메뉴 건너뛰기




Volumn 19, Issue 3, 2014, Pages 24-29

Polymorph myths

Author keywords

[No Author keywords available]

Indexed keywords

ACETAZOLAMIDE; BARBITURIC ACID DERIVATIVE; CARBAMAZEPINE; CHALCONE; FLUFENAMIC ACID; GLYCINE; MANNITOL; PAROXETINE; PHENYLBUTAZONE; RANITIDINE; RIMONABANT; RITONAVIR; SULFATHIAZOLE;

EID: 84907368874     PISSN: 13608606     EISSN: None     Source Type: Trade Journal    
DOI: None     Document Type: Review
Times cited : (6)

References (61)
  • 5
    • 79960037731 scopus 로고    scopus 로고
    • Quality by design (QbD) based crystallization process development for the polymorphs of tolbutamide
    • Thinunahari S, Chow PS, Tan RBH (2011) Quality by design (QbD) based crystallization process development for the polymorphs of tolbutamide. Cryst Growth Des 11:3027-3038
    • (2011) Cryst Growth des , vol.11 , pp. 3027-3038
    • Thinunahari, S.1    Chow, P.S.2    Tan, R.B.H.3
  • 6
    • 17644407654 scopus 로고    scopus 로고
    • Crystalline polymorph selection and discovery with polymer heteronuclei
    • DOI 10.1021/ja042561m
    • Price CP, Gresniak AL, Matzger AJ (2005) Crystalline polymorph selection and discovery with polymer heteronuclei J Amer Chem Soc 127:5512-5517 (Pubitemid 40569862)
    • (2005) Journal of the American Chemical Society , vol.127 , Issue.15 , pp. 5512-5517
    • Price, C.P.1    Grzesiak, A.L.2    Matzger, A.J.3
  • 7
    • 35148817932 scopus 로고    scopus 로고
    • Survival of the fittest polymorph: How fast nucleation can lose out to fast growth
    • Yu L (2007) Survival of the fittest polymorph: how fast nucleation can lose out to fast growth. CrystEngComm 9:741-751
    • (2007) CrystEngComm , vol.9 , pp. 741-751
    • Yu, L.1
  • 9
    • 25444456397 scopus 로고    scopus 로고
    • Effect of supersaturation on the crystallization of phenylbutazone polymorphs
    • Datta S, Grant DWJ (2005) Effect of supersaturation on the crystallization of phenylbutazone polymorphs Cryst Res Technol 40: 233-242
    • (2005) Cryst Res Technol , vol.40 , pp. 233-242
    • Datta, S.1    Grant, D.W.J.2
  • 10
    • 84860467345 scopus 로고    scopus 로고
    • Direct comparison of α and γ growth rates in acidic and basic solution: New insights into glycine polymorphism
    • Han G, Chow PS, Tan RBH (2012) Direct comparison of α and γ growth rates in acidic and basic solution: New insights into glycine polymorphism. Cryst Growth Des 12:2213-2220
    • (2012) Cryst Growth des , vol.12 , pp. 2213-2220
    • Han, G.1    Chow, P.S.2    Tan, R.B.H.3
  • 11
    • 0031048775 scopus 로고    scopus 로고
    • The polymorphic drug substances of the european pharmacopoeia. Part 9. Physicochemical properties and crystal structure of acetazolamide crystal forms
    • DOI 10.1021/js960264c
    • Greisser U, Burger A, Mereiter K (1997) The polymorphic drug substances of the European pharmacopoeia part 9. Properties and crystal structure of acetazolamide crystal forms J Pharm Sci 86: 352-358 (Pubitemid 27113771)
    • (1997) Journal of Pharmaceutical Sciences , vol.86 , Issue.3 , pp. 352-358
    • Griesser, U.J.1    Burger, A.2    Mereiter, K.3
  • 12
    • 0032392648 scopus 로고    scopus 로고
    • Development of a seeding technique for the crystallisation of the metastable A modification of Abecarnil
    • Beckmann W, Nikisch K, Budde U (1998) Development of a seeding technique for the crystallisation of the metastable A modification of Abecarnil. Org Process Res Dev 2:298-304
    • (1998) Org Process Res Dev , vol.2 , pp. 298-304
    • Beckmann, W.1    Nikisch, K.2    Budde, U.3
  • 15
    • 84874496375 scopus 로고    scopus 로고
    • Crystal nucleation kinetics in confined spaces
    • Kozisek Z (2013) Crystal nucleation kinetics in confined spaces. CrystEngComm 15:2269-2274
    • (2013) CrystEngComm , vol.15 , pp. 2269-2274
    • Kozisek, Z.1
  • 16
    • 0023171650 scopus 로고
    • PHASE TRANSFORMATIONS IN EMULSIONS: PART II: POLYMORPHISM FOR ORGANIC SUBSTANCES.
