SCOPUS 정보 검색 플랫폼

Volumn 5, Issue 10, 2014, Pages 3929-3935

Polythiazole linkers as functional rigid connectors: A new RGD cyclopeptide with enhanced integrin selectivity

(10) Ruiz Rodriguez J a Miguel, M b Preciado, S b Acosta, G A a,d Adan, J c Bidon Chanal, A d Luque, F J d Mitjans, F c Lavilla, R b,d Albericio, F a,d,e

a INSTITUTE FOR RESEARCH IN BIOMEDICINE (Spain)

b Barcelona Science Park (Spain)

c LEITAT TECHNOLOGICAL CENTER (Spain)

d UNIVERSITY OF BARCELONA (Spain)

e UNIVERSITY OF KWAZULU NATAL (South Africa)

Author keywords

[No Author keywords available]

Indexed keywords

AMINO ACIDS;

ANTI-ANGIOGENIC ACTIVITY; CYCLIC DERIVATIVES; CYCLOPEPTIDES; HETEROCYCLIC MOIETIES; INTEGRINS; LINEAR PEPTIDES; PROOF OF CONCEPT; RGD SEQUENCES;

PEPTIDES;

EID: 84906672172 PISSN: 20416520 EISSN: 20416539 Source Type: Journal
DOI: 10.1039/c4sc00572d Document Type: Article

Times cited : (10)

References (52)

1
- 75949085017
- B. Hughes Nat. Rev. Drug Discovery 2010 9 89
- (2010) Nat. Rev. Drug Discovery , vol.9 , pp. 89
- Hughes, B.¹

2
- 85028101312
- A. Mullard Nat. Rev. Drug Discovery 2011 10 82
- (2011) Nat. Rev. Drug Discovery , vol.10 , pp. 82
- Mullard, A.¹

3
- 84856509534
- A. Mullard Nat. Rev. Drug Discovery 2012 11 91
- (2012) Nat. Rev. Drug Discovery , vol.11 , pp. 91
- Mullard, A.¹

4
- 84873348026
- A. Mullard Nat. Rev. Drug Discovery 2013 11 87
- (2013) Nat. Rev. Drug Discovery , vol.11 , pp. 87
- Mullard, A.¹

5
- 84865491407
- F. Albericio H. G. Kruger Future Med. Chem. 2012 4 1527
- (2012) Future Med. Chem. , vol.4 , pp. 1527
- Albericio, F.¹ Kruger, H.G.²

6
- 0003101732
- ed. C. Basava and G. M. Anantharamaiah, Birkhäuser, Boston, MA
- S. A. Kates, N. A. Sole, F. Albericio and G. Barany, in Peptides: Design, Synthesis and Biological Activity, ed., C. Basava, and, G. M. Anantharamaiah, Birkhäuser, Boston, MA, 1994
- (1994) Peptides: Design, Synthesis and Biological Activity
- Kates, S.A.¹ Sole, N.A.² Albericio, F.³ Barany, G.⁴

7
- 77953133405
- S. Royo-Gracia K. Gaus N. Sewald Future Med. Chem. 2009 1 1289
- (2009) Future Med. Chem. , vol.1 , pp. 1289
- Royo-Gracia, S.¹ Gaus, K.² Sewald, N.³

8
- 80053161003
- C. Mas-Moruno J. G. Beck L. Doedens A. O. Frank L. Marinelli S. Cosconati E. Novellino H. Kessler Angew. Chem., Int. Ed. 2011 50 9496
- (2011) Angew. Chem., Int. Ed. , vol.50 , pp. 9496
- Mas-Moruno, C.¹ Beck, J.G.² Doedens, L.³ Frank, A.O.⁴ Marinelli, L.⁵ Cosconati, S.⁶ Novellino, E.⁷ Kessler, H.⁸

9
- 84862558085
- J. Spiegel C. Mas-Moruno H. Kessler W. D. Lubell J. Org. Chem. 2012 77 5271
- (2012) J. Org. Chem. , vol.77 , pp. 5271
- Spiegel, J.¹ Mas-Moruno, C.² Kessler, H.³ Lubell, W.D.⁴

