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Volumn 41, Issue 11, 2015, Pages 1847-1855

Enhancement of docetaxel solubility using binary and ternary solid dispersion systems

Author keywords

Anti cancer; Apparent solubility; Freeze drying; Solubility parameter; Soluplus

Indexed keywords

2 HYDROXYPROPYL BETA CYCLODEXTRIN; DOCETAXEL; POLOXAMER; POVIDONE; SOLUBILIZER; SOLUPLUS; UNCLASSIFIED DRUG; ANTINEOPLASTIC AGENT; EXCIPIENT; MACROGOL DERIVATIVE; POLYVINYL CAPROLACTAM-POLYVINYL ACETATE-POLYETHYLENE GLYCOL GRAFT COPOLYMER; POLYVINYL DERIVATIVE; TAXOID;

EID: 84979523835     PISSN: 03639045     EISSN: 15205762     Source Type: Journal    
DOI: 10.3109/03639045.2015.1014818     Document Type: Article
Times cited : (37)

References (41)
  • 2
    • 45849092587 scopus 로고    scopus 로고
    • Preparation, characterization and in vitro evaluation of solid dispersions containing docetaxel
    • Chen J, Qiu L, Hu M, et al. Preparation, characterization and in vitro evaluation of solid dispersions containing docetaxel. Drug Dev Ind Pharm 2008;34:588-94.
    • (2008) Drug Dev Ind Pharm , vol.34 , pp. 588-594
    • Chen, J.1    Qiu, L.2    Hu, M.3
  • 3
    • 80054697562 scopus 로고    scopus 로고
    • Pharmaceutical development and preliminary clinical testing of an oral solid dispersion formulation of docetaxel (ModraDoc001)
    • Moes JJ, Koolen SL, Huitema AD, et al. Pharmaceutical development and preliminary clinical testing of an oral solid dispersion formulation of docetaxel (ModraDoc001). Int J Pharm 2011;420: 244-50.
    • (2011) Int J Pharm , vol.420 , pp. 244-250
    • Moes, J.J.1    Koolen, S.L.2    Huitema, A.D.3
  • 4
    • 11244321887 scopus 로고    scopus 로고
    • Oral bioavailability of docetaxel in combination with OC144-093 (ONT-093)
    • Kuppens IE, Bosch TM, van Maanen MJ, et al. Oral bioavailability of docetaxel in combination with OC144-093 (ONT-093). Cancer Chemother Pharmacol 2005;55:72-8.
    • (2005) Cancer Chemother Pharmacol , vol.55 , pp. 72-78
    • Kuppens, I.E.1    Bosch, T.M.2    Van Maanen, M.J.3
  • 5
    • 54349088541 scopus 로고    scopus 로고
    • Preparation and characterization of a submicron lipid emulsion of docetaxel: Submicron lipid emulsion of docetaxel
    • Gao K, Sun J, Liu K, et al. Preparation and characterization of a submicron lipid emulsion of docetaxel: submicron lipid emulsion of docetaxel. Drug Dev Ind Pharm 2008;34:1227-37.
    • (2008) Drug Dev Ind Pharm , vol.34 , pp. 1227-1237
    • Gao, K.1    Sun, J.2    Liu, K.3
  • 6
    • 71549157438 scopus 로고    scopus 로고
    • Absence of both cytochrome P450 3A and P-glycoprotein dramatically increases docetaxel oral bioavailability and risk of intestinal toxicity
    • van Waterschoot RA, Lagas JS, Wagenaar E, et al. Absence of both cytochrome P450 3A and P-glycoprotein dramatically increases docetaxel oral bioavailability and risk of intestinal toxicity. Cancer Res 2009;69:8996-9002.