    • Dumas JP, Tounsi F, Babin L (1987) Phase transformations in emulsions part II: Polymorphism for organic substances. J Dispersion Sci Technol 8:29-54 (Pubitemid 17573707)
    • (1987) Journal of Dispersion Science and Technology , vol.8 , Issue.1 , pp. 29-54
    • Dumas, J.P.1    Tounsi, F.2    Babin, L.3
  • 17
    • 34250102892 scopus 로고
    • Thermal analysis and infrared spectroscopic investigations of polymorphic organic compounds
    • Kuhnert-Brandstaetter M, Riedmann (1987) Thermal analysis and infrared spectroscopic investigations of polymorphic organic compounds. Mikrochim Acta II 107-120
    • (1987) Mikrochim Acta , vol.2 , pp. 107-120
    • Kuhnert-Brandstaetter, M.1    Riedmann2
  • 18
    • 27544499568 scopus 로고    scopus 로고
    • Crystallization on confined engineered surfaces: A method to control crystal size and generate different polymorphs
    • DOI 10.1021/ja055416x
    • Lee AY, Lee IS, Dette SS, Boerner J, Myerson AS (2005) Crystallization on confined engineered surfaces: A method to control crystal size and generate different polymorphs. J Amer Chem Soc 127: 14982-14983 (Pubitemid 41547338)
    • (2005) Journal of the American Chemical Society , vol.127 , Issue.43 , pp. 14982-14983
    • Lee, A.Y.1    Lee, I.S.2    Dette, S.S.3    Boerner, J.4    Myerson, A.S.5
  • 20
    • 0346047208 scopus 로고    scopus 로고
    • Polymorph generation in capillary spaces: The preparation and structural analysis of a metastable polymorph of nambumetone
    • Chyall LJ, Tower JM, Coates DA, Houston TL Childs SL (2002) Polymorph generation in capillary spaces: the preparation and structural analysis of a metastable polymorph of nambumetone. Cryst Growth Des 2:505-510
    • (2002) Cryst Growth des , vol.2 , pp. 505-510
    • Chyall, L.J.1    Tower, J.M.2    Coates, D.A.3    Houston, T.L.4    Childs, S.L.5
  • 22
    • 33846529897 scopus 로고    scopus 로고
    • Contact line crystallization to obtain metastable polymorphs
    • Capes JS, Cameron RE (2007) Contact line crystallization to obtain metastable polymorphs. Cryst Growth Des 7:108-112
    • (2007) Cryst Growth des , vol.7 , pp. 108-112
    • Capes, J.S.1    Cameron, R.E.2
  • 23
    • 84907319362 scopus 로고    scopus 로고
    • Access to single crystals of (+/-) form IV of Modafinil by crystallization in gels: Comparison between (+/-) forms I, III, IV and (-) form I
    • Mahieux J, Sanselme M, Cocquerel G (2013) Access to single crystals of (+/-) form IV of Modafinil by crystallization in gels: Comparison between (+/-) forms I, III, IV and (-) form I. Cryst Growth Des 13:98-917
    • (2013) Cryst Growth des , vol.13 , pp. 98-917
    • Mahieux, J.1    Sanselme, M.2    Cocquerel, G.3
  • 25
    • 84887465704 scopus 로고    scopus 로고
    • A method for generating a metastable crystal in a microdroplet
    • Teshima Y, Maeki M, Yamashita K, Miyazaki M (2013) A method for generating a metastable crystal in a microdroplet. CrystEngComm 15, 9874-9877
    • (2013) CrystEngComm , vol.15 , pp. 9874-9877
    • Teshima, Y.1    Maeki, M.2    Yamashita, K.3    Miyazaki, M.4
  • 26
    • 79953852843 scopus 로고    scopus 로고
    • Stable polymorphs crystallized directly under thermodynamic control in three-dimensional nanoconfinement: A generic methodology
    • Nicholson CE, Chen C, Mendis B, Cooper SJ (2011) Stable polymorphs crystallized directly under thermodynamic control in three-dimensional nanoconfinement: a generic methodology. Cryst Growth Des 11:363-366