10
- 84860773239
- M. Marchini M. Mingozzi R. Colombo I. Guzzetti L. Belvisi F. Vasile D. Potenza U. Piarulli D. Arosio C. Gennari Chem.-Eur. J. 2012 18 6195
- (2012) Chem.-Eur. J. , vol.18 , pp. 6195
- Marchini, M.¹ Mingozzi, M.² Colombo, R.³ Guzzetti, I.⁴ Belvisi, L.⁵ Vasile, F.⁶ Potenza, D.⁷ Piarulli, U.⁸ Arosio, D.⁹ Gennari, C.¹⁰

11
- 70849100631
- A. S. M. da Ressurreiçao A. Vidu M. Civera L. Belvisi D. Potenza L. Manzoni S. Ongeri C. Gennari U. Piarulli Chem.-Eur. J. 2009 15 12184
- (2009) Chem.-Eur. J. , vol.15 , pp. 12184
- Da Ressurreiçao, A.S.M.¹ Vidu, A.² Civera, M.³ Belvisi, L.⁴ Potenza, D.⁵ Manzoni, L.⁶ Ongeri, S.⁷ Gennari, C.⁸ Piarulli, U.⁹

12
- 78649529857
- A. O. Frank E. Otto C. Mas-Moruno H. B. Schiller L. Marinelli S. Cosconati A. Bochen D. Vossmeyer G. Zahn R. Stragies E. Novellino H. Kessler Angew. Chem., Int. Ed. 2010 49 9278
- (2010) Angew. Chem., Int. Ed. , vol.49 , pp. 9278
- Frank, A.O.¹ Otto, E.² Mas-Moruno, C.³ Schiller, H.B.⁴ Marinelli, L.⁵ Cosconati, S.⁶ Bochen, A.⁷ Vossmeyer, D.⁸ Zahn, G.⁹ Stragies, R.¹⁰ Novellino, E.¹¹ Kessler, H.¹²

13
- 34250770070
- S. Urman K. Gaus Y. Yang U. Strijowski N. Sewald S. De Pol O. Reiser Angew. Chem., Int. Ed. 2007 46 3976
- (2007) Angew. Chem., Int. Ed. , vol.46 , pp. 3976
- Urman, S.¹ Gaus, K.² Yang, Y.³ Strijowski, U.⁴ Sewald, N.⁵ De Pol, S.⁶ Reiser, O.⁷

14
- 79952741178
- C. Mas-Moruno F. Rechenmacher H. Kessler Anti-Cancer Agents Med. Chem. 2010 10 753
- (2010) Anti-Cancer Agents Med. Chem. , vol.10 , pp. 753
- Mas-Moruno, C.¹ Rechenmacher, F.² Kessler, H.³

15
- 85016509972
- C. Mas-Moruno H. Kessler Methods Princ. Med. Chem. 2013 56 257
- (2013) Methods Princ. Med. Chem. , vol.56 , pp. 257
- Mas-Moruno, C.¹ Kessler, H.²

16
- 84867830537
- C. Scaringi G. Minniti P. Caporello R. M. Enrici Anticancer Res. 2012 32 4213
- (2012) Anticancer Res. , vol.32 , pp. 4213
- Scaringi, C.¹ Minniti, G.² Caporello, P.³ Enrici, R.M.⁴

17
- 84906665252
- For an updated survey of the ongoing clinical trials, search this drug in https://clinicaltrials.gov/

18
- 84860437198
- Z. Hayouka A. Levin M. Hurevich D. E. Shalev A. Loyter G. Gilon A. Friedler Bioorg. Med. Chem. 2012 20 3317
- (2012) Bioorg. Med. Chem. , vol.20 , pp. 3317
- Hayouka, Z.¹ Levin, A.² Hurevich, M.³ Shalev, D.E.⁴ Loyter, A.⁵ Gilon, G.⁶ Friedler, A.⁷

19
- 33847779963
- V. R. Pattabiraman J. L. Stymiest D. J. Derksen N. I. Martin J. C. Vederas Org. Lett. 2007 9 699
- (2007) Org. Lett. , vol.9 , pp. 699
- Pattabiraman, V.R.¹ Stymiest, J.L.² Derksen, D.J.³ Martin, N.I.⁴ Vederas, J.C.⁵

