Unexpected properties of δ-containing GABAA receptors in response to ligands interacting with the α+ β- Site

Neurochemical Research

Volumn 39, Issue 6, 2014, Pages 1057-1067

  Mirheydari, Pantea ^a   Ramerstorfer, Joachim ^a   Varagic, Zdravko ^a   Scholze, Petra ^a   Wimmer, Laurin ^b   Mihovilovic, Marko M ^b   Sieghart, Werner ^a   Ernst, Margot ^a  

^a MEDICAL UNIVERSITY OF VIENNA   (Austria)

^b VIENNA UNIVERSITY OF TECHNOLOGY   (Austria)

Author keywords

CGS 9895; Extrasynaptic receptor; Null modulators; Positive modulators; Pyrazoloquinolinones; Subunit

Indexed keywords

4 AMINOBUTYRIC ACID A RECEPTOR; ALPHA ADRENERGIC RECEPTOR; BENZODIAZEPINE; BETA ADRENERGIC RECEPTOR; LAU 177; LIGAND; QUINOLINE DERIVATIVE; RECEPTOR SUBTYPE; TRACAZOLATE; UNCLASSIFIED DRUG; 4 AMINOBUTYRIC ACID RECEPTOR STIMULATING AGENT; GABRD PROTEIN, RAT; PROTEIN SUBUNIT;

ALPHA CHAIN; ARTICLE; BETA CHAIN; BINDING SITE; CHEMICAL STRUCTURE; ELECTROPHYSIOLOGICAL PROCEDURES; IN VITRO STUDY; MODULATION; NONHUMAN; POINT MUTATION; PRIORITY JOURNAL; STEREOSPECIFICITY; STIMULATION; VOLTAGE CLAMP TECHNIQUE; AGONISTS; ANIMAL; DOSE RESPONSE; FEMALE; METABOLISM; PHYSIOLOGY; PROTEIN SUBUNIT; RAT; XENOPUS LAEVIS;

ANIMALS; BINDING SITES; DOSE-RESPONSE RELATIONSHIP, DRUG; FEMALE; GABA AGONISTS; LIGANDS; PROTEIN SUBUNITS; RATS; RECEPTORS, GABA-A; XENOPUS LAEVIS;

EID: 84901323683     PISSN: 03643190     EISSN: 15736903     Source Type: Journal    
DOI: 10.1007/s11064-013-1156-3     Document Type: Article

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