    • (2009) Cancer Res , vol.69 , pp. 8996-9002
    • Van Waterschoot, R.A.1    Lagas, J.S.2    Wagenaar, E.3
  • 7
    • 0036829187 scopus 로고    scopus 로고
    • Low systemic exposure of oral docetaxel in mice resulting from extensive first-pass metabolism is boosted by ritonavir
    • Bardelmeijer HA, Ouwehand M, Buckle T, et al. Low systemic exposure of oral docetaxel in mice resulting from extensive first-pass metabolism is boosted by ritonavir. Cancer Res 2002;62:6158-64
    • (2002) Cancer Res , vol.62 , pp. 6158-6164
    • Bardelmeijer, H.A.1    Ouwehand, M.2    Buckle, T.3
  • 8
  • 9
    • 77954805866 scopus 로고    scopus 로고
    • Solid dispersion as an approach for bioavailability enhancement of poorly water-soluble drug ritonavir
    • Sinha S, Ali M, Baboota S, et al. Solid dispersion as an approach for bioavailability enhancement of poorly water-soluble drug ritonavir. AAPS PharmSciTech 2010;11:518-27.
    • (2010) AAPS Pharmscitech , vol.11 , pp. 518-527
    • Sinha, S.1    Ali, M.2    Baboota, S.3
  • 10
    • 84896705229 scopus 로고    scopus 로고
    • Influence of different polymers on crystallization tendency and dissolution behavior of cilnidipine in solid dispersions
    • Chen C, Xie X, Li Y, et al. Influence of different polymers on crystallization tendency and dissolution behavior of cilnidipine in solid dispersions. Drug Dev Ind Pharm 2014;40:441-51.
    • (2014) Drug Dev Ind Pharm , vol.40 , pp. 441-451
    • Chen, C.1    Xie, X.2    Li, Y.3
  • 11
    • 0034868680 scopus 로고    scopus 로고
    • The potential of small-scale fusion experiments and the Gordon-Taylor equation to predict the suitability of drug/polymer blends for melt extrusion
    • Forster A, Hempenstall J, Tucker, I, et al. The potential of small-scale fusion experiments and the Gordon-Taylor equation to predict the suitability of drug/polymer blends for melt extrusion. Drug Dev Ind Pharm 2001;27:549-60.
    • (2001) Drug Dev Ind Pharm , vol.27 , pp. 549-560
    • Forster, A.1    Hempenstall, J.2    Tucker, I.3
  • 12
    • 84877077701 scopus 로고    scopus 로고
    • In vitro and in vivo evaluation of amorphous solid dispersions generated by different bench-scale processes, using griseofulvin as a model compound
    • Chiang PC, Cui Y, Ran Y, et al. In vitro and in vivo evaluation of amorphous solid dispersions generated by different bench-scale processes, using griseofulvin as a model compound. AAPS J 2013; 15:608-17.
    • (2013) AAPS J , vol.15 , pp. 608-617
    • Chiang, P.C.1    Cui, Y.2    Ran, Y.3
  • 13
    • 35348987129 scopus 로고    scopus 로고
    • Combined use of crystalline salt forms and precipitation inhibitors to improve oral absorption of celecoxib from solid oral formulations
    • Guzman HR, Tawa M, Zhang Z, et al. Combined use of crystalline salt forms and precipitation inhibitors to improve oral absorption of celecoxib from solid oral formulations. J Pharm Sci 2007;96: 2686-702.
    • (2007) J Pharm Sci , vol.96 , pp. 2686-2702
    • Guzman, H.R.1    Tawa, M.2    Zhang, Z.3
  • 14
    • 84930526016 scopus 로고    scopus 로고
    • Solubility and dissolution enhancement strategies: Current understanding and recent trends
    • Jain S, Patel N, Lin S. Solubility and dissolution enhancement strategies: current understanding and recent trends. Drug Dev Ind Pharm 2014. [Epub ahead of print]. DOI:10.3109/03639045.2014.971027.
    • (2014) Drug Dev Ind Pharm
    • Jain, S.1    Patel, N.2    Lin, S.3
  • 15
    • 77951538902 scopus 로고    scopus 로고
    • Combining HME & solubilization: Soluplus - The solid solution
    • Hardung H, Djuric D, Ali S. Combining HME & solubilization: Soluplus - the solid solution. Drug Deliv Technol 2010;10:20-7.
