Eact, a small molecule activator of TMEM16A, activates TRPV1 and elicits pain- and itch-related behaviours

British Journal of Pharmacology

Volumn 173, Issue 7, 2016, Pages 1208-1218

  Liu, Shenbin ^a,b   Feng, Jing ^a   Luo, Jialie ^a   Yang, Pu ^a   Brett, Thomas J ^a   Hu, Hongzhen ^a  

^a WASHINGTON UNIVERSITY SCHOOL OF MEDICINE   (United States)

^b FUDAN UNIVERSITY   (China)

Author keywords

[No Author keywords available]

Indexed keywords

(3,4,5-TRIMETHOXY-N-(2-METHOXYETHYL)-N-(4-PHENYL-2-THIAZOLYL)BENZAMIDE; BENZAMIDE DERIVATIVE; CHLORIDE CHANNEL; CHLORIDE CHANNEL STIMULATING AGENT; THIAZOLE DERIVATIVE; TMEM16A PROTEIN, MOUSE; TRPV1 PROTEIN, MOUSE; VANILLOID RECEPTOR;

AGONISTS; ANIMAL; ANIMAL BEHAVIOR; CELL CULTURE; CONGENIC STRAIN; DRUG EFFECTS; GENETICS; HUMAN; METABOLISM; PAIN; PAIN RECEPTOR; PRURITUS; PSYCHOLOGY; RAT; SPINAL GANGLION;

ANIMALS; BEHAVIOR, ANIMAL; BENZAMIDES; CELLS, CULTURED; CHLORIDE CHANNEL AGONISTS; CHLORIDE CHANNELS; GANGLIA, SPINAL; HUMANS; MICE, CONGENIC; NOCICEPTORS; PAIN; PRURITUS; RATS; THIAZOLES; TRPV CATION CHANNELS;

EID: 84959572918     PISSN: 00071188     EISSN: 14765381     Source Type: Journal    
DOI: 10.1111/bph.13420     Document Type: Article

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