20
- 79960587086
- R. M. J. Liskamp M. J. Rob D. T. S. Rijkers J. A. W. Kruijtezr J. Kemmink ChemBioChem 2011 12 1626
- (2011) ChemBioChem , vol.12 , pp. 1626
- Liskamp, R.M.J.¹ Rob, M.J.² Rijkers, D.T.S.³ Kruijtezr, J.A.W.⁴ Kemmink, J.⁵

21
- 41549147161
- D. Wang M. Lu P. S. Arora Angew. Chem., Int. Ed. 2008 47 1879
- (2008) Angew. Chem., Int. Ed. , vol.47 , pp. 1879
- Wang, D.¹ Lu, M.² Arora, P.S.³

22
- 84889881224
- S. Y. Shim Y.-W. Kim G. L. Verdine Chem. Biol. Drug Des. 2013 82 635
- (2013) Chem. Biol. Drug Des. , vol.82 , pp. 635
- Shim, S.Y.¹ Kim, Y.-W.² Verdine, G.L.³

23
- 84855584802
- G. L. Verdine G. J. Hilinski Methods Enzymol. 2012 503 3
- (2012) Methods Enzymol. , vol.503 , pp. 3
- Verdine, G.L.¹ Hilinski, G.J.²

24
- 48249146974
- S. Cantel I. A. Le Chevalier M. Scrima J. J. Levy R. D. DiMarchi P. Rovero J. A. Halperin A. M. D'Ursi A. M. Papini M. Chorev J. Org. Chem. 2008 73 5663
- (2008) J. Org. Chem. , vol.73 , pp. 5663
- Cantel, S.¹ Le Chevalier, I.A.² Scrima, M.³ Levy, J.J.⁴ Dimarchi, R.D.⁵ Rovero, P.⁶ Halperin, J.A.⁷ D'Ursi, A.M.⁸ Papini, A.M.⁹ Chorev, M.¹⁰

25
- 80055006128
- ed. S. Braese and K. J. Banert, Wiley & Sons Ltd., Chichester, UK
- C. W. Tornoee and M. Meldal, Organic Azides, ed., S. Braese, and, K. J. Banert, Wiley & Sons Ltd., Chichester, UK, 2010, pp. 285-310
- (2010) Organic Azides , pp. 285-310
- Tornoee, C.W.¹ Meldal, M.²

26
- 79959712132
- J. Zhang J. Kemmink D. T. S. Rijkers R. M. J. Liskamp Org. Lett. 2011 13 3438
- (2011) Org. Lett. , vol.13 , pp. 3438
- Zhang, J.¹ Kemmink, J.² Rijkers, D.T.S.³ Liskamp, R.M.J.⁴

27
- 84858972640
- B. Thomas M. Fiore I. Bossu P. Dumy O. Renaudet Beilstein J. Org. Chem. 2012 8 421 427
- (2012) Beilstein J. Org. Chem. , vol.8 , pp. 421-427
- Thomas, B.¹ Fiore, M.² Bossu, I.³ Dumy, P.⁴ Renaudet, O.⁵

28
- 44449109082
- C. T. Walsh E. M. Nolan Proc. Natl. Acad. Sci. U. S. A. 2008 105 5655
- (2008) Proc. Natl. Acad. Sci. U. S. A. , vol.105 , pp. 5655
- Walsh, C.T.¹ Nolan, E.M.²

29
- 0036734093
- R. O. Hynes Nat. Med. 2002 8 918
- (2002) Nat. Med. , vol.8 , pp. 918
- Hynes, R.O.¹

30
- 72949119124
- J. S. Desgrosellier D. A. Cheresh Nature Rev. Cancer 2010 10 9
- (2010) Nature Rev. Cancer , vol.10 , pp. 9
- Desgrosellier, J.S.¹ Cheresh, D.A.²

31
- 70349921610
- M. Hoefling H. Kessler K.-E. Gottschalk Angew. Chem., Int. Ed. 2009 48 6590
- (2009) Angew. Chem., Int. Ed. , vol.48 , pp. 6590
- Hoefling, M.¹ Kessler, H.² Gottschalk, K.-E.³

32
- 67651122837
- M. Schottelius B. Laufer H. Kessler H.-J. Wester Acc. Chem. Res. 2009 42 969
- (2009) Acc. Chem. Res. , vol.42 , pp. 969
- Schottelius, M.¹ Laufer, B.² Kessler, H.³ Wester, H.-J.⁴

