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Bioorganic and Medicinal Chemistry Letters

Volumn 24, Issue 24, 2014, Pages 5621-5626

Structure activity relationship study of curcumin analogues toward the amyloid-beta aggregation inhibitor

(5) Endo, Hitoshi a Nikaido, Yuri a Nakadate, Mamiko a Ise, Satomi a Konno, Hiroyuki a

a YAMAGATA UNIVERSITY (Japan)

Author keywords

Aggregation inhibitor; Alzheimer's disease; Amyloid beta; Curcumin; Water solubility

Indexed keywords

1,3 DIKETONE; 3,4 DIMETHOXYBENZALDEHYDE; ALKENE; AMYLOID BETA PROTEIN; BISMETHOXYCURCUMIN; CATECHOL PYROGALLOL; CURCUMIN; DESMETHYL CURCUMIN; M PHENOL; O HYDROXY CURCUMIN DERIVATIVE; O PHENOL; P HYDROXY; PHENOL; PHENYL DIKETONE; TETRAHYDROCURCUMIN; UNCLASSIFIED DRUG; WATER; PROTEIN BINDING;

ALDOL REACTION; ARTICLE; DRUG BIOAVAILABILITY; DRUG CONJUGATION; DRUG POTENCY; DRUG STRUCTURE; ENZYME ACTIVITY; ENZYME INHIBITION; HUMAN; HYDROPHOBICITY; MOLECULAR INTERACTION; PHARMACOPHORE; PROTEIN AGGREGATION; REACTION OPTIMIZATION; SOLUBILITY; STRUCTURE ACTIVITY RELATION; ANTAGONISTS AND INHIBITORS; CHEMISTRY; CONFORMATION; KINETICS; METABOLISM; QUANTUM THEORY; SYNTHESIS;

AMYLOID BETA-PEPTIDES; CURCUMIN; HUMANS; KINETICS; MOLECULAR CONFORMATION; PROTEIN BINDING; QUANTUM THEORY; SOLUBILITY; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84911872504 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2014.10.076 Document Type: Article

Times cited : (45)

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