    • (2010) Drug Deliv Technol , vol.10 , pp. 20-27
    • Hardung, H.1    Djuric, D.2    Ali, S.3
  • 16
    • 84875274738 scopus 로고    scopus 로고
    • Soluplus: A novel polymeric solubilizer for optimization of Carvedilol solid dispersions: Formulation design and effect of method of preparation
    • Shamma RN, Basha M. Soluplus: a novel polymeric solubilizer for optimization of Carvedilol solid dispersions: formulation design and effect of method of preparation. Powder Technol 2013;237:406-14.
    • (2013) Powder Technol , vol.237 , pp. 406-414
    • Shamma, R.N.1    Basha, M.2
  • 17
    • 84902239752 scopus 로고    scopus 로고
    • Data mining of solubility parameters for computational prediction of drug-excipient miscibility
    • Alhalaweh A, Alzghoul A, Kaialy W. Data mining of solubility parameters for computational prediction of drug-excipient miscibility. Drug Dev Ind Pharm 2014;40:904-9.
    • (2014) Drug Dev Ind Pharm , vol.40 , pp. 904-909
    • Alhalaweh, A.1    Alzghoul, A.2    Kaialy, W.3
  • 18
    • 0035845751 scopus 로고    scopus 로고
    • Selection of excipients for melt extrusion with two poorly water-soluble drugs by solubility parameter calculation and thermal analysis
    • Forster A, Hempenstall J, Tucker I, et al. Selection of excipients for melt extrusion with two poorly water-soluble drugs by solubility parameter calculation and thermal analysis. Int J Pharm 2001;226: 147-61.
    • (2001) Int J Pharm , vol.226 , pp. 147-161
    • Forster, A.1    Hempenstall, J.2    Tucker, I.3
  • 19
    • 84879009609 scopus 로고    scopus 로고
    • Prediction of drug-polymer miscibility through the use of solubility parameter-based Flory--uggins interaction parameter and the experimental validation: PEG as model polymer
    • Thakral S, Thakral NK. Prediction of drug-polymer miscibility through the use of solubility parameter-based Flory--uggins interaction parameter and the experimental validation: PEG as model polymer. J Pharm Sci 2013;102:2254-63.
    • (2013) J Pharm Sci , vol.102 , pp. 2254-2263
    • Thakral, S.1    Thakral, N.K.2
  • 20
    • 84875214001 scopus 로고    scopus 로고
    • Cyclodextrin-water soluble polymer ternary complexes enhance the solubility and dissolution behaviour of poorly soluble drugs. Case example: Itraconazole
    • Taupitz T, Dressman JB, Buchanan CM, et al. Cyclodextrin-water soluble polymer ternary complexes enhance the solubility and dissolution behaviour of poorly soluble drugs. Case example: itraconazole. Eur J Pharm Biopharm 2013;83:378-87.
    • (2013) Eur J Pharm Biopharm , vol.83 , pp. 378-387
    • Taupitz, T.1    Dressman, J.B.2    Buchanan, C.M.3
  • 22
    • 84916937130 scopus 로고    scopus 로고
    • Docetaxel epimerization in silicone films: A case of drug excipient incompatibility
    • Mohsin S, Arellano IH, Choudhury NR, et al. Docetaxel epimerization in silicone films: a case of drug excipient incompatibility. Drug Test Anal 2014;6:1076-84.
    • (2014) Drug Test Anal , vol.6 , pp. 1076-1084
    • Mohsin, S.1    Arellano, I.H.2    Choudhury, N.R.3
  • 23
    • 0034633805 scopus 로고    scopus 로고
    • Simple and sensitive high-performance liquid chromatography method for the determination of docetaxel in human plasma or urine
    • Garg MB, Ackland SP. Simple and sensitive high-performance liquid chromatography method for the determination of docetaxel in human plasma or urine. J Chromatogr B Biomed Sci Appl 2000;748: 383-8.
