
(2014)
Drug Dev Ind Pharm
, vol.40
, pp. 441-451
-
-
Chen, C.1
Xie, X.2
Li, Y.3
-
11
-
-
0034868680
-
The potential of small-scale fusion experiments and the Gordon-Taylor equation to predict the suitability of drug/polymer blends for melt extrusion
-
Forster A, Hempenstall J, Tucker, I, et al. The potential of small-scale fusion experiments and the Gordon-Taylor equation to predict the suitability of drug/polymer blends for melt extrusion. Drug Dev Ind Pharm 2001;27:549-60.
-
(2001)
Drug Dev Ind Pharm
, vol.27
, pp. 549-560
-
-
Forster, A.1
Hempenstall, J.2
Tucker, I.3
-
12
-
-
84877077701
-
In vitro and in vivo evaluation of amorphous solid dispersions generated by different bench-scale processes, using griseofulvin as a model compound
-
Chiang PC, Cui Y, Ran Y, et al. In vitro and in vivo evaluation of amorphous solid dispersions generated by different bench-scale processes, using griseofulvin as a model compound. AAPS J 2013; 15:608-17.
-
(2013)
AAPS J
, vol.15
, pp. 608-617
-
-
Chiang, P.C.1
Cui, Y.2
Ran, Y.3
-
13
-
-
35348987129
-
Combined use of crystalline salt forms and precipitation inhibitors to improve oral absorption of celecoxib from solid oral formulations
-
Guzman HR, Tawa M, Zhang Z, et al. Combined use of crystalline salt forms and precipitation inhibitors to improve oral absorption of celecoxib from solid oral formulations. J Pharm Sci 2007;96: 2686-702.
-
(2007)
J Pharm Sci
, vol.96
, pp. 2686-2702
-
-
Guzman, H.R.1
Tawa, M.2
Zhang, Z.3
-
14
-
-
84930526016
-
Solubility and dissolution enhancement strategies: Current understanding and recent trends
-
Jain S, Patel N, Lin S. Solubility and dissolution enhancement strategies: current understanding and recent trends. Drug Dev Ind Pharm 2014. [Epub ahead of print]. DOI:10.3109/03639045.2014.971027.
-
(2014)
Drug Dev Ind Pharm
-
-
Jain, S.1
Patel, N.2
Lin, S.3
-
15
-
-
77951538902
-
Combining HME & solubilization: Soluplus - The solid solution
-
Hardung H, Djuric D, Ali S. Combining HME & solubilization: Soluplus - the solid solution. Drug Deliv Technol 2010;10:20-7.
-
(2010)
Drug Deliv Technol
, vol.10
, pp. 20-27
-
-
Hardung, H.1
Djuric, D.2
Ali, S.3
-
16
-
-
84875274738
-
Soluplus: A novel polymeric solubilizer for optimization of Carvedilol solid dispersions: Formulation design and effect of method of preparation
-
Shamma RN, Basha M. Soluplus: a novel polymeric solubilizer for optimization of Carvedilol solid dispersions: formulation design and effect of method of preparation. Powder Technol 2013;237:406-14.
-
(2013)
Powder Technol
, vol.237
, pp. 406-414
-
-
Shamma, R.N.1
Basha, M.2
-
17
-
-
84902239752
-
Data mining of solubility parameters for computational prediction of drug-excipient miscibility
-
Alhalaweh A, Alzghoul A, Kaialy W. Data mining of solubility parameters for computational prediction of drug-excipient miscibility. Drug Dev Ind Pharm 2014;40:904-9.
-
(2014)
Drug Dev Ind Pharm
, vol.40
, pp. 904-909
-
-
Alhalaweh, A.1
Alzghoul, A.2
Kaialy, W.3
-
18
-
-
0035845751
-
Selection of excipients for melt extrusion with two poorly water-soluble drugs by solubility parameter calculation and thermal analysis
-
Forster A, Hempenstall J, Tucker I, et al. Selection of excipients for melt extrusion with two poorly water-soluble drugs by solubility parameter calculation and thermal analysis. Int J Pharm 2001;226: 147-61.
-
(2001)
Int J Pharm
, vol.226
, pp. 147-161
-
-
Forster, A.1
Hempenstall, J.2
Tucker, I.3
-
19
-
-
84879009609
-
Prediction of drug-polymer miscibility through the use of solubility parameter-based Flory--uggins interaction parameter and the experimental validation: PEG as model polymer
-
Thakral S, Thakral NK. Prediction of drug-polymer miscibility through the use of solubility parameter-based Flory--uggins interaction parameter and the experimental validation: PEG as model polymer. J Pharm Sci 2013;102:2254-63.