    • (2011) Cryst Growth des , vol.11 , pp. 363-366
    • Nicholson, C.E.1    Chen, C.2    Mendis, B.3    Cooper, S.J.4
  • 27
    • 34548558727 scopus 로고    scopus 로고
    • Crystallization of soluble proteins in vapour diffusion for Xray crystallography
    • Benvenuti M, Mangani S (2007) Crystallization of soluble proteins in vapour diffusion for Xray crystallography. Nature Protocols 2:1633-1653
    • (2007) Nature Protocols , vol.2 , pp. 1633-1653
    • Benvenuti, M.1    Mangani, S.2
  • 28
    • 84862534163 scopus 로고    scopus 로고
    • Non-amorphism in flufenamic acid and a new record for a polymorphic compound with solved structures
    • Lopez-Mejiers V, Kampf JW Matzger AJ (2012) Non-amorphism in flufenamic acid and a new record for a polymorphic compound with solved structures. J Amer Chem Soc 134:9872-9875
    • (2012) J Amer Chem Soc , vol.134 , pp. 9872-9875
    • Lopez-Mejiers, V.1    Kampf, J.W.2    Matzger, A.J.3
  • 29
    • 0017599263 scopus 로고
    • Crystallographic properties of flufenamic acid
    • Krc J (1977) Crystallographic properties of flufenamic acid Microscope 25:31-54
    • (1977) Microscope , vol.25 , pp. 31-54
    • Krc, J.1
  • 31
    • 84907330844 scopus 로고
    • Molecular compounds, crystalline solid solutions and new cases of polymorphism in barbiturates II. Mikrochim Acta 50:1055-1074: (1963): Idem III
    • Kuhnert-Brandstaetter M Aepers M (1962) Molecular compounds, crystalline solid solutions and new cases of polymorphism in barbiturates II. Mikrochim Acta 50:1055-1074: (1963): idem III. Mikrochim Acta 2:360-363
    • (1962) Mikrochim Acta , vol.2 , pp. 360-363
    • Kuhnert-Brandstaetter, M.1    Aepers, M.2
  • 32
    • 74049123587 scopus 로고    scopus 로고
    • Structural features, phase relationships and transformation behaviour of the polymorphs I-VI of phenobarbitone
    • Zencirci N, Gelbrich T, Apperley DC, Harris RK, Kahlenberg V Griesser U (2012) Structural features, phase relationships and transformation behaviour of the polymorphs I-VI of phenobarbitone. Cryst Growth Des 10:302-313
    • (2012) Cryst Growth des , vol.10 , pp. 302-313
    • Zencirci, N.1    Gelbrich, T.2    Apperley, D.C.3    Harris, R.K.4    Kahlenberg, V.5    Griesser, U.6
  • 34
    • 84918353099 scopus 로고
    • Systematic investigation of the polymorphism of organic substances
    • Weygand C (1929) Systematic investigation of the polymorphism of organic substances. Liebigs Ann 472:143-179
    • (1929) Liebigs Ann , vol.472 , pp. 143-179
    • Weygand, C.1
  • 36
    • 84907307557 scopus 로고
    • Repertoire des composés organiques polymorphes
    • Deffet L (1942) Repertoire des composés organiques polymorphes. Desoer Liege
    • (1942) Desoer Liege
    • Deffet, L.1
  • 37
    • 84879005796 scopus 로고    scopus 로고
    • Rimonabant dimorphism and the pressure-temperature phase diagram. A delicate case of overall monotropic behaviour
    • Perrin M-A, Bauer M, Barrio M, Tament JL, Ceolin R, Rietvelt IB (2013) Rimonabant dimorphism and the pressure-temperature phase diagram. A delicate case of overall monotropic behaviour. J Pharm Sci 102:2311-2321
    • (2013) J Pharm Sci , vol.102 , pp. 2311-2321
    • Perrin, M.-A.1    Bauer, M.2    Barrio, M.3    Tament, J.L.4    Ceolin, R.5    Rietvelt, I.B.6
  • 38
    • 0842306206 scopus 로고    scopus 로고
    • Qualitative and quantitative study of polymorphic forms in drug formulations by near infrared FT-Raman spectroscopy
    • DOI 10.1016/j.molstruc.2003.09.002
