Agonist and antagonist binding in human glycine receptors

Biochemistry

Volumn 53, Issue 38, 2014, Pages 6041-6051

  Yu, Rilei ^a   Hurdiss, Eliott ^b   Greiner, Timo ^b   Lape, Remigijus ^b   Sivilotti, Lucia ^b   Biggin, Philip C ^a  

^a UNIVERSITY OF OXFORD   (United Kingdom)

^b UNIVERSITY COLLEGE LONDON   (United Kingdom)

Author keywords

[No Author keywords available]

Indexed keywords

GLYCINE RECEPTOR;

GLYCINE; GLYCINE RECEPTOR; GLYCINE RECEPTOR AGONIST; GLYCINE RECEPTOR ANTAGONIST; STRYCHNINE; WATER;

ARTICLE; CONFORMATIONAL TRANSITION; CONTROLLED STUDY; DRUG BINDING SITE; DRUG CONFORMATION; DRUG RECEPTOR BINDING; EMBRYO; HUMAN; HUMAN CELL; LIGAND BINDING; MOLECULAR DYNAMICS; MOLECULAR INTERACTION; MOLECULAR MODEL; MOLECULAR SIZE; PATCH CLAMP TECHNIQUE; PROTEIN INTERACTION; SITE DIRECTED MUTAGENESIS; VALIDATION STUDY; AGONISTS; ANTAGONISTS AND INHIBITORS; CHEMICAL STRUCTURE; ENZYME ACTIVE SITE; METABOLISM; PROTEIN CONFORMATION;

CATALYTIC DOMAIN; HUMANS; MODELS, MOLECULAR; PROTEIN CONFORMATION; RECEPTORS, GLYCINE;

EID: 84907462413     PISSN: 00062960     EISSN: 15204995     Source Type: Journal    
DOI: 10.1021/bi500815f     Document Type: Article

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