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ChemMedChem

Volumn 9, Issue 11, 2014, Pages 2439-2444

In vitro antiamoebic activity evaluation and docking studies of metronidazole-triazole hybrids

(6) Negi, Beena a Raj, K Kranthi a,b Siddiqui, Shadab Miyan c Ramachandran, Dittakavi b Azam, Amir c Rawat, Diwan S a

a UNIVERSITY OF DELHI (India)

b ACHARYA NAGARJUNA UNIVERSITY (India)

c JAMIA MILLIA ISLAMIA CENTRAL UNIVERSITY (India)

Author keywords

antiprotozoal agents; Entamoeba histolytica; inhibitors; metronidazole; thioredoxin reductase

Indexed keywords

2 PYRIDYL (1,2,3 TRIAZOLYL)METRONIDAZOLE; ARGININE; METRONIDAZOLE; THIOREDOXIN REDUCTASE; TRIAZOLE DERIVATIVE; UNCLASSIFIED DRUG; ANTIPROTOZOAL AGENT;

AMEBIASIS; ARTICLE; DRUG ACTIVITY; DRUG CONFORMATION; DRUG SCREENING; DRUG STRUCTURE; ENTAMOEBA HISTOLYTICA; IN VITRO STUDY; MOLECULAR DOCKING; NONHUMAN; PRIORITY JOURNAL; BINDING SITE; CHEMISTRY; DRUG EFFECTS; ENZYMOLOGY; IC50; METABOLISM; PROTEIN TERTIARY STRUCTURE;

ANTIPROTOZOAL AGENTS; BINDING SITES; ENTAMOEBA HISTOLYTICA; INHIBITORY CONCENTRATION 50; METRONIDAZOLE; MOLECULAR DOCKING SIMULATION; PROTEIN STRUCTURE, TERTIARY; THIOREDOXIN-DISULFIDE REDUCTASE; TRIAZOLES;

EID: 84927158464 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201402240 Document Type: Article

Times cited : (24)

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