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Angewandte Chemie - International Edition

Volumn 54, Issue 12, 2015, Pages 3735-3739

Fragment screening and druggability assessment for the CBP/p300 KIX domain through protein-observed 19F NMR spectroscopy

(3) Gee, Clifford T a Koleski, Edward J a Pomerantz, William C K a

a UNIVERSITY OF MINNESOTA (United States)

Author keywords

biomolecular NMR; fluorine; fragment screening; protein protein interactions; transcription

Indexed keywords

CHEMICAL ANALYSIS; FLUORINE; LIGANDS; MOLECULES; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; SPECTRUM ANALYSIS; TRANSCRIPTION; TRANSCRIPTION FACTORS;

AROMATIC SIDE CHAINS; BIO-MOLECULAR; CONFORMATIONAL DYNAMICS; CREB BINDING PROTEINS; MEDICINAL CHEMISTRY; PROTEIN-PROTEIN INTERACTIONS; STRUCTURAL INFORMATION; TRANSCRIPTION FACTOR BINDING;

PROTEINS;

CYCLIC AMP RESPONSIVE ELEMENT BINDING PROTEIN BINDING PROTEIN; E1A ASSOCIATED P300 PROTEIN; EP300 PROTEIN, HUMAN; FLUORINE; LIGAND; PROTEIN BINDING;

ANIMAL; BINDING SITE; CHEMISTRY; HUMAN; METABOLISM; NUCLEAR MAGNETIC RESONANCE; PROTEIN DOMAIN; PROTEIN TERTIARY STRUCTURE; STRUCTURE ACTIVITY RELATION;

ANIMALS; BINDING SITES; CREB-BINDING PROTEIN; E1A-ASSOCIATED P300 PROTEIN; FLUORINE; HUMANS; LIGANDS; NUCLEAR MAGNETIC RESONANCE, BIOMOLECULAR; PROTEIN BINDING; PROTEIN INTERACTION DOMAINS AND MOTIFS; PROTEIN STRUCTURE, TERTIARY; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84924373564 PISSN: 14337851 EISSN: 15213773 Source Type: Journal
DOI: 10.1002/anie.201411658 Document Type: Article

Times cited : (43)

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