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Volumn 21, Issue 16, 2015, Pages 6265-6271

Cyclic isoDGR and RGD Peptidomimetics Containing Bifunctional Diketopiperazine Scaffolds are Integrin Antagonists

(11) Panzeri, Silvia a Zanella, Simone b Arosio, Daniela c Vahdati, Leila a Dal Corso, Alberto b Pignataro, Luca b,c Paolillo, Mayra d Schinelli, Sergio d Belvisi, Laura b,c Gennari, Cesare b,c Piarulli, Umberto a

a UNIVERSITY OF INSUBRIA (Italy)

b UNIVERSITY OF MILAN (Italy)

c CNR Consiglio Nazionale delle Ricerche (Italy)

d UNIVERSITY OF PAVIA (Italy)

Author keywords

cell adhesion; drug design; drug discovery; peptidomimetics; phosphorylation

Indexed keywords

CELL ADHESION; CELL DEATH; CELLS; CYTOLOGY; DRUG PRODUCTS; LIGANDS; MOBILE SECURITY; PHOSPHORYLATION;

COMPETITIVE BINDING ASSAY; DIKETOPIPERAZINES; DRUG DESIGN; DRUG DISCOVERY; GLIOBLASTOMA CELLS; INTEGRIN RECEPTORS; PEPTIDOMIMETICS; TRANSDUCTION PATHWAYS;

SCAFFOLDS (BIOLOGY);

ALPHAVBETA5 INTEGRIN; ANTINEOPLASTIC AGENT; CYCLOPEPTIDE; PEPTIDOMIMETIC AGENT; PHARMACOLOGY; PIPERAZINEDIONE; VITRONECTIN RECEPTOR;

APOPTOSIS; CHEMISTRY; DRUG EFFECTS; DRUG THERAPY; GLIOBLASTOMA; HUMAN; METABOLISM; SIGNAL TRANSDUCTION; TUMOR CELL LINE;

ANTINEOPLASTIC AGENTS; APOPTOSIS; CELL LINE, TUMOR; CHEMISTRY; DIKETOPIPERAZINES; DRUG EFFECTS; DRUG THERAPY; GLIOBLASTOMA; HUMANS; INTEGRIN ALPHAVBETA3; METABOLISM; PEPTIDES, CYCLIC; PEPTIDOMIMETICS; PHARMACOLOGY; RECEPTORS, VITRONECTIN; SIGNAL TRANSDUCTION;

EID: 84926288646 PISSN: 09476539 EISSN: 15213765 Source Type: Journal
DOI: 10.1002/chem.201406567 Document Type: Article

Times cited : (36)

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