Site-specific fluorescence reveals distinct structural changes with GABA receptor activation and antagonism

Nature Neuroscience

Volumn 5, Issue 11, 2002, Pages 1163-1168

  Chang, Yongchang ^a   Weiss, David S ^a  

^a University of Alabama at Birmingham   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

3 AMINOPROPANEPHOSPHINIC ACID; 3 AMINOPROPYL(METHYL)PHOSPHINIC ACID; 4 AMINOBUTYRIC ACID RECEPTOR; 4 AMINOBUTYRIC ACID RECEPTOR BLOCKING AGENT; CROTONIC ACID DERIVATIVE; CYSTEINE; GABAERGIC RECEPTOR AFFECTING AGENT; PICROTOXIN;

ALLOSTERISM; AMINO TERMINAL SEQUENCE; ANIMAL CELL; ARTICLE; CONFORMATIONAL TRANSITION; CONTROLLED STUDY; DRUG BINDING SITE; DRUG RECEPTOR BINDING; ELECTROPHYSIOLOGY; FEMALE; FLUORESCENCE; LIGAND BINDING; NONHUMAN; OOCYTE; PRIORITY JOURNAL; PROTEIN DOMAIN; SYNAPTIC TRANSMISSION; XENOPUS LAEVIS;

ALLOSTERIC REGULATION; ANIMALS; BINDING, COMPETITIVE; FEMALE; FLUORESCENT DYES; GABA ANTAGONISTS; GAMMA-AMINOBUTYRIC ACID; ION CHANNEL GATING; OOCYTES; PICROTOXIN; PROTEIN STRUCTURE, TERTIARY; RECEPTORS, GABA; RECOMBINANT PROTEINS; STRUCTURE-ACTIVITY RELATIONSHIP; XENOPUS LAEVIS;

EID: 0036830645     PISSN: 10976256     EISSN: None     Source Type: Journal    
DOI: 10.1038/nn926     Document Type: Article

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