-
(2013)
J Pharm Sci
, vol.102
, pp. 2254-2263
-
-
Thakral, S.1
Thakral, N.K.2
-
20
-
-
84875214001
-
Cyclodextrin-water soluble polymer ternary complexes enhance the solubility and dissolution behaviour of poorly soluble drugs. Case example: Itraconazole
-
Taupitz T, Dressman JB, Buchanan CM, et al. Cyclodextrin-water soluble polymer ternary complexes enhance the solubility and dissolution behaviour of poorly soluble drugs. Case example: itraconazole. Eur J Pharm Biopharm 2013;83:378-87.
-
(2013)
Eur J Pharm Biopharm
, vol.83
, pp. 378-387
-
-
Taupitz, T.1
Dressman, J.B.2
Buchanan, C.M.3
-
22
-
-
84916937130
-
Docetaxel epimerization in silicone films: A case of drug excipient incompatibility
-
Mohsin S, Arellano IH, Choudhury NR, et al. Docetaxel epimerization in silicone films: a case of drug excipient incompatibility. Drug Test Anal 2014;6:1076-84.
-
(2014)
Drug Test Anal
, vol.6
, pp. 1076-1084
-
-
Mohsin, S.1
Arellano, I.H.2
Choudhury, N.R.3
-
23
-
-
0034633805
-
Simple and sensitive high-performance liquid chromatography method for the determination of docetaxel in human plasma or urine
-
Garg MB, Ackland SP. Simple and sensitive high-performance liquid chromatography method for the determination of docetaxel in human plasma or urine. J Chromatogr B Biomed Sci Appl 2000;748: 383-8.
-
(2000)
J Chromatogr B Biomed Sci Appl
, vol.748
, pp. 383-388
-
-
Garg, M.B.1
Ackland, S.P.2
-
24
-
-
0032726595
-
Solubility parameters as predictors of miscibility in solid dispersions
-
Greenhalgh DJ, Williams AC, Timmins P, et al. Solubility parameters as predictors of miscibility in solid dispersions. J Pharm Sci 1999;88:1182-90.
-
(1999)
J Pharm Sci
, vol.88
, pp. 1182-1190
-
-
Greenhalgh, D.J.1
Williams, A.C.2
Timmins, P.3
-
26
-
-
38049173112
-
Predicting the solubility of the anti-cancer agent docetaxel in small molecule excipients using computational methods
-
Huynh L, Grant J, Leroux JC, et al. Predicting the solubility of the anti-cancer agent docetaxel in small molecule excipients using computational methods. Pharm Res 2008;25:147-57.
-
(2008)
Pharm Res
, vol.25
, pp. 147-157
-
-
Huynh, L.1
Grant, J.2
Leroux, J.C.3
-
27
-
-
80051793564
-
Bivalent sequential binding of docetaxel to methyl-beta-cyclodextrin
-
Mazzaferro S, Bouchemal K, Gallard JF, et al. Bivalent sequential binding of docetaxel to methyl-beta-cyclodextrin. Int J Pharm 2011; 416:171-80.
-
(2011)
Int J Pharm
, vol.416
, pp. 171-180
-
-
Mazzaferro, S.1
Bouchemal, K.2
Gallard, J.F.3
-
28
-
-
84878880994
-
Sulfobutylether-beta-cyclodextrin/chitosan nanoparticles enhance the oral permeability and bioavailability of docetaxel
-
Wu J, Shen Q, Fang L. Sulfobutylether-beta-cyclodextrin/chitosan nanoparticles enhance the oral permeability and bioavailability of docetaxel. Drug Dev Ind Pharm 2013;39:1010-9.
-
(2013)
Drug Dev Ind Pharm
, vol.39
, pp. 1010-1019
-
-
Wu, J.1
Shen, Q.2
Fang, L.3
-
29
-
-
33845714689
-
Alternative drug formulations of docetaxel: A review
-
Engels FK, Mathot RA, Verweij J. Alternative drug formulations of docetaxel: a review. Anticancer Drugs 2007;18:95-103.
-
(2007)
Anticancer Drugs
, vol.18
, pp. 95-103
-
-
Engels, F.K.1
Mathot, R.A.2
Verweij, J.3
-
30
-
-
0035710530
-
Docetaxel: Solid state characterization by X-ray powder diffraction and thermogravimetry
-
Pr10-221-Pr10-6
-
Zaske L, Perrin M-A, Leveiller F. Docetaxel: solid state characterization by X-ray powder diffraction and thermogravimetry. J Phys IV France 2001;11:Pr10-221-Pr10-6.
-
(2001)
J Phys IV France
, vol.11
-
-
Zaske, L.1
Perrin, M.-A.2
Leveiller, F.3
-
32
-
-
0030896467
-
The use of solubility parameters in pharmaceutical dosage form design
-
Hancock BC, York P, Rowe RC. The use of solubility parameters in pharmaceutical dosage form design. Int J Pharm 1997;148:1-21.
