High-throughput screening for allosteric modulators of GPCRs

Methods in Molecular Biology

Volumn 1335, Issue , 2015, Pages 223-240

  Bertekap, Robert L ^a   Burford, Neil T ^a   Li, Zhuyin ^a   Alt, Andrew ^a  

^a NONE

Author keywords

Allosteric; Calcium flux; FDSS; FLIPR; G protein coupled receptor; HTS; NAM; PAM; SAM

Indexed keywords

G PROTEIN COUPLED RECEPTOR; LIGAND; CALCIUM;

ALLOSTERISM; ARTICLE; BINDING SITE; HIGH THROUGHPUT SCREENING; MOLECULAR LIBRARY; PRIORITY JOURNAL; RECEPTOR UPREGULATION; SIGNAL TRANSDUCTION; AGONISTS; CELL LINE; CHEMISTRY; DRUG EFFECTS; METABOLISM; PRECLINICAL STUDY; PROCEDURES;

ALLOSTERIC REGULATION; CALCIUM; CELL LINE; DRUG EVALUATION, PRECLINICAL; HIGH-THROUGHPUT SCREENING ASSAYS; RECEPTORS, G-PROTEIN-COUPLED;

EID: 84938828476     PISSN: 10643745     EISSN: None     Source Type: Book Series    
DOI: 10.1007/978-1-4939-2914-6_15     Document Type: Article

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