33
- 68249117645
- T. Weide A. Modlinger H. Kessler Top. Curr. Chem. 2007 272 1
- (2007) Top. Curr. Chem. , vol.272 , pp. 1
- Weide, T.¹ Modlinger, A.² Kessler, H.³

34
- 77950674729
- L. Auzzas F. Zanardi L. Battistini P. Burreddu P. Carta G. Rassu C. Curti G. Casiraghi Curr. Med. Chem. 2010 17 1255
- (2010) Curr. Med. Chem. , vol.17 , pp. 1255
- Auzzas, L.¹ Zanardi, F.² Battistini, L.³ Burreddu, P.⁴ Carta, P.⁵ Rassu, G.⁶ Curti, C.⁷ Casiraghi, G.⁸

35
- 84874612648
- A. Bochen U. K. Marelli E. Otto D. Pallarola C. Mas-Moruno F. Saverio di Leva H. Boehm J. P. Spatz E. Novellino H. Kessler L. Marinelli J. Med. Chem. 2013 56 1509
- (2013) J. Med. Chem. , vol.56 , pp. 1509
- Bochen, A.¹ Marelli, U.K.² Otto, E.³ Pallarola, D.⁴ Mas-Moruno, C.⁵ Saverio Di Leva, F.⁶ Boehm, H.⁷ Spatz, J.P.⁸ Novellino, E.⁹ Kessler, H.¹⁰ Marinelli, L.¹¹

36
- 79952016219
- M. Aufort M. Gonera J. Le Gal B. Czarny L. Le Clainche R. Thai C. Dugave ChemBioChem 2011 12 583
- (2011) ChemBioChem , vol.12 , pp. 583
- Aufort, M.¹ Gonera, M.² Le Gal, J.³ Czarny, B.⁴ Le Clainche, L.⁵ Thai, R.⁶ Dugave, C.⁷

37
- 84899579958
- S. Neubauer F. Rechenmacher R. Brimioulle F. Saverio Di Leva A. Bochen T. R. Sobahi M. Schottelius E. Novellino C. Mas-Moruno L. Marinelli H. Kessler J. Med. Chem. 2014 57 3410
- (2014) J. Med. Chem. , vol.57 , pp. 3410
- Neubauer, S.¹ Rechenmacher, F.² Brimioulle, R.³ Saverio Di Leva, F.⁴ Bochen, A.⁵ Sobahi, T.R.⁶ Schottelius, M.⁷ Novellino, E.⁸ Mas-Moruno, C.⁹ Marinelli, L.¹⁰ Kessler, H.¹¹

38
- 84862015364
- P.-P. Lv Y.-F. Ma R. Yu H. Yue D.-Z. Ni W. Wei G.-H. Ma Mol. Pharmaceutics 2012 9 1736
- (2012) Mol. Pharmaceutics , vol.9 , pp. 1736
- Lv, P.-P.¹ Ma, Y.-F.² Yu, R.³ Yue, H.⁴ Ni, D.-Z.⁵ Wei, W.⁶ Ma, G.-H.⁷

39
- 84862270302
- F. Bianchini N. Cini A. Trabocchi A. Bottoncetti S. Raspanti E. Vanzi G. Menchi A. Guarna A. Pupi L. Calorini J. Med. Chem. 2012 55 5024
- (2012) J. Med. Chem. , vol.55 , pp. 5024
- Bianchini, F.¹ Cini, N.² Trabocchi, A.³ Bottoncetti, A.⁴ Raspanti, S.⁵ Vanzi, E.⁶ Menchi, G.⁷ Guarna, A.⁸ Pupi, A.⁹ Calorini, L.¹⁰

40
- 77956849861
- K.-T. Yong I. Roy W.-C. Lawb R. Hub Chem. Commun. 2010 46 7136
- (2010) Chem. Commun. , vol.46 , pp. 7136
- Yong, K.-T.¹ Roy, I.² Lawb, W.-C.³ Hub, R.⁴

41
- 84899827304
- J. Simecek J. Notni T. G. Kapp H. Kessler H.-J. Wester Mol. Pharm. 2014 11 1687
- (2014) Mol. Pharm. , vol.11 , pp. 1687
- Simecek, J.¹ Notni, J.² Kapp, T.G.³ Kessler, H.⁴ Wester, H.-J.⁵