-
(1997)
Int J Pharm
, vol.148
, pp. 1-21
-
-
Hancock, B.C.1
York, P.2
Rowe, R.C.3
-
33
-
-
33749442356
-
Theoretical and practical approaches for prediction of drug-polymer miscibility and solubility
-
Marsac PJ, Shamblin SL, Taylor LS. Theoretical and practical approaches for prediction of drug-polymer miscibility and solubility. Pharm Res 2006;23:2417-26.
-
(2006)
Pharm Res
, vol.23
, pp. 2417-2426
-
-
Marsac, P.J.1
Shamblin, S.L.2
Taylor, L.S.3
-
34
-
-
68249128120
-
Supersaturating drug delivery systems: The answer to solubility-limited oral bioavailability?
-
Brouwers J, Brewster ME, Augustijns P. Supersaturating drug delivery systems: the answer to solubility-limited oral bioavailability? J Pharm Sci 2009;98:2549-72.
-
(2009)
J Pharm Sci
, vol.98
, pp. 2549-2572
-
-
Brouwers, J.1
Brewster, M.E.2
Augustijns, P.3
-
35
-
-
80055000199
-
Influence of polymer chemistry on crystal growth inhibition of two chemically diverse organic molecules
-
Kestur US, Van Eerdenbrugh B, Taylor LS. Influence of polymer chemistry on crystal growth inhibition of two chemically diverse organic molecules. CrystEngComm 2011;13:6712-18.
-
(2011)
Crystengcomm
, vol.13
, pp. 6712-6718
-
-
Kestur, U.S.1
Van Eerdenbrugh, B.2
Taylor, L.S.3
-
36
-
-
0035895236
-
Crystallization of hydrocortisone acetate: Influence of polymers
-
Raghavan SL, Trividic A, Davis AF, et al. Crystallization of hydrocortisone acetate: influence of polymers. Int J Pharm 2001; 212:213-21.
-
(2001)
Int J Pharm
, vol.212
, pp. 213-221
-
-
Raghavan, S.L.1
Trividic, A.2
Davis, A.F.3
-
37
-
-
0023891244
-
Cyclodextrins increase surface tension and critical micelle concentrations of detergent solutions
-
Saenger W, Muller-Fahrnow A. Cyclodextrins increase surface tension and critical micelle concentrations of detergent solutions. Angew Chem Int Ed Engl 1988;27:393-4.
-
(1988)
Angew Chem Int Ed Engl
, vol.27
, pp. 393-394
-
-
Saenger, W.1
Muller-Fahrnow, A.2
-
38
-
-
36248993922
-
New insights in cyclodextrin: Surfactant mixed systems from the use of neutral and anionic cyclodextrin derivatives
-
García-Río L, Méndez M, Paleo MR, et al. New insights in cyclodextrin: surfactant mixed systems from the use of neutral and anionic cyclodextrin derivatives. J Phys Chem B 2007;111: 12756-64.
-
(2007)
J Phys Chem B
, vol.111
, pp. 12756-12764
-
-
García-Río, L.1
Méndez, M.2
Paleo, M.R.3
-
39
-
-
84905456922
-
Evaluation of different screening methods to understand the dissolution behaviors of amorphous solid dispersions
-
Lee TW, Boersen NA, Yang G, et al. Evaluation of different screening methods to understand the dissolution behaviors of amorphous solid dispersions. Drug Dev Ind Pharm 2014;40: 1072-83.
-
(2014)
Drug Dev Ind Pharm
, vol.40
, pp. 1072-1083
-
-
Lee, T.W.1
Boersen, N.A.2
Yang, G.3
-
40
-
-
84932615507
-
Amorphous azithromycin with improved aqueous solubility and intestinal membrane permeability
-
[Epub ahead of print]
-
Aucamp M, Odendaal R, Liebenberg W, et al. Amorphous azithromycin with improved aqueous solubility and intestinal membrane permeability. Drug Dev Ind Pharm 2014. [Epub ahead of print]. DOI: 10.3109/03639045.2014.931967.
-
(2014)
Drug Dev Ind Pharm
-
-
Aucamp, M.1
Odendaal, R.2
Liebenberg, W.3
-
41
-
-
33751014029
-
Formulation of poorly water-soluble drugs for oral administration: Physicochemical and physiological issues and the lipid formulation classification system
-
Pouton CW. Formulation of poorly water-soluble drugs for oral administration: physicochemical and physiological issues and the lipid formulation classification system. Eur J Pharm Sci 2006;29: 278-87.
-
(2006)
Eur J Pharm Sci
, vol.29
, pp. 278-287
-
-
Pouton, C.W.1
|