    • (2000) J Chromatogr B Biomed Sci Appl , vol.748 , pp. 383-388
    • Garg, M.B.1    Ackland, S.P.2
  • 24
    • 0032726595 scopus 로고    scopus 로고
    • Solubility parameters as predictors of miscibility in solid dispersions
    • Greenhalgh DJ, Williams AC, Timmins P, et al. Solubility parameters as predictors of miscibility in solid dispersions. J Pharm Sci 1999;88:1182-90.
    • (1999) J Pharm Sci , vol.88 , pp. 1182-1190
    • Greenhalgh, D.J.1    Williams, A.C.2    Timmins, P.3
  • 26
    • 38049173112 scopus 로고    scopus 로고
    • Predicting the solubility of the anti-cancer agent docetaxel in small molecule excipients using computational methods
    • Huynh L, Grant J, Leroux JC, et al. Predicting the solubility of the anti-cancer agent docetaxel in small molecule excipients using computational methods. Pharm Res 2008;25:147-57.
    • (2008) Pharm Res , vol.25 , pp. 147-157
    • Huynh, L.1    Grant, J.2    Leroux, J.C.3
  • 27
    • 80051793564 scopus 로고    scopus 로고
    • Bivalent sequential binding of docetaxel to methyl-beta-cyclodextrin
    • Mazzaferro S, Bouchemal K, Gallard JF, et al. Bivalent sequential binding of docetaxel to methyl-beta-cyclodextrin. Int J Pharm 2011; 416:171-80.
    • (2011) Int J Pharm , vol.416 , pp. 171-180
    • Mazzaferro, S.1    Bouchemal, K.2    Gallard, J.F.3
  • 28
    • 84878880994 scopus 로고    scopus 로고
    • Sulfobutylether-beta-cyclodextrin/chitosan nanoparticles enhance the oral permeability and bioavailability of docetaxel
    • Wu J, Shen Q, Fang L. Sulfobutylether-beta-cyclodextrin/chitosan nanoparticles enhance the oral permeability and bioavailability of docetaxel. Drug Dev Ind Pharm 2013;39:1010-9.
    • (2013) Drug Dev Ind Pharm , vol.39 , pp. 1010-1019
    • Wu, J.1    Shen, Q.2    Fang, L.3
  • 29
    • 33845714689 scopus 로고    scopus 로고
    • Alternative drug formulations of docetaxel: A review
    • Engels FK, Mathot RA, Verweij J. Alternative drug formulations of docetaxel: a review. Anticancer Drugs 2007;18:95-103.
    • (2007) Anticancer Drugs , vol.18 , pp. 95-103
    • Engels, F.K.1    Mathot, R.A.2    Verweij, J.3
  • 30
    • 0035710530 scopus 로고    scopus 로고
    • Docetaxel: Solid state characterization by X-ray powder diffraction and thermogravimetry
    • Pr10-221-Pr10-6
    • Zaske L, Perrin M-A, Leveiller F. Docetaxel: solid state characterization by X-ray powder diffraction and thermogravimetry. J Phys IV France 2001;11:Pr10-221-Pr10-6.
    • (2001) J Phys IV France , vol.11
    • Zaske, L.1    Perrin, M.-A.2    Leveiller, F.3
  • 32
    • 0030896467 scopus 로고    scopus 로고
    • The use of solubility parameters in pharmaceutical dosage form design
    • Hancock BC, York P, Rowe RC. The use of solubility parameters in pharmaceutical dosage form design. Int J Pharm 1997;148:1-21.
    • (1997) Int J Pharm , vol.148 , pp. 1-21
    • Hancock, B.C.1    York, P.2    Rowe, R.C.3
  • 33
    • 33749442356 scopus 로고    scopus 로고
    • Theoretical and practical approaches for prediction of drug-polymer miscibility and solubility
    • Marsac PJ, Shamblin SL, Taylor LS. Theoretical and practical approaches for prediction of drug-polymer miscibility and solubility. Pharm Res 2006;23:2417-26.
    • (2006) Pharm Res , vol.23 , pp. 2417-2426
    • Marsac, P.J.1    Shamblin, S.L.2    Taylor, L.S.3
  • 34
    • 68249128120 scopus 로고    scopus 로고
    • Supersaturating drug delivery systems: The answer to solubility-limited oral bioavailability?