    • Auer ME, Griesser UJ, Sawatski J (2003) Qualitative and quantitative study of polymorphic forms in drug formulations by near FT-Raman spectroscopy. J Mol Sci 661-662:307-317 (Pubitemid 38169065)
    • (2003) Journal of Molecular Structure , vol.661-662 , Issue.1-3 , pp. 307-317
    • Auer, M.E.1    Griesser, U.J.2    Sawatzki, J.3
  • 39
    • 21344473636 scopus 로고    scopus 로고
    • Statistical analysis of differences in the Raman spectra of polymorphs
    • DOI 10.1002/jps.20355
    • Mehrens SM, Kale UJ, Qu X, (2005) Statistical analysis of differences in the Raman spectra of polymorphs. J Pharm Sci 94:1354-1367 (Pubitemid 40904198)
    • (2005) Journal of Pharmaceutical Sciences , vol.94 , Issue.6 , pp. 1354-1367
    • Mehrens, S.M.1    Kale, U.J.2    Qu, X.3
  • 40
    • 33750906393 scopus 로고    scopus 로고
    • Characterization of temperature-induced phase transformations in five polymorphs of sulfathiazole by terahertz pulsed spectroscopy and differential scanning calorimetry
    • Zeitler JA, Newnham DA, Taday PF, Threlfall TL, Lancaster RW, Berg RW, Strachan CJ, Pepper M, Gordon KC, Rades T (2006) Characterization of temperature-induced phase transformations in five polymorphs of sulfathiazole by terahertz pulsed spectroscopy and differential scanning calorimetry. J Pharm Sci 95:2485-2498
    • (2006) J Pharm Sci , vol.95 , pp. 2485-2498
    • Zeitler, J.A.1    Newnham, D.A.2    Taday, P.F.3    Threlfall, T.L.4    Lancaster, R.W.5    Berg, R.W.6    Strachan, C.J.7    Pepper, M.8    Gordon, K.C.9    Rades, T.10
  • 41
    • 84858804231 scopus 로고    scopus 로고
    • Atomic pairwise distribution function analysis of the amorphous phase prepared by different routes
    • Boetker JP, Koradia V, Savolainen M, Rades T, Rantanen J (2012) Atomic pairwise distribution function analysis of the amorphous phase prepared by different routes. Pharmaceutics 4:93-103
    • (2012) Pharmaceutics , vol.4 , pp. 93-103
    • Boetker, J.P.1    Koradia, V.2    Savolainen, M.3    Rades, T.4    Rantanen, J.5
  • 43
    • 0347365744 scopus 로고    scopus 로고
    • Structural and thermodynamic explanations of Ostwald's rule
    • Threlfall TL (2003) Structural and thermodynamic explanations of Ostwald's rule. Org Process Res Dev 7:1017-1027
    • (2003) Org Process Res Dev , vol.7 , pp. 1017-1027
    • Threlfall, T.L.1
  • 44
    • 42949121619 scopus 로고    scopus 로고
    • Characterization of the "hygroscopic" properties of active pharmaceutical ingredients
    • Newman AW, Reutzel-Edens SM, Zografi G (2008) Characterization of the "hygroscopic" properties of active pharmaceutical ingredients. J Pharm Sci 97:1047-1059
    • (2008) J Pharm Sci , vol.97 , pp. 1047-1059
    • Newman, A.W.1    Reutzel-Edens, S.M.2    Zografi, G.3
  • 45
    • 15444379969 scopus 로고    scopus 로고
    • Solid state structures and temperature/evacuation-induced dehydration of sodium saccharinate 1.875 hydrate
    • Naumov P, Jovanovski G, Gupee O, Kaitner B, Rae AD, Ng SW (2005) Solid state structures and temperature/evacuation-induced dehydration of sodium saccharinate 1.875 hydrate. Angew Chem Int Eng 44:1251
    • (2005) Angew Chem Int Eng , vol.44 , pp. 1251
    • Naumov, P.1    Jovanovski, G.2    Gupee, O.3    Kaitner, B.4    Rae, A.D.5    Ng, S.W.6
  • 47
    • 0034680560 scopus 로고    scopus 로고
    • Efficient pyridinyl functionalization: Synthesis of 10,10-bis(2-fluoro-4- pyridinyl)methyl}9(10H)-anthacenone (DMP543) an acetylcholine release enhancing agent