42
- 84886001885
- S. Neubauer F. Rechenmacher A. J. Beer F. Curnis K. Pohle C. D'Alessandria H.-J. Wester U. Reuning A. Corti M. Schwaiger H. Kessler Angew. Chem., Int. Ed. 2013 52 11656
- (2013) Angew. Chem., Int. Ed. , vol.52 , pp. 11656
- Neubauer, S.¹ Rechenmacher, F.² Beer, A.J.³ Curnis, F.⁴ Pohle, K.⁵ D'Alessandria, C.⁶ Wester, H.-J.⁷ Reuning, U.⁸ Corti, A.⁹ Schwaiger, M.¹⁰ Kessler, H.¹¹

43
- 35648951171
- R. A. Hughes C. J. Moody Angew. Chem., Int. Ed. 2007 46 7930
- (2007) Angew. Chem., Int. Ed. , vol.46 , pp. 7930
- Hughes, R.A.¹ Moody, C.J.²

44
- 61449199502
- Z. Jin Nat. Prod. Rep. 2009 26 382
- (2009) Nat. Prod. Rep. , vol.26 , pp. 382
- Jin, Z.¹

45
- 0035001744
- B. J. MacLean P. G. Pickup J. Mater. Chem. 2001 11 1357
- (2001) J. Mater. Chem. , vol.11 , pp. 1357
- Maclean, B.J.¹ Pickup, P.G.²

46
- 3843120058
- L. Marinelli K.-E. Gottschalk A. Meyer E. Novellino H. Kessler J. Med. Chem. 2004 47 4166
- (2004) J. Med. Chem. , vol.47 , pp. 4166
- Marinelli, L.¹ Gottschalk, K.-E.² Meyer, A.³ Novellino, E.⁴ Kessler, H.⁵

47
- 77955456458
- J. D. Butler K. C. Coffman K. T. Ziebart M. D. Toney M. J. Kurth Chem.-Eur. J. 2010 16 9002 9005
- (2010) Chem.-Eur. J. , vol.16 , pp. 9002-9005
- Butler, J.D.¹ Coffman, K.C.² Ziebart, K.T.³ Toney, M.D.⁴ Kurth, M.J.⁵

48
- 0035900963
- Y. Singh N. Sokolenko M. J. Kelso L. R. Gahan G. Abbenante D. P. Fairlie J. Am. Chem. Soc. 2001 123 333
- (2001) J. Am. Chem. Soc. , vol.123 , pp. 333
- Singh, Y.¹ Sokolenko, N.² Kelso, M.J.³ Gahan, L.R.⁴ Abbenante, G.⁵ Fairlie, D.P.⁶

49
- 0032847943
- I. G. Stankova G. I. Videnov E. V. Golovinsky G. Jung J. Pept. Sci. 1999 5 392
- (1999) J. Pept. Sci. , vol.5 , pp. 392
- Stankova, I.G.¹ Videnov, G.I.² Golovinsky, E.V.³ Jung, G.⁴

50
- 78651410967
- A. Nefzi J. E. Fenwick Tetrahedron Lett. 2011 52 817
- (2011) Tetrahedron Lett. , vol.52 , pp. 817
- Nefzi, A.¹ Fenwick, J.E.²

51
- 0037493198
- J. O. Nam J. E. Kim H. W. Jeong S. J. Lee B. H. Lee J. Y. Choi R. W. Park J. Y. Park I. S. Kim J. Biol. Chem. 2003 278 25902
- (2003) J. Biol. Chem. , vol.278 , pp. 25902
- Nam, J.O.¹ Kim, J.E.² Jeong, H.W.³ Lee, S.J.⁴ Lee, B.H.⁵ Choi, J.Y.⁶ Park, R.W.⁷ Park, J.Y.⁸ Kim, I.S.⁹

52
- 71849097295
- WO 2012062777 A1 20120518
- Part of these results are covered by a patent: F. Mitjans, J. Adan, C. Calvis, F. Albericio, R. Lavilla and J. Ruiz Rodriguez, PCT Int. Appl., WO 2012062777 A1 20120518, 2012
- (2012) PCT Int. Appl.
- Mitjans, F.¹ Adan, J.² Calvis, C.³ Albericio, F.⁴ Lavilla, R.⁵ Ruiz Rodriguez, J.⁶

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.