    • Brouwers J, Brewster ME, Augustijns P. Supersaturating drug delivery systems: the answer to solubility-limited oral bioavailability? J Pharm Sci 2009;98:2549-72.
    • (2009) J Pharm Sci , vol.98 , pp. 2549-2572
    • Brouwers, J.1    Brewster, M.E.2    Augustijns, P.3
  • 35
    • 80055000199 scopus 로고    scopus 로고
    • Influence of polymer chemistry on crystal growth inhibition of two chemically diverse organic molecules
    • Kestur US, Van Eerdenbrugh B, Taylor LS. Influence of polymer chemistry on crystal growth inhibition of two chemically diverse organic molecules. CrystEngComm 2011;13:6712-18.
    • (2011) Crystengcomm , vol.13 , pp. 6712-6718
    • Kestur, U.S.1    Van Eerdenbrugh, B.2    Taylor, L.S.3
  • 36
    • 0035895236 scopus 로고    scopus 로고
    • Crystallization of hydrocortisone acetate: Influence of polymers
    • Raghavan SL, Trividic A, Davis AF, et al. Crystallization of hydrocortisone acetate: influence of polymers. Int J Pharm 2001; 212:213-21.
    • (2001) Int J Pharm , vol.212 , pp. 213-221
    • Raghavan, S.L.1    Trividic, A.2    Davis, A.F.3
  • 37
    • 0023891244 scopus 로고
    • Cyclodextrins increase surface tension and critical micelle concentrations of detergent solutions
    • Saenger W, Muller-Fahrnow A. Cyclodextrins increase surface tension and critical micelle concentrations of detergent solutions. Angew Chem Int Ed Engl 1988;27:393-4.
    • (1988) Angew Chem Int Ed Engl , vol.27 , pp. 393-394
    • Saenger, W.1    Muller-Fahrnow, A.2
  • 38
    • 36248993922 scopus 로고    scopus 로고
    • New insights in cyclodextrin: Surfactant mixed systems from the use of neutral and anionic cyclodextrin derivatives
    • García-Río L, Méndez M, Paleo MR, et al. New insights in cyclodextrin: surfactant mixed systems from the use of neutral and anionic cyclodextrin derivatives. J Phys Chem B 2007;111: 12756-64.
    • (2007) J Phys Chem B , vol.111 , pp. 12756-12764
    • García-Río, L.1    Méndez, M.2    Paleo, M.R.3
  • 39
    • 84905456922 scopus 로고    scopus 로고
    • Evaluation of different screening methods to understand the dissolution behaviors of amorphous solid dispersions
    • Lee TW, Boersen NA, Yang G, et al. Evaluation of different screening methods to understand the dissolution behaviors of amorphous solid dispersions. Drug Dev Ind Pharm 2014;40: 1072-83.
    • (2014) Drug Dev Ind Pharm , vol.40 , pp. 1072-1083
    • Lee, T.W.1    Boersen, N.A.2    Yang, G.3
  • 40
    • 84932615507 scopus 로고    scopus 로고
    • Amorphous azithromycin with improved aqueous solubility and intestinal membrane permeability
    • [Epub ahead of print]
    • Aucamp M, Odendaal R, Liebenberg W, et al. Amorphous azithromycin with improved aqueous solubility and intestinal membrane permeability. Drug Dev Ind Pharm 2014. [Epub ahead of print]. DOI: 10.3109/03639045.2014.931967.
    • (2014) Drug Dev Ind Pharm
    • Aucamp, M.1    Odendaal, R.2    Liebenberg, W.3
  • 41
    • 33751014029 scopus 로고    scopus 로고
    • Formulation of poorly water-soluble drugs for oral administration: Physicochemical and physiological issues and the lipid formulation classification system
    • Pouton CW. Formulation of poorly water-soluble drugs for oral administration: physicochemical and physiological issues and the lipid formulation classification system. Eur J Pharm Sci 2006;29: 278-87.
    • (2006) Eur J Pharm Sci , vol.29 , pp. 278-287
    • Pouton, C.W.1


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