    • Pesti JA, Huhn JF, Yin J, Xing Y, Fortunak JM, Earl RA (2000) Efficient pyridinyl functionalization: Synthesis of 10,10-bis[(2-fluoro-4-pyridinyl) methyl}9(10H)-anthacenone (DMP543) an acetylcholine release enhancing agent. J Org Chem 65:7718-7722
    • (2000) J Org Chem , vol.65 , pp. 7718-7722
    • Pesti, J.A.1    Huhn, J.F.2    Yin, J.3    Xing, Y.4    Fortunak, J.M.5    Earl, R.A.6
  • 48
    • 0001732841 scopus 로고
    • Studies of the formation and transformation of solid substances
    • Ostwald W (1897) Studies of the formation and transformation of solid substances. Zeits Phys Chem 22:289-330
    • (1897) Zeits Phys Chem , vol.22 , pp. 289-330
    • Ostwald, W.1
  • 50
    • 0000776859 scopus 로고
    • Polymorphism
    • Fox D, Labes MM, Weissberger A Wiley-Interscience New York
    • Mc Crone WC (1965) Polymorphism. In physics and chemistry of the solid state Fox D, Labes MM, Weissberger A Wiley-Interscience New York Vol 2 725-767
    • (1965) Physics and Chemistry of the Solid State , vol.2 , pp. 725-767
    • Mc Crone, W.C.1
  • 51
    • 25444489017 scopus 로고    scopus 로고
    • And another comment on pseudopolymorphism
    • Bernstein J (2005) ...And another comment on pseudopolymorphism. Cryst Growth Des 5:1661-1662
    • (2005) Cryst Growth des , vol.5 , pp. 1661-1662
    • Bernstein, J.1
  • 52
    • 19744382415 scopus 로고    scopus 로고
    • Pseudopolymorph: A polemic
    • Seddon K (2004) Pseudopolymorph: a polemic. Cryst Growth Des 4:1087
    • (2004) Cryst Growth des , vol.4 , pp. 1087
    • Seddon, K.1
  • 54
    • 8844247861 scopus 로고    scopus 로고
    • Crystal and co-crystal
    • Desiraju GR (2004) Crystal and co-crystal. Cryst Growth Des 4:1089-1096
    • (2004) Cryst Growth des , vol.4 , pp. 1089-1096
    • Desiraju, G.R.1
  • 57
    • 0032531779 scopus 로고    scopus 로고
    • Disappearing polymorphs and the role of reaction by-products: The case of sulphathiazole
    • DOI 10.1016/S0378-5173(98)00205-1, PII S0378517398002051
    • Blagden N, Davey RJ, Roberts R, Rowe R (1998) Disappearing polymorphs and the role of reaction byproducts: the case of sulfathiazole. Int J Pharm 172:169-177 (Pubitemid 28430254)
    • (1998) International Journal of Pharmaceutics , vol.172 , Issue.1-2 , pp. 169-177
    • Blagden, N.1    Davey, R.J.2    Rowe, R.3    Roberts, R.4
  • 58
    • 33845281790 scopus 로고
    • Giorgio Piccardi (1895-1972) Italian physical chemist and master of the sun
    • Kaufmann GB, Belloni L (1987) Giorgio Piccardi (1895-1972) Italian physical chemist and master of the sun. J Chem Ed 64:205-8:
    • (1987) J Chem Ed , vol.64 , pp. 205-208
    • Kaufmann, G.B.1    Belloni, L.2
  • 59
    • 72849175720 scopus 로고
    • Surrounding space and life. Effect of terrestrial solar and cosmic phenomena on physico-chemical and biological processes
    • Piccardi G (1960) Surrounding space and life. Effect of terrestrial solar and cosmic phenomena on physico-chemical and biological processes. Minerva Medica 51:1554-1555
    • (1960) Minerva Medica , vol.51 , pp. 1554-1555
    • Piccardi, G.1
  • 60
    • 0031808764 scopus 로고    scopus 로고
    • Physicochemical characterization of the orthorhombic polymorph of paracetamol crystallised from solution
    • Nichols G, Frampton CS (1998) Physicochemical characterization of the orthorhombic polymorph of paracetamol crystallised from solution. J Pharm Sci 87:684-693
    • (1998) J Pharm Sci , vol.87 , pp. 684-693
    • Nichols, G.1    Frampton, C.S.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.